Synthesis and inhibitory potential towards acetylcholinesterase, butyrylcholinesterase and lipoxygenase of some variably substituted chalcones

Journal of Enzyme Inhibition and Medicinal Chemistry

Volumn 20, Issue 1, 2005, Pages 41-47

  Hasan, Aurangzeb ^a   Khan, Khalid M ^b   Sher, Mohammed ^a   Maharvi, Ghulam M ^b   Nawaz, Sarfraz A ^b   Choudhary, M I ^b   Rahman, Atta Ur ^b   Supuran, Claudiu T ^c  

^a QUAID I AZAM UNIVERSITY   (Pakistan)

^b UNIVERSITY OF KARACHI   (Pakistan)

^c UNIVERSITY OF FLORENCE   (Italy)

Author keywords

Acetylcholinesterase; Butyrylcholinesterase; Chalcones; Lipoxygenase

Indexed keywords

3 (2 HYDROXYPHENYL) 1 PHENYL 2 PROPENE 1 ONE; 3 (3 HYDROXYPHENYL) 1 PHENYL 2 PROPENE 1 ONE; 3 (3 METHOXYPHENYL) 1 (2' HYDROXYPHENYL) 2 PROPENE 1 ONE; 3 (3 METHYLPHENYL) 1 (2' HYDROXY 5' CHLOROPHENYL) 2 PROPENE 1 ONE; 3 (3,4 DIMETHOXYPHENYL) 1 (2' HYDROXYPHENYL) 2 PROPENE 1 ONE; 3 (3,4 DIMETHOXYPHENYL) 1 PHENYL 2 PROPENE 1 ONE; 3 (4 CHLOROPHENYL) 1 (2' HYDROXY 5' CHLOROPHENYL) 2 PROPENE 1 ONE; 3 (4 HYDROXYPHENYL) 1 PHENYL 2 PROPENE 1 ONE; 3 (4 METHOXYPHENYL) 1 (2' HYDROXYPHENYL) 2 PROPENE 1 ONE; 3 (4 METHOXYPHENYL) 1 PHENYL 2 PROPENE 1 ONE; 3 PHENYL 1 (2' HYDROXY 5' CHLOROPHENYL) 2 PROPENE 1 ONE; 3 PHENYL 1 (2' HYDROXYPHENYL) 2 PROPENE 1 ONE; ACETOPHENONE DERIVATIVE; ACETYLCHOLINESTERASE; BENZALDEHYDE DERIVATIVE; CHALCONE DERIVATIVE; CHOLINESTERASE; CHOLINESTERASE INHIBITOR; LIPOXYGENASE; LIPOXYGENASE INHIBITOR; UNCLASSIFIED DRUG;

ARTICLE; CHOLINESTERASE INHIBITION; CONCENTRATION RESPONSE; CONTROLLED STUDY; DRUG MECHANISM; DRUG STRUCTURE; DRUG SYNTHESIS; ENZYME INHIBITION; PRIORITY JOURNAL; STRUCTURE ANALYSIS;

ACETYLCHOLINESTERASE; ANIMALS; BUTYRYLCHOLINESTERASE; CHALCONES; CHOLINESTERASE INHIBITORS; ELECTROPHORUS; HORSES; INHIBITORY CONCENTRATION 50; LIPOXYGENASE; LIPOXYGENASE INHIBITORS; MOLECULAR STRUCTURE;

EID: 17144362548     PISSN: 14756366     EISSN: None     Source Type: Journal    
DOI: 10.1080/14756360400015231     Document Type: Article

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