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Volumn 68, Issue 10-13, 2003, Pages 995-1003

Regulation of gene expression by PRA-910, a novel progesterone receptor modulator, in T47D cells

Author keywords

Affymetrix GeneChip ; PRA 910; Progesterone; Progesterone receptor; Progesterone receptor modulator; Steroid

Indexed keywords

MIFEPRISTONE; P4; PRA 910; PROGESTERONE; PROGESTERONE RECEPTOR MODULATOR; UNCLASSIFIED DRUG;

EID: 0345735761     PISSN: 0039128X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0039-128X(03)00119-3     Document Type: Conference Paper
Times cited : (10)

References (29)
  • 1
    • 0025239785 scopus 로고
    • Two distinct estrogen-regulated promoters generate transcripts encoding two functionally different human progesterone receptor forms a and B
    • Kastner P., Krust A., Turcotte B., Stropp U., Tora L., Gronemeyer H.et al. Two distinct estrogen-regulated promoters generate transcripts encoding two functionally different human progesterone receptor forms A and B. EMBO J. 9:1990;1603-1614.
    • (1990) EMBO J. , vol.9 , pp. 1603-1614
    • Kastner, P.1    Krust, A.2    Turcotte, B.3    Stropp, U.4    Tora, L.5    Gronemeyer, H.6
  • 3
    • 0034622974 scopus 로고    scopus 로고
    • Subgroup of reproductive functions of progesterone mediated by progesterone receptor-B isoform
    • Mulac-Jericevic B., Mullinax R.A., DeMayo F.J., Lydon J.P., Conneely O.M. Subgroup of reproductive functions of progesterone mediated by progesterone receptor-B isoform. Science. 289:2000;1751-1754.
    • (2000) Science , vol.289 , pp. 1751-1754
    • Mulac-Jericevic, B.1    Mullinax, R.A.2    Demayo, F.J.3    Lydon, J.P.4    Conneely, O.M.5
  • 4
    • 0036745890 scopus 로고    scopus 로고
    • Progesterone regulation of reproductive function through functionally distinct progesterone receptor isoforms
    • Conneely O.M., Jericevic B.M. Progesterone regulation of reproductive function through functionally distinct progesterone receptor isoforms. Rev. Endocr. Metab. Disord. 3:2002;201-209.
    • (2002) Rev. Endocr. Metab. Disord. , vol.3 , pp. 201-209
    • Conneely, O.M.1    Jericevic, B.M.2
  • 6
    • 0037179638 scopus 로고    scopus 로고
    • 6-Aryl-1,4-dihydro-benzo[d][1,3]oxazin-2-ones: A novel class of potent, selective, and orally active nonsteroidal progesterone receptor antagonists
    • Zhang P., Terefenko E.A., Fensome A., Wrobel J., Winneker R., Lundeen S.et al. 6-Aryl-1,4-dihydro-benzo[d][1,3]oxazin-2-ones: a novel class of potent, selective, and orally active nonsteroidal progesterone receptor antagonists. J. Med. Chem. 45:2002;4379-4382.
    • (2002) J. Med. Chem. , vol.45 , pp. 4379-4382
    • Zhang, P.1    Terefenko, E.A.2    Fensome, A.3    Wrobel, J.4    Winneker, R.5    Lundeen, S.6
  • 7
    • 0033673829 scopus 로고    scopus 로고
    • In vitro characterization of trimegestone: A potent and selective progestin
    • Zhang Z., Lundeen S.G., Zhu Y., Carver J.M., Winneker R.C. In vitro characterization of trimegestone: a potent and selective progestin. Steroids. 65:2000;637-643.
    • (2000) Steroids , vol.65 , pp. 637-643
    • Zhang, Z.1    Lundeen, S.G.2    Zhu, Y.3    Carver, J.M.4    Winneker, R.C.5
  • 8
    • 0034822884 scopus 로고    scopus 로고
    • Rat uterine complement C3 expression as a model for progesterone receptor modulators: Characterization of the new progestin trimegestone
