A convenient synthesis of monocationic 1-[(cyclic amidino)methyl]thymines

Synthetic Communications

Volumn 27, Issue 19, 1997, Pages 3431-3440

  Spychała, Jarosław ^a  

^a ADAM MICKIEWICZ UNIVERSITY   (Poland)

Author keywords

[No Author keywords available]

Indexed keywords

THYMINE DERIVATIVE;

ARTICLE; DRUG SYNTHESIS; IN VITRO STUDY; INFRARED SPECTROPHOTOMETRY; MASS SPECTROMETRY; METHODOLOGY; NUCLEAR MAGNETIC RESONANCE SPECTROSCOPY; REACTION ANALYSIS;

EID: 0142110800     PISSN: 00397911     EISSN: None     Source Type: Journal    
DOI: 10.1080/00397919708005644     Document Type: Article

References (26)

1. Borthwick, A. D., and Biggadike, K. Tetrahedron 1992, 48, 571.
2. Grangier, G., Aitken, D. J., Guillaume, D., and Husson, H.-P. Tetrahedron Lett. 1994, 35, 4355.
3. Wilson, W. D, Ratmeyer, L., Cegla, M. T., Spychala, J., Boykin, D., Demeunynck, M., Lhomme, J., Krishnan, G., Kennedy, D., Vinayak, R., and Zon, G. New J. Chem. 1994, 18, 419.
4. Chen, X., Bastow, K., Goz, B., Kucera, L., Morris-Natschke, S. L., and Ishaq, K. S. Antiviral Chem. Chemother. 1996, 7, 108.
5. Hiebl, J., Zbiral, E., von Janta-Lipinski, M., Balzarini, J., and De Clercq, E. Antiviral Chem. Chemother. 1996, 7, 173.
6. Fedorov, I.I., Kazmina, E.M., Gurskaya, G.V., Jasko, MV, Zavodnic, V.E., Balzarini, J., De Clercq, E., Faraj, A., Sommadossi, J.-P., Imbach, J.-L., and Gosselin, G. J. Med Chem. 1997, 40, 486.
7. Hong, C. I., Nechaev, A., Kirisits, A. J., Vig, R., West, C. R., Manouilov, K. K., and Chu, C. K. J. Med. Chem. 1996, 39, 1771.
8. Undheim, K., and Benneche, T. in Comprehensive Heterocyclic Chemistry II, vol. 6, Katritzky, A.R., Rees, C.W., Scriven, E.F.V., and Boulton, A.J. (Eds.), 1996, 93.
9. Borg, N., Zhou, X.-X., Johansson, N.-G., Öberg, B., and Stahle, L. Antiviral Chem. Chemother. 1997, 8, 47.
10. Mansour, T. S., and Jin, H. Bioorg. Med. Chem. Lett. 1991, 1, 757.
11. Grout, R. J. in The Chemistry of Amidines and Imidates. Patai, S. (Ed.), John Wiley & Sons, An Interscience Publication, London, 1975, 255.
12. Gould, L., and Reddy, C. V. R. Am. Heart J. 1976, 92, 397.
13. Rosati, G. F., and Poletto, M. G. Farmaco Ed. Prat. 1966, 21, 204.
14. Faust, J. A., Mori, A., and Sahyun, M. J. Am. Chem. Soc. 1959, 81, 2214.
15. Forssell, G. Ber. 1891, 24, 1846.
16. Boyd, G. V. in The Chemistry of Amidines and Imidates, vol. 2, Patai, S., and, Rappoport, Z. (Eds.), John Wiley & Sons, Chichester, New York, 1991, 339.
17. Gabriel, S., and Heymann, P. Ber. 1890, 23, 157.
18. Kindler, K. Ann. 1923, 431, 187.
19. Erlenmeyer, H., and Degen, K., Helv. Chim. Acta, 1946, 29, 1080.
20. Kornfeld, E. C. J. Org. Chem. 1951, 16, 131.
21. Pickering, M. V., Srivastava, P. C., Witkowski, J. T., and Robins, R. K. in Nucleic Acid Chemistry, Improved and New Synthetic Procedures,Methods and Techniques, part one, Townsend, L. B., and Tipson, R. S. (Eds.), John Wiley & Sons, Inc., New York, Chichester, Brisbane, Toronto, 1978, 145.
22. Bulychev, Y. N., Korbukh, I. A., and Preobrazhenskaya, M.N. in Nucleic Acid Chemistry,Improved and New Synthetic Procedures,Methods and Techniques, part three, Townsend, L. B., and Tipson, R. S.(Eds.), John Wiley & Sons,Inc., New York, Chichester, Brisbane, Toronto, Singapore, 1986, 218.
23. Cristalli, G., Eleuteri, A., Franchetti, P., Grifantini, M., Vittori, S., and Lupidi, G. J. Med. Chem. 1991, 34, 1187.
24. Ward, A. D., and Baker, B. R. J. Med. Chem. 1977, 20, 88.
25. Chavis, C., Dumont, F., Wightman, R., Ziegler, J.-C., and Imbach, J.-L. in Nucleic Acid Chemistry, Improved and New Synthetic Procedures,Methods and Techniques, part three, Townsend, L. B., and Tipson, R. S. (Eds.). John Wiley & Sons,Inc., New York, Chichester, Brisbane, Toronto, 1986, 76.
26. Singh, H., Aggarwal, P., and Kumar, S. Synthesis 1990, 520.