trans-Dihydroxypiperidines: Synthesis, Stereochemistry, and Anti-HIV Activity

Doklady Chemistry

Volumn 391, Issue 4-6, 2003, Pages 195-199

  Grishina, G V ^a   Borisenko, A A ^a   Nosan', Z G ^a   Veselov, I S ^a   Ashkinadze, L D ^a   Karamov, E V ^b   Kornilaeva, G V ^c   Zefirov, N S ^a  

^a MOSCOW STATE UNIVERSITY   (Russian Federation)

^b D I IVANOVSKY INSTITUTE OF VIROLOGY   (Russian Federation)

^c NONE

Author keywords

[No Author keywords available]

Indexed keywords

ANTI HUMAN IMMUNODEFICIENCY VIRUS AGENT; PIPERIDINE DERIVATIVE;

ARTICLE; CELL LINE; CHIRALITY; CONFORMATIONAL TRANSITION; CONTROLLED STUDY; DRUG CONFORMATION; DRUG STRUCTURE; DRUG SYNTHESIS; ENANTIOMER; HUMAN; HUMAN CELL; HUMAN IMMUNODEFICIENCY VIRUS; HUMAN IMMUNODEFICIENCY VIRUS INFECTION; PHARMACOPHORE; STEREOCHEMISTRY; T CELL LYMPHOMA; TRANS ISOMER;

EID: 0041879928     PISSN: 00125008     EISSN: None     Source Type: Journal    
DOI: 10.1023/A:1025307617288     Document Type: Article

References (15)

1. De Clercq, E., J. Med. Chem., 1995, vol. 38, pp. 2491-2497.
2. Fleet, G.W.J., Karpas, A., Dwek, R.A., et al., FEBS Lett., 1988, vol. 237, pp. 128-132.
3. Rajni Garg, Satya P. Gupta, Hua Gao, et al., Chem. Rev., 1999, vol. 99, pp. 3525-3601.
4. Polt, R., Sames, D., and Chruma, J., J. Org. Chem., 1999, vol. 64, pp. 6147-6158.
5. Pistia-Brueggeman, G. and Hollingsworth, R.I., Tetrahedron, 2001, vol. 57, pp. 8773-8778.
6. Grishina, G.V., Karamov, E.V., Kornilaeva, G.V., et al., RF Patent 2 198 658, Byull. Izobret., 2003, no. 5.
7. Maksimova, T.N., Mochalin, V.B., and Unkovskii, B.V., Khim. Geterotsikl. Soedin., 1980, no. 6, pp. 783-786.
8. Lukes, R., Collect. Czechosl. Chem. Commun., 1947, vol. 12, pp. 71-74.
9. Leonard, N.E. and Gash, V.W., J. Am. Chem. Soc., 1954, vol. 76, pp. 2781-2784.
10. Judin, L.G., Zh. Obshch. Khim., 1957, vol. 27, pp. 3021-3024.
11. Kost, A.N., Vest. Mosk. Univ., 1956, vol. 11, no. 1, pp. 209-211.
12. Oediger, H. and Joop, N., Justus Liebigs Ann. Chem., 1972, vol. 764, pp. 21-27.
13. Schmidle, C.J. and Mansfield, R.C., J. Am. Chem. Soc., 1956, vol. 78, pp. 425-428.
14. Chabrier, P., Najer, H., Giudicelli, M., and Joannic, M., Bull. Soc. Chim. France, 1957, vols. 11-12, pp. 1365-1369.
15. Terent'ev, P.B., Zil'bershtein, T.M., Borisenko, A.A., et al., Khim. Geterotsikl. Soedin., 2003.