Fluorine-substitution in cholesteryl ester transfer protein inhibitors (CETP-inhibitors) - Biology, chemistry, SAR, and properties

Chimia

Volumn 58, Issue 3, 2004, Pages 123-127

  Paulsen, Holger ^a   Schmeck, Carsten ^a   Brandes, Arndt ^a   Schmidt, Gunter ^a   Stoltefuss, Jürgen ^a   Wirtz, Stephan N ^a   Lögers, Michael ^a   Naab, Paul ^a   Bremm, Klaus Dieter ^a   Bischoff, Hilmar ^a   Schmidt, Delf ^a   Zaiss, Siegfried ^a   Antons, Stefan ^a  

^a BAYER AG   (Germany)

Author keywords

Cholesteryl ester transfer protein; Domino reaction; Hantzsch reaction HDL C elevation; Oxazaborolidine reduction

Indexed keywords

CHOLESTEROL ESTER TRANSFER PROTEIN; FLUORINE DERIVATIVE; HIGH DENSITY LIPOPROTEIN CHOLESTEROL; LOW DENSITY LIPOPROTEIN CHOLESTEROL;

ATHEROGENESIS; CONFERENCE PAPER; DRUG ACTIVITY; DRUG EFFECT; DRUG INHIBITION; DRUG SCREENING; DRUG SYNTHESIS; STRUCTURE ACTIVITY RELATION;

EID: 11144356393     PISSN: 00094293     EISSN: None     Source Type: Journal    
DOI: 10.2533/000942904777678082     Document Type: Conference Paper

References (10)

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