Synthesis and in vitro antitrypanosomal activity of novel Nifurtimox analogues

Bioorganic and Medicinal Chemistry Letters

Volumn 15, Issue 5, 2005, Pages 1417-1421

  Pozas, Rocío ^a   Carballo, Javier ^a   Castro, Clementina ^a   Rubio, Julieta ^a  

^a UNIVERSIDAD NACIONAL AUTÓNOMA DE MÉXICO   (Mexico)

Author keywords

Antiparasites; Antitrypanosomal activity; Nifurtimox analogues; Trypanosoma cruzi

Indexed keywords

ANTITRYPANOSOMAL AGENT; BENZYL DERIVATIVE; FURAN; N (4 CHLORO 2 BENZOTHIAZOLE) 3 (5 NITRO 2 FURYL)PROPENAMIDE; N (4 CHLOROBENZYL) 3 (5 NITRO 2 FURYL)PROPENAMIDE; N BENZYL 3 (2 FURYL)PROPENAMIDE; N BENZYL 3 (5 NITRO 2 FURYL)PROPENAMIDE; N BENZYL 3 (5 NITROTHIOPHEN 2 YL)PROPENAMIDE; N BENZYL 3 (THIOPHEN 2 YL)PROPENAMIDE; N ISOBUTYL 3 (5 NITRO 2 FURYL)PROPENAMIDE; N PIPERONYL 3 (5 NITRO 2 FURYL)PROPENAMIDE; NIFURTIMOX; NITROFURAN DERIVATIVE; NITROREDUCTASE; UNCLASSIFIED DRUG;

ANTIPROTOZOAL ACTIVITY; ARTICLE; CELL DEATH; CONTROLLED STUDY; DRUG SYNTHESIS; EPIMASTIGOTE; NONHUMAN; TRYPANOSOMA CRUZI;

TRIXIS; TRYPANOSOMA; TRYPANOSOMA CRUZI;

EID: 13944280211     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2005.01.002     Document Type: Article

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