Amino acid conjugates as κ opioid receptor agonists

Bioorganic and Medicinal Chemistry Letters

Volumn 15, Issue 5, 2005, Pages 1279-1282

  Kumar, Virendra ^a   Guo, Deqi ^a   Daubert, Jeffrey D ^a   Cassel, Joel A ^a   DeHaven, Robert N ^a   Mansson, Erik ^a   DeHaven Hudkins, Diane L ^a   Maycock, Alan L ^a  

^a ADOLOR CORPORATION   (United States)

Author keywords

Amino acid conjugates; Kappa opioid receptor agonists

Indexed keywords

ACETAMIDE DERIVATIVE; AMINO ACID DERIVATIVE; KAPPA OPIATE RECEPTOR; KAPPA OPIATE RECEPTOR AGONIST; OPIATE RECEPTOR;

AMINO ACID SUBSTITUTION; ARTICLE; DRUG CONJUGATION; DRUG POTENCY; DRUG RECEPTOR BINDING; DRUG SELECTIVITY; DRUG STRUCTURE; DRUG SYNTHESIS; IN VITRO STUDY; RECEPTOR AFFINITY; STRUCTURE ANALYSIS;

EID: 13944261906     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2005.01.038     Document Type: Article

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