Discovery of thioazepinone ligands for Src SH2: From non-specific to specific binding

Bioorganic and Medicinal Chemistry Letters

Volumn 11, Issue 16, 2001, Pages 2127-2131

  Lesuisse, Dominique ^a   Deprez, Pierre ^a   Albert, Eva ^a   Duc, Tran Thien ^a   Sortais, Benoit ^a   Gofflo, Dominique ^a   Jean Baptiste, Véronique ^a   Marquette, Jean Pierre ^a   Schoot, Bernard ^a   Sarubbi, Edoardo ^a   Lange, Gudrun ^a   Broto, Pierre ^a   Mandine, Eliane ^a  

^a SANOFI   (France)

Author keywords

[No Author keywords available]

Indexed keywords

AZEPINE DERIVATIVE; LIGAND; PROTEIN TYROSINE KINASE; PROTEIN TYROSINE KINASE SH2; THIOAZEPINONE; UNCLASSIFIED DRUG;

ARTICLE; BINDING AFFINITY; CRYSTALLIZATION; DRUG DESIGN; DRUG STRUCTURE; DRUG SYNTHESIS; LIGAND BINDING; PROTEIN BINDING;

AZEPINES; BINDING SITES; LIGANDS; MODELS, MOLECULAR; ONCOGENE PROTEIN PP60(V-SRC); SRC HOMOLOGY DOMAINS;

EID: 17944369560     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-894X(01)00386-9     Document Type: Article

References (16)