Discovery of a novel, potent and selective human β 3- adrenergic receptor agonist

Bioorganic and Medicinal Chemistry Letters

Volumn 15, Issue 2, 2005, Pages 251-254

  Nakajima, Yutaka ^a   Hamashima, Hitoshi ^a   Washizuka, Ken Ichi ^a   Tomishima, Yasuyo ^a   Ohtake, Hiroaki ^a   Imamura, Emiko ^a   Miura, Toshiko ^a   Kayakiri, Hiroshi ^a   Kato, Masayuki ^a  

^a ASTELLAS PHARMA INC   (Japan)

Author keywords

3 Adrenergic receptor agonist

Indexed keywords

BETA 3 ADRENERGIC RECEPTOR STIMULATING AGENT; BETA ADRENERGIC RECEPTOR STIMULATING AGENT;

ARTICLE; CONTROLLED STUDY; DOG; DRUG BIOAVAILABILITY; DRUG IDENTIFICATION; DRUG POTENCY; DRUG STRUCTURE; DRUG SYNTHESIS; EXPERIMENTAL MODEL; NONHUMAN; STRUCTURE ACTIVITY RELATION; STRUCTURE ANALYSIS;

ADRENERGIC BETA-AGONISTS; ANIMALS; CHO CELLS; CRICETINAE; HUMANS; MODELS, CHEMICAL; RECEPTORS, ADRENERGIC, BETA-3; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 10644240662     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2004.11.001     Document Type: Article

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