Thermodynamics of partitioning of benzocaine in some organic solvent/buffer and liposome systems

Chemical and Pharmaceutical Bulletin

Volumn 51, Issue 3, 2003, Pages 237-240

  Ávila, Carolina Mercedes ^a   Martínez, Fleming ^a  

^a UNIVERSIDAD NACIONAL DE COLOMBIA   (Colombia)

Author keywords

Benzocaine; Liposome; Partition coefficient; Partitioning; Thermodynamic

Indexed keywords

BENZOCAINE; CYCLOHEXANE; DIMYRISTOYLPHOSPHATIDYLCHOLINE; DIPALMITOYLPHOSPHATIDYLCHOLINE; LIPOSOME; MYRISTIC ACID ISOPROPYL ESTER; OCTANOL; ORGANIC SOLVENT; BUFFER; SOLVENT;

ARTICLE; ENTHALPY; ENTROPY; LIPOPHILICITY; PARTITION COEFFICIENT; TEMPERATURE; THERMODYNAMICS; CHEMISTRY; COMPARATIVE STUDY; METABOLISM;

BENZOCAINE; BUFFERS; LIPOSOMES; SOLVENTS; THERMODYNAMICS;

EID: 0142009517     PISSN: 00092363     EISSN: 13475223     Source Type: Journal    
DOI: 10.1248/cpb.51.237     Document Type: Article

References (38)

1. Catterall W., Mackie K., "Goodman & Gilman's. The Pharmacological Basis of Therapeutics," 10th edn., Chapter 15, ed. by Hardman J. G., Limbird L. E., Gilman A. G., McGraw-Hill, New York, 2001.
2. Wang H. H., Earnest J., Limbacher H. P., Proc. Natl. Acad. Sci. U.S.A., 80, 5297-5301 (1983).
3. Peters H., Moll F., Arzneim.-Forsch./Drug Res., 45, 1253-1256 (1995).
4. Sanchez V., Arthur G. R., Strichartz G. R., Anesth. Analg., 66, 159-165 (1987).
5. Fleming R., Guy R. H., Hadgraft J., J. Pharm. Sci., 72, 142-145 (1983).
6. Strichartz G. R., Sanchez V., Arthur G. R., Chafetz R., Martin D., Anesth. Analg., 71, 158-170 (1990).
7. Seeman P., Pharmacol. Rev., 24, 583-655 (1972).
8. Betageri G. V., Nayernama A., Habib M. J., Int. J. Pharm. Adv., 1, 310-319 (1996).
9. Leo A., Hansch C., Elkins D., Chem. Rev., 71, 525-616 (1971).
10. Diamond J. M., Katz Y., J. Membr. Biol., 17, 121-154 (1974).
11. Sangster J., "Octanol-Water Partition Coefficients: Fundamentals and Physical Chemistry," John Wiley & Sons, Chichester, UK, 1997.
12. Barker N., Hadgraft J., Int. J. Pharmaceut., 8, 193-202 (1981).
13. Pozzo A. D., Donzelli G., Liggeri E., Rodriguez L., J. Pharm. Sci., 80, 54-57 (1991).
14. Jaiswal J., Poduri R., Panchagnula R., Int. J. Pharmaceut., 179, 129-134 (1999).
15. Rogers J. A., Davis S. S., Biochim. Biophys. Acta, 598, 392-404 (1980).
16. Anderson N. H., Davis S. S., James M., Kojima I., J. Pharm. Sci., 72, 443-448 (1983).
17. Ahmed M., Burton J. S., Hadgraft J., Kellaway I. W., J. Membr. Biol., 58, 181-189 (1981).
18. Ahmed A. M. S., Farah F. H., Kellaway I. W., Pharm. Res., 3, 119-124 (1985).
19. Betageri G. V., Rogers J. A., Int. J. Pharmaceut., 36, 165-173 (1987).
20. Betageri G. V., Dipali S. R., J. Pharm. Pharmacol., 45, 931-933 (1993).
21. Go M. L., Ngiam T. L., Rogers J. A., Chem. Pharm. Bull., 43, 289-294 (1995).
22. Go M. L., Ngiam T. L., Chem. Pharm. Bull., 45, 2055-2060 (1997).
23. Avila C. M., B.Sc. Thesis, National University of Colombia, 2001.
24. Bangham A. D., Phys. Chem. Lipids, 64, 275-285 (1993).
25. Lasic D. D., Sci. Med., 1996, (May/June), 34-43 (1996).
26. Beltrán O. C., Escobar M. J., Jiménez F., Barbosa H. J., Martínez F., Rev. Col. Cienc. Quím. Farm., 28, 117-122 (1999).
27. Cevc G., "Liposomes Technology," Vol. 1, Chapter 1, ed. by Gregoriadis G., CRC Press, Boca Raton, 1993.
28. Martin A. N., Bustamante P., Chun A. H. C., "Physical Pharmacy: Physical Chemical Principles in the Pharmaceutical Sciences," 4th edn., Lea & Febiger, Philadelphia, 1993.
29. Florence A. T., Attwood D., "Physicochemical Principles of Pharmacy," 3rd edn., MacMillan Press, London, 1998.
30. Martínez F., Tello M., Gómez A., Rev. Col. Cienc. Quím. Farm., 29, 16-25 (2000).
31. Budavari S., O'Neil M. J., Smith A., Heckelman P. E., Kinneary J. F., "The Merck Index, An Encyclopedia of Chemicals, Drugs, and Biologicals," 12th edn., Merck & Co., Inc., Whitehouse Station, N.J., 1996.
32. Pinto L. M., Yokaichiya D. K., Fraceto L. F., de Paula E., Biophys. Chem., 87, 213-222 (2000).
33. Bevington P. R., "Data Reduction and Error Analysis for the Physical Sciences," McGraw-Hill Book Co., New York, 1969.
34. Koynova R., Caffrey M., Biochim. Biophys. Acta, 1376, 91-145 (1998).
35. Lipidat: Lipid thermotropic phase transition database, Ohio State University. Internet: 〈http://www.lipidat.chemistry.ohio-state.edu〉, 15 July 2001.
36. Seiler P., Eur. J. Med. Chem.-Chim. Ther., 9, 473-479 (1974).
37. DeBolt S. E., Kollman P. A., J. Am. Chem. Soc., 117, 5316-5340 (1995).
38. Martínez F., Ph.D. Thesis, National University of Colombia, 2001.