Strategy and tactics in combinatorial organic synthesis. Applications to drug discovery

Chimia

Volumn 51, Issue 11, 1997, Pages 821-825

  Gordon, Eric M ^a   Patel, Dinesh V ^b   Jacobs, Jeffrey W ^b   Gordeev, Mikhail F ^b   Zhou, Joseph ^b  

^a Versicor Inc   (United States)

^b NONE

Author keywords

[No Author keywords available]

Indexed keywords

EID: 0040685387     PISSN: 00094293     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article

References (19)

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2. M.A. Gallop, R.W. Barrett, W.J. Dower, S.P.A. Fodor, E.M. Gordon, J. Med. Chem. 1994, 37, 1233; E.M. Gordon, R.W. Barrett, W.J. Dower, S.P.A. Fodor, M.A. Gallop, ibid. 1994, 37, 1385.
3. E.M. Gordon, M.A. Gallop, D.V. Patel, Acc. Chem. Rese. 1996, 29, 144.
4. W. Carruthers, 'Cycloaddition Reactions in Organic Synthesis', Pergamon Press, Oxford, 1990.
5. For a review, see G.I. Georg, V.T. Ravikumar, in 'The Organic Chemistry of β-Lactams', Ed. G.I. Georg, Verlag Chemie, New York, 1993, p. 295-368.
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7. G.C. Look, C.P. Holmes, J.P. Chinn, M.A. Gallop, J. Org. Chem. 1994, 59, 7588; W.L. Fitch, G. Detre, C.P. Holmes, J.N. Shoolery, P.A. Keifer, ibid. 1994, 59, 7955.
8. G.C. Look, C.P. Holmes, J.P. Chinn, M.A. Gallop, J. Org. Chem. 1994, 59, 7588; W.L. Fitch, G. Detre, C.P. Holmes, J.N. Shoolery, P.A. Keifer, ibid. 1994, 59, 7955.
9. 'Solid Phase Synthesis of Beta-Sultams', M.F. Gordeev, E.M. Gordon, D.V. Patel, J. Org. Chem., in press.
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12. M.M. Murphy, J.R. Schullek, E.M. Gordon, M.A. Gallop, J. Am. Chem. Soc. 1995, 117, 7029.
13. M.F. Gordeev, D.V. Patel, E.M. Gordon, J. Org. Chem. 1996, 61, 924.
14. M.F. Gordeev, B. England, R.W. Barrett, E.M. Gordon, D.V. Patel, unpublished results.
15. M.F. Gordeev, D.V. Patel, J. Wu, E.M. Gordon, Tetrahedron Lett. 1996, 4643.
16. A. Atuegbu, D. Maclean, C. Nguyen, E.M. Gordon, J.W. Jacobs, Bioorg. Med. Chem. 1996, 4, 1097.
17. 'Cephalosporins and Penicillins; Chemistry and Biology', Ed. E.H. Flynn. Academic Press, New York, 1973.
18. 'Beta-Lactam Antibiotics; Chemistry and Biology', Eds. R.B. Morin and M. Gorman. Academic Press, New York, 1982, Vol. 1-3.
19. J. Zhou, J. W. Jacobs, unpublished observations.