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Volumn 310, Issue 3, 2003, Pages 785-790

Binding characteristics of SSR180575, a potent and selective peripheral benzodiazepine ligand

Author keywords

Binding characteristics; Cell; Mitochondria; Peripheral benzodiazepine receptor; SSR180575

Indexed keywords

7 CHLORO N,N,5 TRIMETHYL 4 OXO 3 PHENYL 3,5 DIHYDRO 4H PYRIDAZINO[4,5 B]INDOL 1 ACETAMIDE; BENZODIAZEPINE DERIVATIVE; BENZODIAZEPINE RECEPTOR; SSR 180575; UNCLASSIFIED DRUG;

EID: 0141645393     PISSN: 0006291X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bbrc.2003.09.079     Document Type: Article
Times cited : (36)

References (16)
  • 1
    • 0017730392 scopus 로고
    • High densities of benzodiazepine receptors in human cortical areas
    • Braestrup C., Albrechtsen R., Squires R.F. High densities of benzodiazepine receptors in human cortical areas. Nature. 269:1977;5702-5704.
    • (1977) Nature , vol.269 , pp. 5702-5704
    • Braestrup, C.1    Albrechtsen, R.2    Squires, R.F.3
  • 2
    • 0031893596 scopus 로고    scopus 로고
    • Topological analysis of the peripheral benzodiazepine receptor in yeast mitochondrial membranes supports a five-transmembrane structure
    • Joseph-Liauzun E., Delmas P., Shire D., Ferrara P. Topological analysis of the peripheral benzodiazepine receptor in yeast mitochondrial membranes supports a five-transmembrane structure. J. Biol. Chem. 273:1998;2146-2152.
    • (1998) J. Biol. Chem. , vol.273 , pp. 2146-2152
    • Joseph-Liauzun, E.1    Delmas, P.2    Shire, D.3    Ferrara, P.4
  • 3
    • 0026639447 scopus 로고
    • Biochemical, physiological, and pathological aspects of the PBR
    • Gavish M., Katz Y., Bar-Ami S., Weizman R. Biochemical, physiological, and pathological aspects of the PBR. J. Neurochem. 58:1992;1589-1601.
    • (1992) J. Neurochem. , vol.58 , pp. 1589-1601
    • Gavish, M.1    Katz, Y.2    Bar-Ami, S.3    Weizman, R.4
  • 4
    • 0026591024 scopus 로고
    • Isolation of the mitochondrial benzodiazepine receptor: Association with the voltage-dependent anion channel and the adenine nucleotide carrier
    • McEnery M.W., Snowman A.M., Trifiletti R.R., Snyder S.H. Isolation of the mitochondrial benzodiazepine receptor: association with the voltage-dependent anion channel and the adenine nucleotide carrier. Proc. Natl. Acad. Sci. USA. 89:1992;3170-3174.
    • (1992) Proc. Natl. Acad. Sci. USA , vol.89 , pp. 3170-3174
    • McEnery, M.W.1    Snowman, A.M.2    Trifiletti, R.R.3    Snyder, S.H.4
  • 5
    • 0018347895 scopus 로고
    • Characterization of benzodiazepine binding sites in cultured cells of neural origin
    • Syapin P.J., Skolnick P. Characterization of benzodiazepine binding sites in cultured cells of neural origin. J. Neurochem. 32:1979;1047-1051.
    • (1979) J. Neurochem. , vol.32 , pp. 1047-1051
    • Syapin, P.J.1    Skolnick, P.2
  • 6
    • 0020576925 scopus 로고
    • Peripheral benzodiazepine binding sites: Effect of PK 11195, 1-(2-chlorophenyl)-N-methyl-N-(1-methylpropyl)-3-isoquinolinecarboxamide. I. In vitro studies
    • Le Fur G., Perrier M.L., Vaucher N., Imbault F., Flamier A., Benavides J., Uzan A., Renault C., Dubroeucq M.C., Gueremy C. Peripheral benzodiazepine binding sites: effect of PK 11195, 1-(2-chlorophenyl)-N-methyl-N-(1-methylpropyl)-3-isoquinolinecarboxamide. I. In vitro studies. Life Sci. 32:1983;1839-1847.
    • (1983) Life Sci. , vol.32 , pp. 1839-1847
