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Volumn 261, Issue 1-2, 2003, Pages 69-80

PLGA-PEG microspheres of teverelix: Influence of polymer type on microsphere characteristics and on teverelix in vitro release

Author keywords

Coacervation; GnRH antagonists; In vitro release; Microspheres; PEG; PLGA PEG

Indexed keywords

COPOLYMER; GLYCOLIC ACID DERIVATIVE; MACROGOL; MICROSPHERE; POLY(LACTIC GLYCOLIC ACID); POLYMER; TEVERELIX; UNCLASSIFIED DRUG;

EID: 0042026308     PISSN: 03785173     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0378-5173(03)00272-2     Document Type: Article
Times cited : (32)

References (32)
  • 1
    • 0024319040 scopus 로고
    • In vivo characteristics of low molecular weight copoly(L-lactic acid/glycolic acid) formulations with controlled release of luteinizing hormone-releasing hormone agonist
    • Asano M., Fukuzaki H., Yoshida M., Kumakura M., Mashimo T., Yuasa H., Imai K., Yamanaka H., Suzuki K. In vivo characteristics of low molecular weight copoly(L-lactic acid/glycolic acid) formulations with controlled release of luteinizing hormone-releasing hormone agonist. J. Control. Rel. 9:1989;111-122.
    • (1989) J. Control. Rel. , vol.9 , pp. 111-122
    • Asano, M.1    Fukuzaki, H.2    Yoshida, M.3    Kumakura, M.4    Mashimo, T.5    Yuasa, H.6    Imai, K.7    Yamanaka, H.8    Suzuki, K.9
  • 4
    • 0030630036 scopus 로고    scopus 로고
    • Protein delivery from biodegradable microspheres
    • Cleland J.L. Protein delivery from biodegradable microspheres. Pharm. Biotechnol. 10:1997;1-43.
    • (1997) Pharm. Biotechnol. , vol.10 , pp. 1-43
    • Cleland, J.L.1
  • 7
    • 0029411935 scopus 로고
    • Synthesis and properties of novel block copolymers containing poly(lactic-glycolic acid) and poly(ethylene glycol) segments
    • Ferruti P., Penco M., D'Addato P., Ranucci E., Deghenghi R. Synthesis and properties of novel block copolymers containing poly(lactic-glycolic acid) and poly(ethylene glycol) segments. Biomaterials. 16:1995b;1423-1428.
    • (1995) Biomaterials , vol.16 , pp. 1423-1428
    • Ferruti, P.1    Penco, M.2    D'Addato, P.3    Ranucci, E.4    Deghenghi, R.5
  • 8
    • 0018737940 scopus 로고
    • Biodegradable polymers for use in surgery - Polyglycolic/poly(lactic acid) homo- and copolymers: 1
    • Gilding D.K., Reed A.M. Biodegradable polymers for use in surgery - polyglycolic/poly(lactic acid) homo- and copolymers: 1. Polymer. 20:1979;1459-1464.
    • (1979) Polymer , vol.20 , pp. 1459-1464
    • Gilding, D.K.1    Reed, A.M.2
  • 9
    • 0031845276 scopus 로고    scopus 로고
    • Controlled drug delivery by biodegradable poly(ester) devices: Different preparative approaches
    • Jain R., Shah N.H., Malick A.W., Rhodes C.T. Controlled drug delivery by biodegradable poly(ester) devices: different preparative approaches. Drug Develop. Ind. Pharm. 24:1998;703-727.
    • (1998) Drug Develop. Ind. Pharm. , vol.24 , pp. 703-727
    • Jain, R.1    Shah, N.H.2    Malick, A.W.3    Rhodes, C.T.4
  • 10
    • 0033844242 scopus 로고    scopus 로고
    • Controlled release of drugs from injectable in situ formed biodegradable PLGA microspheres: Effect of various formulation variables
