Neat reaction of carboxylic acid methyl esters and amines for efficient parallel synthesis of scaffold amide libraries

Comptes Rendus Chimie

Volumn 6, Issue 5-6, 2003, Pages 631-633

  Machetti, Fabrizio ^a   Bucelli, Ilaria ^a   Indiani, Giovanni ^a   Guarna, Antonio ^a  

^a UNIVERSITY OF FLORENCE   (Italy)

Author keywords

Amides; Libraries; Neat reaction; Scaffold

Indexed keywords

AMIDE; AMINE; CARBOXYLIC ACID DERIVATIVE; ESTER;

ARTICLE; CHEMICAL REACTION; CHEMICAL STRUCTURE; CONTROLLED STUDY; HEATING; MOLECULAR LIBRARY; SYNTHESIS;

EID: 0041859456     PISSN: 16310748     EISSN: None     Source Type: Journal    
DOI: 10.1016/S1631-0748(03)00097-3     Document Type: Article

References (17)

1. Dolle R.E. Nelson K.H.J. J. Comb. Chem. 1 1999 235
2. Guarna A. Guidi A. Machetti F. Menchi G. Occhiato E.G. Scarpi D. Sisi S. Trabocchi A. J. Org. Chem. 64 1999 7347
3. Machetti F. Occhiato E.G. Menchi G. Scarpi D. Guarna A. PCT Int. Appl. 2001 WO 0164686
4. Guarna A. Bucelli I. Machetti F. Menchi G. Occhiato E G. Scarpi D. Trabocchi A. Tetrahedron 58 2002 9865
5. Pederson B.S. Sheibye S. Nilsson N.H. Lawesson S.-O. Bull. Soc. Chim. Belg. 87 1978 223
6. Russel P.B. J. Am. Chem. Soc. 72 1950 1853
7. Levi E.M. Mao C.L. Hauser C.R. Can. J. Chem. 47 1969 3761
8. Yang K.-W. Cannon J.G. Rose J.G. Tetrahedron Lett. 11 1970 1791
9. Houghton R.P. Williams C.S. Tetrahedron Lett. 8 1967 3929
10. Evans D.A. Tetrahedron Lett. 10 1969 1573
11. Chan H.-T. Wong L.T.L. J. Org. Chem. 34 1969 2766
12. Openshaw H.I. Wittaker N. J. Chem. Soc. C 1969 89
13. De Feo R.J. Strickler P.D. J. Org. Chem. 28 1963 2915
14. Wang W.-B. Roskamp E.J. J. Org. Chem. 57 1992 6101
15. Dolle R.E. Nicolaou K.C. J. Am. Chem. Soc. 107 1985 1695
16. Chou W.-C. Tan C.-W. Chen S.-F. Ku H. J. Org. Chem. 63 1998 10015
17. Altamura M. Canfarini F. Catalioto R.-M. Guidi A. Pasqui F. Renzetti A.R. Triolo A. Maggi C.A. Biorg. Med. Chem. Lett. 12 2002 2945