Agonist induction, conformational selection, and mutant receptors

FEBS Letters

Volumn 556, Issue 1-3, 2004, Pages 13-18

  Giraldo, Jesús ^a  

^a INSTITUT DE NEUROCIÈNCIES   (Spain)

Author keywords

Agonist induction; Conformational selection; G protein coupled receptor; Multiple state; Mutant receptor; Signal transduction

Indexed keywords

LIGAND; RECEPTOR;

AGONIST; ARTICLE; BINDING AFFINITY; CONCENTRATION (PARAMETERS); CONFORMATION; CORRELATION ANALYSIS; DRUG EFFECT; DRUG MECHANISM; DRUG POTENCY; EQUILIBRIUM CONSTANT; MOLECULAR MECHANICS; MUTANT; MUTATION; PRIORITY JOURNAL; PROCESS MODEL; PROTEIN CONFORMATION; PROTEIN INTERACTION; QUANTITATIVE ANALYSIS; RECEPTOR BINDING; SIMULATION; THERMODYNAMICS; WILD TYPE;

EID: 0347985770     PISSN: 00145793     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0014-5793(03)01404-2     Document Type: Article

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