    • Lundeen S.G., Zhang Z., Zhu Y., Carver J.M., Winneker R.C. Rat uterine complement C3 expression as a model for progesterone receptor modulators: characterization of the new progestin trimegestone. J. Steroid Biochem. Mol. Biol. 78:2001;137-143.
    • (2001) J. Steroid Biochem. Mol. Biol. , vol.78 , pp. 137-143
    • Lundeen, S.G.1    Zhang, Z.2    Zhu, Y.3    Carver, J.M.4    Winneker, R.C.5
  • 10
    • 0037085303 scopus 로고    scopus 로고
    • Differential gene regulation by the two progesterone receptor isoforms in human breast cancer cells
    • Richer J.K., Jacobsen B.M., Manning N.G., Abel M.G., Wolf D.M., Horwitz K.B. Differential gene regulation by the two progesterone receptor isoforms in human breast cancer cells. J. Biol. Chem. 277:2002;5209-5218.
    • (2002) J. Biol. Chem. , vol.277 , pp. 5209-5218
    • Richer, J.K.1    Jacobsen, B.M.2    Manning, N.G.3    Abel, M.G.4    Wolf, D.M.5    Horwitz, K.B.6
  • 11
    • 0025988519 scopus 로고
    • Progestin regulation of alkaline phosphatase in the human breast cancer cell line T47D
    • Di Lorenzo D., Albertini A., Zava D. Progestin regulation of alkaline phosphatase in the human breast cancer cell line T47D. Cancer Res. 51:1991;4470-4475.
    • (1991) Cancer Res. , vol.51 , pp. 4470-4475
    • Di Lorenzo, D.1    Albertini, A.2    Zava, D.3
  • 12
    • 0027201658 scopus 로고
    • Progesterone induced expression of alkaline phosphatase is associated with a secretory phenotype in T47D breast cancer cells
    • Di Lorenzo D., Gianni M., Savoldi G.F., Ferrari F., Albertini A., Garattini E. Progesterone induced expression of alkaline phosphatase is associated with a secretory phenotype in T47D breast cancer cells. Biochem. Biophys. Res. Commun. 192:1993;1077-1082.
    • (1993) Biochem. Biophys. Res. Commun. , vol.192 , pp. 1077-1082
    • Di Lorenzo, D.1    Gianni, M.2    Savoldi, G.F.3    Ferrari, F.4    Albertini, A.5    Garattini, E.6
  • 13
    • 0030910244 scopus 로고    scopus 로고
    • Novel progesterone target genes identified by an improved differential display technique suggest that progestin-induced growth inhibition of breast cancer cells coincides with enhancement of differentiation
    • Kester H.A., van der Leede B.M., van der Saag P.T., van der Burg B. Novel progesterone target genes identified by an improved differential display technique suggest that progestin-induced growth inhibition of breast cancer cells coincides with enhancement of differentiation. J. Biol. Chem. 272:1997;16637-16643.
    • (1997) J. Biol. Chem. , vol.272 , pp. 16637-16643
    • Kester, H.A.1    Van Der Leede, B.M.2    Van Der Saag, P.T.3    Van Der Burg, B.4
  • 14
    • 0033582334 scopus 로고    scopus 로고
    • Claudin multigene family encoding four-transmembrane domain protein components of tight junction strands
    • Morita K., Furuse M., Fujimoto K., Tsukita S. Claudin multigene family encoding four-transmembrane domain protein components of tight junction strands. Proc. Natl. Acad. Sci. U.S.A. 96:1999;511-516.
    • (1999) Proc. Natl. Acad. Sci. U.S.A. , vol.96 , pp. 511-516
    • Morita, K.1    Furuse, M.2    Fujimoto, K.3    Tsukita, S.4
  • 15
    • 0034599992 scopus 로고    scopus 로고
    • Pores in the wall: Claudins constitute tight junction strands containing aqueous pores
    • Tsukida S., Furuse M. Pores in the wall: claudins constitute tight junction strands containing aqueous pores. J. Cell Biol. 149:2000;13-16.
    • (2000) J. Cell Biol. , vol.149 , pp. 13-16
    • Tsukida, S.1    Furuse, M.2
  • 16
    • 0027487161 scopus 로고