    • Jain R., Rhodes C.T., Railkar A.M., Malick A.W., Shah N.H. Controlled release of drugs from injectable in situ formed biodegradable PLGA microspheres: effect of various formulation variables. Eur. J. Pharm. Biopharm. 50:2000;257-262.
    • (2000) Eur. J. Pharm. Biopharm. , vol.50 , pp. 257-262
    • Jain, R.1    Rhodes, C.T.2    Railkar, A.M.3    Malick, A.W.4    Shah, N.H.5
  • 11
    • 0025053154 scopus 로고
    • Biodegradable poly(lactic acid) and poly(lactide-co-glycolide) microspheres: Problems associated with preparative techniques and release properties
    • Jalid R., Nixon J.R. Biodegradable poly(lactic acid) and poly(lactide-co-glycolide) microspheres: problems associated with preparative techniques and release properties. J. Microencapsul. 7:1990;297-325.
    • (1990) J. Microencapsul. , vol.7 , pp. 297-325
    • Jalid, R.1    Nixon, J.R.2
  • 12
    • 0001855042 scopus 로고
    • Controlled release of bioactive agents from lactide/glycolide polymers
    • Chasin, M., Langer, R. (Eds.). Marcel Dekker, New York
    • Lewis, D.H., 1990. Controlled release of bioactive agents from lactide/glycolide polymers. In: Chasin, M., Langer, R. (Eds.), Biodegradable Polymers as Drug Delivery Systems. Marcel Dekker, New York, pp. 1-41.
    • (1990) Biodegradable Polymers as Drug Delivery Systems , pp. 1-41
    • Lewis, D.H.1
  • 13
    • 0032989754 scopus 로고    scopus 로고
    • Pulsatile release from subcutaneous implants
    • Medlicott N.J., Tucker I.G. Pulsatile release from subcutaneous implants. Adv. Drug Deliv. Rev. 38:1999;139-149.
    • (1999) Adv. Drug Deliv. Rev. , vol.38 , pp. 139-149
    • Medlicott, N.J.1    Tucker, I.G.2
  • 14
    • 0027235096 scopus 로고
    • Microencapsulation by coacervation of poly(lactide-co-glycolide): II. Encapsulation of a dispersed aqueous phase
    • Nihant N., Stassen S., Grandfils C., Jerôme R., Teyssié Ph. Microencapsulation by coacervation of poly(lactide-co-glycolide): II. Encapsulation of a dispersed aqueous phase. Polym. Int. 32:1993;171-176.
    • (1993) Polym. Int. , vol.32 , pp. 171-176
    • Nihant, N.1    Stassen, S.2    Grandfils, C.3    Jerôme, R.4    Teyssié, Ph.5
  • 15
    • 0028467817 scopus 로고
    • Microencapsulation by coacervation of poly(lactide-co-glycolide): III. Characterisation of the final microspheres
    • Nihant N., Stassen S., Grandfils C., Jérôme R., Teyssié Ph., Goffinet G. Microencapsulation by coacervation of poly(lactide-co-glycolide): III. Characterisation of the final microspheres. Polym. Int. 34:1994;289-299.
    • (1994) Polym. Int. , vol.34 , pp. 289-299
    • Nihant, N.1    Stassen, S.2    Grandfils, C.3    Jérôme, R.4    Teyssié, Ph.5    Goffinet, G.6
  • 16
    • 0029092709 scopus 로고
    • Microencapsulation by coacervation of poly(lactide-co-glycolide): IV. Effect of the processing parameters on coacervation and encapsulation
    • Nihant N., Grandfils C., Jérôme R., Teyssié Ph. Microencapsulation by coacervation of poly(lactide-co-glycolide): IV. Effect of the processing parameters on coacervation and encapsulation. J. Control. Rel. 35:1995;117-125.
    • (1995) J. Control. Rel. , vol.35 , pp. 117-125
    • Nihant, N.1    Grandfils, C.2    Jérôme, R.3    Teyssié, Ph.4
