Assessment of new 6-Cl-HOBt based coupling reagents for peptide synthesis. Part 1: Coupling efficiency study

Letters in Peptide Science

Volumn 9, Issue 2-3, 2002, Pages 119-123

  Sabatino, Giuseppina ^a   Mulinacci, Barbara ^a   Alcaro, Maria C ^a   Chelli, Mario ^a   Rovero, Paolo ^b   Papini, Anna M ^a  

^a UNIVERSITY OF FLORENCE   (Italy)

^b UNIVERSITY OF SALERNO   (Italy)

Author keywords

Automatic solid phase peptide synthesis; Coupling reagents; HCTU; TCTU

Indexed keywords

ACYL CARRIER PROTEIN; ALANINE; AMINE; AMMONIUM DERIVATIVE; ASPARAGINE; ASPARTIC ACID; GLYCINE; ISOLEUCINE; PEPTIDE; PHOSPHONIUM DERIVATIVE; REAGENT; TYROSINE; VALINE;

AMINO ACID SEQUENCE; CHEMICAL REACTION; CHEMICAL STRUCTURE; CONFERENCE PAPER; DIFFUSION; ENANTIOSELECTIVITY; PEPTIDE SYNTHESIS; SEQUENCE ANALYSIS; SOLUBILITY;

EID: 0242500411     PISSN: 09295666     EISSN: None     Source Type: Journal    
DOI: 10.1023/A:1024140900571     Document Type: Conference Paper

References (13)

1. Albericio, F. and Kates, S. A., In Solid-Phase Synthesis: A Practical Guide, S. A. Kates and F. Albericio (eds), Marcel Dekker, New York, 2000, pp. 275-330.
2. Albericio, F., Bofill, J. M., El-Faham, A. and Kates, S. A., J. Org. Chem., 63 (1998) 9678.
3. Albericio, F., Bailén, M. A., Chinchilla, R., Dodsworth, D. J. and Nájera, C., Tetrahedron, 57 (2001) 9607.
4. König, W. and Geiger, R., Chem. Ber., 103 (1970) 788.
5. Carpino, L. A., J. Am. Chem. Soc., 115 (1993) 4397.
6. Carpino, L. A., El-Faham, A., Minor, C. A. and Albericio, F., J. Chem. Soc., Chem Commun., (1994) 201.
7. Knorr, R., Trzeciak, A., Bannwarth, W. and Gillessen, D., Tetrahedron Lett., 30 (1989) 1927.
8. Castro, B., Dormoy, J. R., Evin, G. and Selve, C., Tetrahedron Lett., (1975) 1219.
9. Israeli Patent Application No: IL141804.
10. Kaminski, Z. J., Paneth, P. and Rudzinki, J., J. Org. Chem., 63 (1998) 4248.
11. Falchi, A., Giacomelli, G., Porcheddu, A. and Taddei, M., Synlett, (2000) 275.
12. Atherton, E. and Sheppard, R. C., In Solid Phase Peptide Synthesis: A Practical Approach, D. Rickwood and B. D. Hames (eds), IRL Press, Oxford, 1989, p. 117.
13. Kunishima, M., Kawachi, C., Morita, J., Terao, K., Iwasaki, F. and Tani, S., Tetrahedron, 55 (1999) 13159.