메뉴 건너뛰기




Volumn 26, Issue 2, 2005, Pages 166-170

Modulation of P-glycoprotein function by amlodipine derivatives in brain microvessel endothelial cells of rats

Author keywords

Amlodipine derivatives; Blood brain barrier; CJX1; CJX2; P glycoprotein; Vascular endothelium; Verapamil

Indexed keywords

AMLODIPINE; CJX 1; CJX 2; GLYCOPROTEIN P; RHODAMINE 123; UNCLASSIFIED DRUG;

EID: 13444274764     PISSN: 16714083     EISSN: None     Source Type: Journal    
DOI: 10.1111/j.1745-7254.2005.00528.x     Document Type: Article
Times cited : (9)

References (18)
  • 1
    • 0029954843 scopus 로고    scopus 로고
    • P-glycoprotein-a mediator of multidrug resistance in tumour cells
    • Germann UA. P-glycoprotein-a mediator of multidrug resistance in tumour cells. Eur J Cancer 1996; 32A: 927-44.
    • (1996) Eur J Cancer , vol.32 A , pp. 927-944
    • Germann, U.A.1
  • 2
    • 0027218689 scopus 로고
    • Biochemistry of multidrug resistance mediated by the multidrug transporter
    • Gottesman MM, Pastan I. Biochemistry of multidrug resistance mediated by the multidrug transporter. Annu Rev Biochem 1993; 62: 385-427.
    • (1993) Annu Rev Biochem , vol.62 , pp. 385-427
    • Gottesman, M.M.1    Pastan, I.2
  • 3
    • 0028249115 scopus 로고
    • The MDR superfamily of genes and its biological implications
    • Childs S, Ling V. The MDR superfamily of genes and its biological implications. Important Adv Oncol 1994; 21-36.
    • (1994) Important Adv Oncol , pp. 21-36
    • Childs, S.1    Ling, V.2
  • 4
    • 2342436512 scopus 로고    scopus 로고
    • PET studies on P-glycoprotein function in the blood-brain barrier: How it affects uptake and binding of drugs within the CNS
    • Elsinga PH, Hendrikse NH, Bart J, Vaalburg W, van Waarde A. PET studies on P-glycoprotein function in the blood-brain barrier: how it affects uptake and binding of drugs within the CNS. Curr Pharm Des 2004; 10: 1493-503.
    • (2004) Curr Pharm des , vol.10 , pp. 1493-1503
    • Elsinga, P.H.1    Hendrikse, N.H.2    Bart, J.3    Vaalburg, W.4    Van Waarde, A.5
  • 5
    • 0142105939 scopus 로고    scopus 로고
    • In vivo saturation of the transport of vinblastine and colchicine by P-glycoprotein at the rat blood-brain barrier
    • Cisternino S, Rousselle C, Debray M, Scherrmann JM. In vivo saturation of the transport of vinblastine and colchicine by P-glycoprotein at the rat blood-brain barrier. Pharm Res 2003; 20: 1607-11.
    • (2003) Pharm Res , vol.20 , pp. 1607-1611
    • Cisternino, S.1    Rousselle, C.2    Debray, M.3    Scherrmann, J.M.4
  • 6
    • 0037036215 scopus 로고    scopus 로고
    • Effect of endotoxin on doxorubicin transport across blood-brain barrier and P-glycoprotein function in mice
    • Zhao YL, Du J, Kanazawa H, Sugawara A, Takagi K, Kitaichi K, et al. Effect of endotoxin on doxorubicin transport across blood-brain barrier and P-glycoprotein function in mice. Eur J Pharmacol 2002; 445: 115-23.
    • (2002) Eur J Pharmacol , vol.445 , pp. 115-123
    • Zhao, Y.L.1    Du, J.2    Kanazawa, H.3    Sugawara, A.4    Takagi, K.5    Kitaichi, K.6
  • 7
    • 0027998226 scopus 로고
    • In vivo evidence for ATP-dependent and P-glycoprotein-mediated transport of cyclosporin a at the blood-brain barrier
    • Sakata A, Tamai I, Kawazu K, Deguchi Y, Ohnishi T, Saheki A, et al. In vivo evidence for ATP-dependent and P-glycoprotein-mediated transport of cyclosporin A at the blood-brain barrier. Biochem Pharmacol 1994; 48: 1989-92.
    • (1994) Biochem Pharmacol , vol.48 , pp. 1989-1992
    • Sakata, A.1    Tamai, I.2    Kawazu, K.3    Deguchi, Y.4    Ohnishi, T.5    Saheki, A.6
  • 8
    • 0023892070 scopus 로고
    • Modification of cytotoxic drug resistance by nonimmuno-suppressive cyclosporins
    • Twentyman PR. Modification of cytotoxic drug resistance by nonimmuno-suppressive cyclosporins. Br J Cancer 1988; 57: 254-8.
    • (1988) Br J Cancer , vol.57 , pp. 254-258
    • Twentyman, P.R.1
  • 9
    • 0033053573 scopus 로고    scopus 로고
    • Combinations of P-glycoprotein blockers, verapamil, PSC833, and cremophor act differently on the multidrug resistance associated protein (MRP) and on P-glycoprotein (Pgp)
    • Aszalos A, Thompson K, Yin JJ, Ross DD. Combinations of P-glycoprotein blockers, verapamil, PSC833, and cremophor act differently on the multidrug resistance associated protein (MRP) and on P-glycoprotein (Pgp). Anticancer Res 1999; 19: 1053-64.
    • (1999) Anticancer Res , vol.19 , pp. 1053-1064
    • Aszalos, A.1    Thompson, K.2    Yin, J.J.3    Ross, D.D.4
  • 10
    • 10744219744 scopus 로고    scopus 로고