  • 17
    • 0343907187 scopus 로고    scopus 로고
    • One and three-month release injectable microspheres of the LH-RH superagonist leuprorelin acetate
    • Okada H. One and three-month release injectable microspheres of the LH-RH superagonist leuprorelin acetate. Adv. Drug Deliv. Rev. 28:1997;43-70.
    • (1997) Adv. Drug Deliv. Rev. , vol.28 , pp. 43-70
    • Okada, H.1
  • 18
    • 84986743677 scopus 로고
    • New high-molecular-weight poly(ester-carbonates) by chain extension of poly(lactic-glycolic acid)
    • Penco M., Ranucci E., Bignotti F., Ferruti P. New high-molecular-weight poly(ester-carbonates) by chain extension of poly(lactic-glycolic acid). Macromol. Rapid. Comm. 15:1994;683-690.
    • (1994) Macromol. Rapid. Comm. , vol.15 , pp. 683-690
    • Penco, M.1    Ranucci, E.2    Bignotti, F.3    Ferruti, P.4
  • 19
    • 0030207709 scopus 로고    scopus 로고
    • Degradation behaviour of block copolymers containing poly(lactic-glycolic acid) and poly(ethylene glycol) segments
    • Penco M., Marcioni S., Ferruti P., D'Antone S., Deghenghi R. Degradation behaviour of block copolymers containing poly(lactic-glycolic acid) and poly(ethylene glycol) segments. Biomaterials. 17:1996a;1583-1590.
    • (1996) Biomaterials , vol.17 , pp. 1583-1590
    • Penco, M.1    Marcioni, S.2    Ferruti, P.3    D'Antone, S.4    Deghenghi, R.5
  • 20
    • 0030142023 scopus 로고    scopus 로고
    • Poly(ester-carbonates) containing poly(lactic-glycolic acid) and poly(ethylene glycol) segments
    • Penco M., Becattini M., Ferruti P., D'Antone S., Deghenghi R. Poly(ester-carbonates) containing poly(lactic-glycolic acid) and poly(ethylene glycol) segments. Polym. Adv. Technol. 7:1996b;536-542.
    • (1996) Polym. Adv. Technol. , vol.7 , pp. 536-542
    • Penco, M.1    Becattini, M.2    Ferruti, P.3    D'Antone, S.4    Deghenghi, R.5
  • 21
    • 0025000345 scopus 로고
    • Influence of average molecular weights of poly(D,L-lactic acid-co-glycolic acid) copolymers 50/50 on phase separation and in vitro drug release from microspheres
    • Ruiz J.M., Busnel J.P., Benoit J.P. Influence of average molecular weights of poly(D,L-lactic acid-co-glycolic acid) copolymers 50/50 on phase separation and in vitro drug release from microspheres. Pharm. Res. 7:1990;928-934.
    • (1990) Pharm. Res. , vol.7 , pp. 928-934
    • Ruiz, J.M.1    Busnel, J.P.2    Benoit, J.P.3
  • 22
    • 0033368407 scopus 로고    scopus 로고
    • Effect of γ-irradiation on peptide-containing hydrophilic poly(D,L-lactide-co-glycolide) microspheres
    • Shameem M., Lee H., Burton K., Thanoo B.C., Deluca P.P. Effect of γ-irradiation on peptide-containing hydrophilic poly(D,L-lactide-co-glycolide) microspheres. PDA J. Pharm. Sci. Technol. 53:1999;309-313.
    • (1999) PDA J. Pharm. Sci. Technol. , vol.53 , pp. 309-313
    • Shameem, M.1    Lee, H.2    Burton, K.3    Thanoo, B.C.4    Deluca, P.P.5
  • 23
    • 0028375551 scopus 로고
    • Microencapsulation by coacervation of poly(lactide-co-glycolide): 1. Physico-chemical characteristics of the phase separation process
