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Bioorganic and Medicinal Chemistry Letters

Volumn 15, Issue 6, 2005, Pages 1743-1747

Further studies on ethenyl and ethynyl-4-phenylamino-3- quinolinecarbonitriles: Identification of a subnanomolar Src kinase inhibitor

(5) Sosa, Ana Carolina Barrios a,b Boschelli, Diane H a Wu, Biqi a Wang, Yan a Golas, Jennifer M a

a WYETH RESEARCH (United States)

b Roche Carolina (United States)

Author keywords

3 Quinolinecarbonitriles; Kinase; Src

Indexed keywords

ENZYME INHIBITOR; ETHENYL 4 PHENYLAMINO 3 QUINOLINECARBONITRILE DERIVATIVE; ETHYNYL 4 PHENYLAMINO 3 QUINOLINECARBONITRILE DERIVATIVE; OXIDE; PROTEIN TYROSINE KINASE; PROTEIN TYROSINE KINASE INHIBITOR; PYRIDINE DERIVATIVE; UNCLASSIFIED DRUG;

ANIMAL EXPERIMENT; ARTICLE; CONTROLLED STUDY; DRUG IDENTIFICATION; DRUG POTENCY; DRUG SYNTHESIS; ENZYME INHIBITION; MOUSE; NONHUMAN;

EID: 14644413418 PISSN: 0960894X EISSN: None Source Type: Journal
DOI: 10.1016/j.bmcl.2005.01.004 Document Type: Article

Times cited : (23)

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