    • Le Fur, G.1    Perrier, M.L.2    Vaucher, N.3    Imbault, F.4    Flamier, A.5    Benavides, J.6    Uzan, A.7    Renault, C.8    Dubroeucq, M.C.9    Gueremy, C.10
  • 7
    • 0022574416 scopus 로고
    • The peripheral-type benzodiazepine receptor. Localization to the mitochondrial outer membrane
    • Anholt R.R., Pedersen P.L., De Souza E.B., Snyder S.H. The peripheral-type benzodiazepine receptor. Localization to the mitochondrial outer membrane. J. Biol. Chem. 261:1986;576-583.
    • (1986) J. Biol. Chem. , vol.261 , pp. 576-583
    • Anholt, R.R.1    Pedersen, P.L.2    De Souza, E.B.3    Snyder, S.H.4
  • 8
    • 0029915241 scopus 로고    scopus 로고
    • Involvement of peripheral benzodiazepine receptors in the protection of hematopoietic cells against oxygen radical damage
    • Carayon P., Portier M., Dussossoy D., Bord A., Petitpretre G., Canat X., Le Fur G., Casellas P. Involvement of peripheral benzodiazepine receptors in the protection of hematopoietic cells against oxygen radical damage. Blood. 87:1996;3170-3178.
    • (1996) Blood , vol.87 , pp. 3170-3178
    • Carayon, P.1    Portier, M.2    Dussossoy, D.3    Bord, A.4    Petitpretre, G.5    Canat, X.6    Le Fur, G.7    Casellas, P.8
  • 9
    • 0027234336 scopus 로고
    • The mitochondrial permeability transition pore may comprise VDAC molecules: I. Binary structure and voltage dependence of the pore
    • Szabo I., Zoratti M. The mitochondrial permeability transition pore may comprise VDAC molecules: I. Binary structure and voltage dependence of the pore. FEBS Lett. 330:1993;201-205.
    • (1993) FEBS Lett. , vol.330 , pp. 201-205
    • Szabo, I.1    Zoratti, M.2
  • 11
    • 0041932414 scopus 로고    scopus 로고
    • Role of peripheral benzodiazepine receptors in mitochondrial, cellular and cardiac damage induced by oxidative stress and ischemia-reperfusion
    • Leducq N., Bono F., Sulpice T., Vin V., Janiak P., Le Fur G., O'Connor S.E., Herbert J.M. Role of peripheral benzodiazepine receptors in mitochondrial, cellular and cardiac damage induced by oxidative stress and ischemia-reperfusion. J. Pharmacol. Exp. Ther. 306:2003;828-837.
    • (2003) J. Pharmacol. Exp. Ther. , vol.306 , pp. 828-837
    • Leducq, N.1    Bono, F.2    Sulpice, T.3    Vin, V.4    Janiak, P.5    Le Fur, G.6    O'Connor, S.E.7    Herbert, J.M.8
  • 13
    • 0041809082 scopus 로고    scopus 로고
    • The peripheral benzodiazepine receptor: A promising therapeutic drug target
    • Galiegue S., Tinel N., Casellas P. The peripheral benzodiazepine receptor: a promising therapeutic drug target. Curr. Med. Chem. 10:2003;1563-1572.
    • (2003) Curr. Med. Chem. , vol.10 , pp. 1563-1572
    • Galiegue, S.1    Tinel, N.2    Casellas, P.3
  • 15
    • 0028067990 scopus 로고
    • Rapid isolation of highly productive recombinant Chinese hamster ovary cell lines
    • Miloux B., Lupker J.H. Rapid isolation of highly productive recombinant Chinese hamster ovary cell lines. Gene. 149:1994;341-344.
    • (1994) Gene , vol.149 , pp. 341-344
    • Miloux, B.1    Lupker, J.H.2
  • 16
    • 0033536556 scopus 로고    scopus 로고
    • Specific binding of benzodiazepines to human breast cancer cell lines
    • Beinlich A., Strohmeier R., Kaufmann M., Kuhl H. Specific binding of benzodiazepines to human breast cancer cell lines. Life Sci. 65:1999;2099-2108.
    • (1999) Life Sci. , vol.65 , pp. 2099-2108
    • Beinlich, A.1    Strohmeier, R.2    Kaufmann, M.3    Kuhl, H.4


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.