Effects of TAK-802, a novel acetylcholinesterase inhibitor, on distension-induced rhythmic bladder contractions in rats and guinea pigs

European Journal of Pharmacology

Volumn 485, Issue 1-3, 2004, Pages 299-305

  Nagabukuro, Hiroshi ^a   Okanishi, Satoshi ^a   Imai, Shigemitsu ^a   Ishichi, Yuji ^a   Ishihara, Yuji ^a   Doi, Takayuki ^a  

^a TAKEDA PHARMACEUTICAL COMPANY LIMITED   (Japan)

Author keywords

(Guinea pig); (Rat); Acetylcholinesterase inhibitor; Bladder; Micturition; TAK 802

Indexed keywords

8 [3 [1 [(3 FLUOROPHENYL)METHYL] 4 PIPERIDINYL] 1 OXOPROPYL] 1,2,5,6 TETRAHYDRO 4H PYRROLO[3,2,1 IJ]QUINOLIN 4 ONE; ACETYLCHOLINE; ACETYLCHOLINESTERASE; ATROPINE; BETHANECHOL; CHOLINESTERASE; CHOLINESTERASE INHIBITOR; DISTIGMINE; MUSCARINIC AGENT; NEOSTIGMINE; NICOTINIC AGENT; TAK 802; UNCLASSIFIED DRUG; URETHAN;

ACETYLCHOLINE RELEASE; ANESTHESIA; ANIMAL EXPERIMENT; ARTICLE; BLADDER CONTRACTION; BLADDER DISTENSION; CONTROLLED STUDY; DOSE RESPONSE; DRUG ACTIVITY; DRUG DETERMINATION; DRUG EFFECT; DRUG EFFICACY; DRUG MECHANISM; DRUG POTENCY; DRUG SCREENING; DRUG SELECTIVITY; ENZYME ACTIVITY; ENZYME INHIBITION; ERYTHROCYTE; GUINEA PIG; IC 50; INHIBITION KINETICS; MALE; MEASUREMENT; NERVE CONDUCTION; NONHUMAN; PRIORITY JOURNAL; RAT; REFLEX;

EID: 1642497566     PISSN: 00142999     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.ejphar.2003.11.045     Document Type: Article

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