    • Molecular cloning and primary structure of Man9-mannosidase from human kidney
    • Bause E., Bieberich E., Rolfs A., Volker C., Schmidt B. Molecular cloning and primary structure of Man9-mannosidase from human kidney. Eur. J. Biochem. 217:1993;535-540.
    • (1993) Eur. J. Biochem. , vol.217 , pp. 535-540
    • Bause, E.1    Bieberich, E.2    Rolfs, A.3    Volker, C.4    Schmidt, B.5
  • 17
    • 0032077354 scopus 로고    scopus 로고
    • Phosphatidylinositol transfer proteins: A requirement in signal transduction and vesicle traffic
    • Cockcroft S. Phosphatidylinositol transfer proteins: a requirement in signal transduction and vesicle traffic. BioEssays. 20:1998;423-432.
    • (1998) BioEssays , vol.20 , pp. 423-432
    • Cockcroft, S.1
  • 18
    • 0026559680 scopus 로고
    • Hormone-induced progesterone receptor phosphorylation consists of sequential DNA-independent and DNA-dependent stages: Analysis with zinc finger mutants and the progesterone antagonist ZK98299
    • Takimoto G.S., Tasset D.M., Eppert A.C., Horwitz K.B. Hormone-induced progesterone receptor phosphorylation consists of sequential DNA-independent and DNA-dependent stages: analysis with zinc finger mutants and the progesterone antagonist ZK98299. Proc. Natl. Acad. Sci. U.S.A. 89:1992;3050-3054.
    • (1992) Proc. Natl. Acad. Sci. U.S.A. , vol.89 , pp. 3050-3054
    • Takimoto, G.S.1    Tasset, D.M.2    Eppert, A.C.3    Horwitz, K.B.4
  • 19
    • 0026768322 scopus 로고
    • A limiting factor mediates the differential activation of promoters by the human progesterone receptor isoforms
    • Meyer M.E., Quirin-Stricker C., Lerouge T., Bocquel M.T., Gronemeyer H. A limiting factor mediates the differential activation of promoters by the human progesterone receptor isoforms. J. Biol. Chem. 267:1992;10882-10887.
    • (1992) J. Biol. Chem. , vol.267 , pp. 10882-10887
    • Meyer, M.E.1    Quirin-Stricker, C.2    Lerouge, T.3    Bocquel, M.T.4    Gronemeyer, H.5
  • 20
    • 0027494065 scopus 로고
    • Antagonist-occupied human progesterone B-receptors activate transcription without binding to progesterone response elements and are dominantly inhibited by A-receptors
    • Tung L., Mohamed M.K., Hoeffler J.P., Takimoto G.S., Horwitz K.B. Antagonist-occupied human progesterone B-receptors activate transcription without binding to progesterone response elements and are dominantly inhibited by A-receptors. Mol. Endocrinol. 7:1993;1256-1265.
    • (1993) Mol. Endocrinol. , vol.7 , pp. 1256-1265
    • Tung, L.1    Mohamed, M.K.2    Hoeffler, J.P.3    Takimoto, G.S.4    Horwitz, K.B.5
  • 21
    • 0027427216 scopus 로고
    • Human progesterone receptor a form is a cell- and promoter-specific repressor of human progesterone receptor B function
    • Vegeto E., Shabaz M.M., Wen D.X., Goldman M.E., O'Malley B.W., McDonnell D.P. Human progesterone receptor A form is a cell- and promoter-specific repressor of human progesterone receptor B function. Mol. Endocrinol. 7:1993;1244-1255.
    • (1993) Mol. Endocrinol. , vol.7 , pp. 1244-1255
    • Vegeto, E.1    Shabaz, M.M.2    Wen, D.X.3    Goldman, M.E.4    O'Malley, B.W.5    McDonnell, D.P.6
  • 22
    • 0027156480 scopus 로고
    • Antagonist-occupied human progesterone receptors bound to DNA are functionally switched to transcriptional agonists by cAMP
    • Sartorius C.A., Tung L., Takimoto G.S., Horwitz K.B. Antagonist-occupied human progesterone receptors bound to DNA are functionally switched to transcriptional agonists by cAMP. J. Biol. Chem. 268:1993;9262-9266.
