A series of heterocyclic inhibitors of phenylalanyl-tRNA synthetases with antibacterial activity

Bioorganic and Medicinal Chemistry Letters

Volumn 14, Issue 5, 2004, Pages 1343-1346

  Yu, Xiang Y ^a   Finn, John ^a   Hill, Jason M ^a   Wang, Zhong G ^a   Keith, Dennis ^a   Silverman, Jared ^a   Oliver, N ^a  

^a CUBIST PHARMACEUTICALS INC   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

ANTIINFECTIVE AGENT; ENZYME INHIBITOR; HETEROCYCLIC COMPOUND; PHENYLALANINE TRANSFER RNA LIGASE; PHENYLALANINE TRANSFER RNA LIGASE INHIBITOR; UNCLASSIFIED DRUG;

ANTIBACTERIAL ACTIVITY; ARTICLE; CRYSTAL STRUCTURE; DRUG SCREENING; DRUG SYNTHESIS; ENZYME INHIBITION; IC 50; MINIMUM INHIBITORY CONCENTRATION; NONHUMAN; STAPHYLOCOCCUS AUREUS;

STAPHYLOCOCCUS; STAPHYLOCOCCUS AUREUS;

EID: 1242316373     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2003.11.082     Document Type: Article

References (6)

1. Yu, X. Y.; Finn, J.; Hill, J. M.; Wang, Z. G.; Keith, D.; Silverman, J.; Oliver, N. Bioorg. Med. Chem. Lett. 2004, 14, preceding paper in this issue. doi: 10.1016/j.bmcl.2003.11.081.
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