One pot synthesis of unsymmetrically functionalized polyamines by a solid phase strategy starting from their symmetrical polyamine-counterparts

Tetrahedron Letters

Volumn 38, Issue 18, 1997, Pages 3219-3222

  Gerardo, Byk ^a   Frederic, Marc ^a   Scherman, Daniel ^a  

^a CNRS   (France)

Author keywords

[No Author keywords available]

Indexed keywords

POLYAMINE;

ARTICLE; DRUG SYNTHESIS; HIGH PERFORMANCE LIQUID CHROMATOGRAPHY; IN VITRO STUDY; METHODOLOGY; NUCLEAR MAGNETIC RESONANCE SPECTROSCOPY; REACTION ANALYSIS; THIN LAYER CHROMATOGRAPHY;

EID: 0343471510     PISSN: 00404039     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0040-4039(97)00582-0     Document Type: Article

References (19)

1. (a) Ganem, B. Acc. Chem. Res. 1982, 15, 290.
2. (b) Bergeron, R.J. Acc. Chem. Res. 1986, 19, 105.
3. (c) Edwards, M.L.; Stemerick D.M.; Kline S.J. Tetrahedron Lett. 1990, 31, 3417.
4. (d) Blagbrough, I.S.; Moya, E.; Walfort, S.P. Tetrahedron Lett. 1996, 37, 551-554.
5. (e) Goulaouic-Dubois, C.; Guggisberg, A.; Hesse, M. Tetrahedron 1995, 51, 12573-12582.
6. Merrifield, R.B. J. Am. Chem. Soc. 1963, 85, 2149.
7. Bycroft, B.W.; Chan, W.C.; Chhabra, S.R.; Hone, N.D. J. Chem. Commun. 1993, 778-779.
8. Personal communication from Fabrice Cornille U266 INSERM-URA D1500 CNRS, Paris-France.
9. Nash, I.A.; Bycroft, B.W.; Chan, W.C. Tetrahedron Lett. 1996, 15, 2625-2628.
10. Bycroft, B.W.; Chan, W.C.; Hone, N.D.; Millington, S.; Nash, I.A. J. Am. Chem. Soc. 1994, 116, 7415-7416.
11. Furka, A.; Sebestyen, F.; Asgedon, M.; Dibo, G.; Int. J. Peptide Protein Res. 1991, 37, 487.
12. Aramaki, Y.; Yasuhara, T.; Higashijima, T.; Yoshioka, M.; Miwa, A.; Kawai, N.; Nakajima, T. Proc. Japan Acad. Sci. 1986, 62B, 359-362.
13. (a) Toki, T.; Yasuhara, T.; Aramaki, Y.; Osowa, K.; Miwa, A.; Kawai, N.; Nakashima, T. Biomedical Res. 1988, 9, 421-428.
14. (b) Yoshioka, M.; Narai, N.; Teshima, T.; Matsumoto, T.; Wakamiya, T.; Shiba, T.; Tokoro, N.; Okauchi, T.; Kono, Y. Chem. Pharm. Bull. 1992, 40, 3005-3008.
15. (a) Granier, C.; Guilard, R. Tetrahedron 1995, 51, 1197-1208.
16. (b) Kaden, T.A.; Studer, M. Helv. Chim. Acta 1986, 69, 2081-2086
17. Yamamoto, H.; Maruoka, K. J. Am. Chem. Soc. 1981, 103, 6133-6136.
18. Koike, T.; Watanabe, T.; Aoki, S.; Kimura, E. and Shiro, M. J. Am. Chem. Soc. 1996, 118, 12696-12703.
19. Kaiser, E.; Colescolt, D.L.; Bossinger, C.D.; Cook, P.I. Anal. Biochem. 1970, 34, 595.