Synthesis of some thiochromone derivatives and activity against Plasmodium falciparum in-vitro

Pharmacy and Pharmacology Communications

Volumn 5, Issue 2, 1999, Pages 107-110

  Charris, J ^a   Dominguez J ^a   Lobo, G ^a   Riggione, F ^b  

^a UNIVERSIDAD CENTRAL DE VENEZUELA   (Venezuela)

^b UNIVERSIDAD CENTRAL DE VENEZUELA   (Venezuela)

Author keywords

[No Author keywords available]

Indexed keywords

ANTIMALARIAL AGENT; GUANIDINE DERIVATIVE; HYDRAZINE; PYRIMETHAMINE; THIOCHROMAN DERIVATIVE;

ARTICLE; CONTROLLED STUDY; DRUG SYNTHESIS; NONHUMAN; PLASMODIUM FALCIPARUM;

EID: 0345130055     PISSN: 14608081     EISSN: None     Source Type: Journal    
DOI: 10.1211/146080899128734541     Document Type: Article

References (7)

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2. Domínguez, J., Basante, W., Charris, J., Riggione, F. (1996a) Synthesis and activity of some quinolone derivatives against Plasmodium falciparum in vitro. Farmaco 51: 407-412
3. Domínguez, J., Charris, J., Iarruso, L., López, S., Lobo, G., Riggione, F. (1996b) Synthesis of pyridopyrimidone derivatives and their activity against P. Falciparum in vitro. Farmaco 51: 781-784
4. Domínguez, J., López, S., Charris, J., Iarruso, L., Lobo, G., Semenov, A., Olson, P. J., Rosenthal, P. J. (1997) Synthesis and antimalarial effects of phenothiazine inhibitors of a Plasmodium falciparum cysteine protease. J. Med. Chem. 40: 2726-2732
5. 13C NMR spectral characterization of some antimalarial tricyclic quinolone derivatives. Magn. Reson. Chem. 36: 454-456
6. Rudorf, W. D. (1977) Heterocyclensynthesen mit o-chlorobenzoylacetonitril. Tetrahedron 34: 725-730
7. Rudorf, W. D., Augustin, M. (1981) Umsetzungen substituierter 1-thiochromone und 4(1H)-chinolone mit nucleophilen. J. Prakt. Chem. 323: 55-62