    • Stassen S., Nihant N., Martin V., Grandfils C., Jérome R., Teyssié Ph. Microencapsulation by coacervation of poly(lactide-co-glycolide): 1. Physico-chemical characteristics of the phase separation process. Polymer. 35:1994;777-785.
    • (1994) Polymer , vol.35 , pp. 777-785
    • Stassen, S.1    Nihant, N.2    Martin, V.3    Grandfils, C.4    Jérome, R.5    Teyssié, Ph.6
  • 28
    • 0025860213 scopus 로고
    • More about the degradation of LA/GA derived matrices in aqueous media
    • Vert M., Li S., Garreau H. More about the degradation of LA/GA derived matrices in aqueous media. J. Control. Rel. 16:1991;15-26.
    • (1991) J. Control. Rel. , vol.16 , pp. 15-26
    • Vert, M.1    Li, S.2    Garreau, H.3
  • 29
    • 0032509909 scopus 로고    scopus 로고
    • Influence of the microencapsulation method and peptide loading on poly(lactic acid) and poly(lactic-co-glycolic acid) degradation during in vitro testing
    • Witschi C., Doelker E. Influence of the microencapsulation method and peptide loading on poly(lactic acid) and poly(lactic-co-glycolic acid) degradation during in vitro testing. J. Control. Rel. 5:1998;327-341.
    • (1998) J. Control. Rel. , vol.5 , pp. 327-341
    • Witschi, C.1    Doelker, E.2
  • 30
    • 0003156346 scopus 로고
    • Preparation, characterisation, and drug delivery applications of microspheres based on biodegradable lactic/glycolic acid polymers
    • Wise, D.L., Trantolo, D.J., Altobelli, D.E., Yaszemski, M.J., Gresser, J.D., Schwartz, E.R. (Eds.). Marcel Dekker, New York
    • Wu, X.S., 1995a. Preparation, characterisation, and drug delivery applications of microspheres based on biodegradable lactic/glycolic acid polymers. In: Wise, D.L., Trantolo, D.J., Altobelli, D.E., Yaszemski, M.J., Gresser, J.D., Schwartz, E.R. (Eds.), Encyclopaedic Handbook of Biomaterials and Bioengineering. Marcel Dekker, New York, pp. 1015-1054.
    • (1995) Encyclopaedic Handbook of Biomaterials and Bioengineering , pp. 1015-1054
    • Wu, X.S.1
  • 31
    • 0003156346 scopus 로고
    • Preparation, characterisation, and drug delivery applications of microspheres based on biodegradable lactic/glycolic acid polymers
    • Wise, D.L., Trantolo, D.J., Altobelli, D.E., Yaszemski, M.J., Gresser, J.D., Schwartz, E.R. (Eds.). Marcel Dekker, New York
    • Wu, X.S., 1995b. Preparation, characterisation, and drug delivery applications of microspheres based on biodegradable lactic/glycolic acid polymers. In: Wise, D.L., Trantolo, D.J., Altobelli, D.E., Yaszemski, M.J., Gresser, J.D., Schwartz, E.R. (Eds.), Encyclopaedic Handbook of Biomaterials and Bioengineering. Marcel Dekker, New York, pp. 1151-1200.
    • (1995) Encyclopaedic Handbook of Biomaterials and Bioengineering , pp. 1151-1200
    • Wu, X.S.1
  • 32
    • 0025700105 scopus 로고
    • Preparation, characterization, and properties of polylactide (PLA)-poly(ethylene glycol) (PEG) copolymers: A potential drug carrier
    • Zhu K.J., Xiangzhou L., Shilin Y. Preparation, characterization, and properties of polylactide (PLA)-poly(ethylene glycol) (PEG) copolymers: a potential drug carrier. J. Appl. Polym. Sci. 39:1990;1-9.
    • (1990) J. Appl. Polym. Sci. , vol.39 , pp. 1-9
    • Zhu, K.J.1    Xiangzhou, L.2    Shilin, Y.3


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.