    • (1993) J. Biol. Chem. , vol.268 , pp. 9262-9266
    • Sartorius, C.A.1    Tung, L.2    Takimoto, G.S.3    Horwitz, K.B.4
  • 23
    • 0028358327 scopus 로고
    • The human progesterone receptor A-form functions as a transcriptional modulator of mineralocorticoid receptor transcriptional activity
    • McDonnell D.P., Shahbaz M.M., Vegeto E., Goldman M.E. The human progesterone receptor A-form functions as a transcriptional modulator of mineralocorticoid receptor transcriptional activity. J. Steroid Biochem. Mol. Biol. 48:1994;425-432.
    • (1994) J. Steroid Biochem. Mol. Biol. , vol.48 , pp. 425-432
    • McDonnell, D.P.1    Shahbaz, M.M.2    Vegeto, E.3    Goldman, M.E.4
  • 24
    • 0032489366 scopus 로고    scopus 로고
    • An N-terminal inhibitory function, IF, suppresses transcription by the A-isoform but not the B-isoform of human progesterone receptors
    • Hovland A.R., Powell R.L., Takimoto G.S., Tung L., Horwitz K.B. An N-terminal inhibitory function, IF, suppresses transcription by the A-isoform but not the B-isoform of human progesterone receptors. J. Biol. Chem. 273:1998;5455-5560.
    • (1998) J. Biol. Chem. , vol.273 , pp. 5455-5560
    • Hovland, A.R.1    Powell, R.L.2    Takimoto, G.S.3    Tung, L.4    Horwitz, K.B.5
  • 25
    • 0033651180 scopus 로고    scopus 로고
    • Progesterone receptor modulators and progesterone antagonists in women's health
    • Spitz I., Chwalisz K. Progesterone receptor modulators and progesterone antagonists in women's health. Steroids. 65:2000;807-815.
    • (2000) Steroids , vol.65 , pp. 807-815
    • Spitz, I.1    Chwalisz, K.2
  • 26
    • 0037062484 scopus 로고    scopus 로고
    • Coactivator/corepressor ratios modulate PR-mediated transcription by selective receptor modulator RU486
    • Lui Z., Auboeuf D., Wong J., Chen J.D., Tsai S.Y., Tsai M.J.et al. Coactivator/corepressor ratios modulate PR-mediated transcription by selective receptor modulator RU486. Proc. Natl. Acad. Sci. U.S.A. 99:2002;7940-7944.
    • (2002) Proc. Natl. Acad. Sci. U.S.A. , vol.99 , pp. 7940-7944
    • Lui, Z.1    Auboeuf, D.2    Wong, J.3    Chen, J.D.4    Tsai, S.Y.5    Tsai, M.J.6
  • 27
    • 0030946198 scopus 로고    scopus 로고
    • Coactivator and corepressor regulation of the agonist/antagonist activity of the mixed antiestrogen, 4-hydroxytamoxifen
    • Smith C.L., Nawaz Z., O'Malley B.W. Coactivator and corepressor regulation of the agonist/antagonist activity of the mixed antiestrogen, 4-hydroxytamoxifen. Mol. Endocrinol. 11:1997;657-666.
    • (1997) Mol. Endocrinol. , vol.11 , pp. 657-666
    • Smith, C.L.1    Nawaz, Z.2    O'Malley, B.W.3
  • 28
    • 0037192501 scopus 로고    scopus 로고
    • Molecular determinants for the tissue specificity of SERMs
    • Shang Y., Brown M. Molecular determinants for the tissue specificity of SERMs. Science. 295:2002;2465-2468.
    • (2002) Science , vol.295 , pp. 2465-2468
    • Shang, Y.1    Brown, M.2
  • 29
    • 0034050902 scopus 로고    scopus 로고
    • Systematic variation in gene expression patterns in human cancer cell lines
    • Ross D.T., Scherf U., Eisen M.B., Perou C.M., Rees C., Spellman P.et al. Systematic variation in gene expression patterns in human cancer cell lines. Nat. Genet. 24:2000;227-235.
    • (2000) Nat. Genet. , vol.24 , pp. 227-235
    • Ross, D.T.1    Scherf, U.2    Eisen, M.B.3    Perou, C.M.4    Rees, C.5    Spellman, P.6


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