Practical synthesis of DQ-113, a new quinolone antibacterial agent, by using the intramolecular Horner-Wadsworth-Emmons reaction

Heterocycles

Volumn 63, Issue 3, 2004, Pages 699-706

  Inagaki, Hiroaki ^a   Takeda, Toshiyaki ^a   Miyauchi, Rie N ^a   Kawakami, Katsuhiro ^a   Takahashi, Hisashi ^a   Takemura, Makoto ^a  

^a DAIICHI SANKYO CO   (Japan)

Author keywords

[No Author keywords available]

Indexed keywords

5 AMINO 7 [4 (1 AMINOCYCLOPROP 1 YL) 3 FLUOROPYRROLIDIN 1 YL] 6 FLUORO 1 (2 FLUOROCYCLOPROPAN 1 YL) 1,4 DIHYDRO 8 METHYL 4 OXOQUINOLINE 3 CARBOXYLIC ACID; DQ 113; QUINOLINE DERIVED ANTIINFECTIVE AGENT; UNCLASSIFIED DRUG;

ARTICLE; DRUG STRUCTURE; DRUG SYNTHESIS; GRAM POSITIVE BACTERIUM; HORNER WADSWORTH EMMONS REACTION; LOW TEMPERATURE; REACTION ANALYSIS; STRUCTURE ANALYSIS; SUBSTITUTION REACTION; TEMPERATURE DEPENDENCE;

EID: 1342331991     PISSN: 03855414     EISSN: None     Source Type: Journal    
DOI: 10.3987/COM-03-9972     Document Type: Article

References (5)

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