An efficient route to 4-(substituted benzyl)piperidines

Tetrahedron Letters

Volumn 44, Issue 45, 2003, Pages 8249-8252

  Furman, Bartłomiej ^a   Dziedzic, Magdalena ^a  

^a INSTITUTE OF ORGANIC CHEMISTRY   (Poland)

Author keywords

Cyclisation; Heck reaction; Piperidines

Indexed keywords

4 METHYLENEPIPERIDINE; IMINE; ORGANOBORON DERIVATIVE; OXYGEN; PALLADIUM; PIPERIDINE DERIVATIVE; SILANE DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; ATMOSPHERE; CATALYSIS; CHEMICAL BOND; CHEMICAL REACTION; CYCLIZATION; DRUG SYNTHESIS;

EID: 0141992099     PISSN: 00404039     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.tetlet.2003.09.075     Document Type: Article

References (19)

1. Ohshima E., Takami H., Harakawa H., Sato H., Obase H., Miki I., Ishii H., Sasaki Y., Ohmori K., Karasawa A., Kubo K. J. Med. Chem. 36:1993;417-420.
2. Shanklin J.R. Jr., Johnson C.P. III, Proakis A.G., Barrett R.J. J. Med. Chem. 34:1991;3011-3022.
3. Roufos I., Hays S., Schwarz R.D. J. Med. Chem. 39:1996;1514-1520.
4. Wick, A.; Frost, J.; Gaudilliere, B.; Bertin, J.; Dupont, R.; Rousseau, J. US Patent 4690931 1987.
5. Zhou Z.-L., Keana J.F.W. J. Org. Chem. 64:1999;3763-3766.
6. Vice S., Bara T., Bauer A., Evans C.A., Ford J., Josien H., McCombie S., Miller M., Nazareno D., Palani A., Tagat J. J. Org. Chem. 66:2001;2487-2492.
7. Rubiralta M., Diez A., Miguel D., Remuson R., Gelas-Mialhe Y. Synth. Commun. 22:1992;359-367.
8. Kobayashi S., Busujima T., Nagayama S. Chem. Commun. 1998;19-20.
9. 2S 251.09800, found 251.09776.
10. Cacchi S., Fabrizi G., Gallina C., Pace P. Synlett. 1997;54-55.
11. Peng S., Qing F-L., Guo Y. Synlett. 1998;859-860.
12. Littke A.F., Fu G.C. J. Am. Chem. Soc. 123:2001;6989-7000.
13. Jung Y.Ch., Mishra R.K., Yoon Ch.H., Jung K.W. Org. Lett. 5:2003;2231-2234.
14. 2S 327.12930, found 327.12919.
15. Smith K.A., Campi E.M., Jackson W.R., Marcuccio S., Naeslund Ch.G.M., Deacon G.B. Synlett. 1997;131-132.
16. Wong M.S., Zhang X.L. Tetrahedron Lett. 42:2001;4087-4089.
17. Parrish J.P., Jung Y.C., Floyd J., Jung K.W. Tetrahedron Lett. 43:2002;7899-7902.
18. Yoshida H., Yamaryo Y., Ohshita J., Kunai A. Tetrahedron Lett. 44:2003;1541-1544.
19. 2S 329.14495, found 329.14479.