    • Effect of an angiotensin II type 1 receptor blocker, valsartan, on neurohumoral factors in patients with hypertension: Comparison with a long-acting calcium channel antagonist, amlodipine
    • Ohbayashi Y, Tsutamoto T, Sakaguchi T, Tanaka T, Kanamori T, Yokohama H, et al. Effect of an angiotensin II type 1 receptor blocker, valsartan, on neurohumoral factors in patients with hypertension: comparison with a long-acting calcium channel antagonist, amlodipine. J Cardiovasc Pharmacol 2003; 42 Suppl 1: S71-4.
    • (2003) J Cardiovasc Pharmacol , vol.42 , Issue.SUPPL. 1
    • Ohbayashi, Y.1    Tsutamoto, T.2    Sakaguchi, T.3    Tanaka, T.4    Kanamori, T.5    Yokohama, H.6
  • 11
    • 0033636618 scopus 로고    scopus 로고
    • Inhibitory potencies of 1,4-dihydropyridine calcium antagonists to P-glycoprotein-mediated transport: Comparison with the effects on CYP3A4
    • Katoh M, Nakajima, M, Yamazaki H, Yokoi T. Inhibitory potencies of 1,4-dihydropyridine calcium antagonists to P-glycoprotein-mediated transport: comparison with the effects on CYP3A4. Pharm Res 2000; 17: 1189-97.
    • (2000) Pharm Res , vol.17 , pp. 1189-1197
    • Katoh, M.1    Nakajima, M.2    Yamazaki, H.3    Yokoi, T.4
  • 12
    • 0026793292 scopus 로고
    • Development and characterization of a rat brain capillary endothelial culture: Towards an in vitro blood-brain barrier
    • Abbott NJ, Hughes CC, Revest PA, Greenwood J. Development and characterization of a rat brain capillary endothelial culture: towards an in vitro blood-brain barrier. J Cell Sci 1992; 103: 23-37.
    • (1992) J Cell Sci , vol.103 , pp. 23-37
    • Abbott, N.J.1    Hughes, C.C.2    Revest, P.A.3    Greenwood, J.4
  • 13
    • 0030604062 scopus 로고    scopus 로고
    • Use of rhodamine 123 to examine the functional activity of P-glycoprotein in primary cultured brain microvessel endothelial cell monolayers
    • Fontaine M, Elmquist WF, Miller DW. Use of rhodamine 123 to examine the functional activity of P-glycoprotein in primary cultured brain microvessel endothelial cell monolayers. Life Sci 1996; 59: 1521-31.
    • (1996) Life Sci , vol.59 , pp. 1521-1531
    • Fontaine, M.1    Elmquist, W.F.2    Miller, D.W.3
  • 14
    • 0036195976 scopus 로고    scopus 로고
    • Microplate screening of the differential effects of test agents on Hoechst 33342, rhodamine 123, and rhodamine 6G accumulation in breast cancer cells that overexpress P-glycoprotein
    • Sarver JG, Klis WA, Byers JP, Erhardt PW. Microplate screening of the differential effects of test agents on Hoechst 33342, rhodamine 123, and rhodamine 6G accumulation in breast cancer cells that overexpress P-glycoprotein. J Biomol Screen 2002; 7: 29-34.
    • (2002) J Biomol Screen , vol.7 , pp. 29-34
    • Sarver, J.G.1    Klis, W.A.2    Byers, J.P.3    Erhardt, P.W.4
  • 15
    • 0030823912 scopus 로고    scopus 로고
    • P-glycoprotein is strongly expressed in the luminal membranes of the endothelium of blood vessels in the brain
    • Beaulieu E, Demeule M, Ghitescu L, Beliveau R. P-glycoprotein is strongly expressed in the luminal membranes of the endothelium of blood vessels in the brain. Biochem J 1997; 326 ( Pt 2): 539-44.
    • (1997) Biochem J , vol.326 , Issue.PART 2 , pp. 539-544
    • Beaulieu, E.1    Demeule, M.2    Ghitescu, L.3    Beliveau, R.4
  • 16
    • 0242557605 scopus 로고    scopus 로고
    • Effect of E6, a novel calmodulin inhibitor, on activity of P-glycoprotein in purified primary cultured rat brain microvessel endothelial cells
    • Zhu HJ, Liu GQ. Effect of E6, a novel calmodulin inhibitor, on activity of P-glycoprotein in purified primary cultured rat brain microvessel endothelial cells. Acta Pharmacol Sin 2003; 24: 1143-9.
    • (2003) Acta Pharmacol Sin , vol.24 , pp. 1143-1149
    • Zhu, H.J.1    Liu, G.Q.2
  • 17
    • 0036299716 scopus 로고    scopus 로고
    • Effects of various principles from Chinese herbal medicine on rhodamine123 accumulation in brain capillary endothelial cells
    • He L, Liu GQ. Effects of various principles from Chinese herbal medicine on rhodamine123 accumulation in brain capillary endothelial cells. Acta Pharmacol Sin 2002; 23: 591-6.
    • (2002) Acta Pharmacol Sin , vol.23 , pp. 591-596
    • He, L.1    Liu, G.Q.2
  • 18
    • 0035371207 scopus 로고    scopus 로고
    • Modulation by LY335979 of P-glycoprotein function in multidrug-resistant cell lines and human natural killer cells
    • Green LJ, Marder P, Slapak CA. Modulation by LY335979 of P-glycoprotein function in multidrug-resistant cell lines and human natural killer cells. Biochem Pharmacol 2001; 61: 1393-9.
    • (2001) Biochem Pharmacol , vol.61 , pp. 1393-1399
    • Green, L.J.1    Marder, P.2    Slapak, C.A.3


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.