Redefining the structure-activity relationships of 2,6-methano-3-benzazocines. Part 2: 8-Formamidocyclazocine analogues

Bioorganic and Medicinal Chemistry Letters

Volumn 13, Issue 11, 2003, Pages 1911-1914

  Wentland, Mark P ^a   Sun, Xufeng ^a   Ye, Yingchun ^a   Lou, Rongliang ^a   Bidlack, Jean M ^b  

^a Research Rensselaer Polytechnic Institute   (United States)

^b UNIVERSITY OF ROCHESTER SCHOOL OF MEDICINE AND DENTISTRY   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

BENZAZOCINE DERIVATIVE; CYCLAZOCINE; KAPPA OPIATE RECEPTOR; MU OPIATE RECEPTOR;

ANTINOCICEPTION; ARTICLE; CONTROLLED STUDY; DRUG RECEPTOR BINDING; DRUG SELECTIVITY; DRUG SYNTHESIS; ENANTIOMER; MOUSE; NONHUMAN; STRUCTURE ACTIVITY RELATION; SUBSTITUTION REACTION;

EID: 0038732519     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-894X(03)00295-6     Document Type: Article

References (22)

1. Part I: Wentland M.P., Lou R., Ye Y., Cohen D.J., Richardson G.P., Bidlack J.M. Bioorg. Med. Chem. Lett. 11:2001;623.
2. Bidlack J.M., Cohen D.J., McLaughlin J.P., Lou R., Ye Y., Wentland M.P. J. Pharmacol. Exp. Ther. 302:2002;374.
3. Archer S., Glick S.D., Bidlack J.M. Neurochem. Res. 21:1996;1369.
4. Wentland M.P., Lou R., Dehnhardt C.M., Duan W., Cohen D.J., Bidlack J.M. Bioorg. Med. Chem. Lett. 11:2001;1717.
5. Wentland, M. P.; Lou, R.; Dehnhardt, C.; Cohen, D. J.; Bidlack, J. M. Abstracts of Papers, Proceedings of the 64th Annual Meeting of the College on Problems of Drug Dependence, Québec City, Québec, Canada, June 8-13, 2002; p 724 [Abstract also published in: Alcohol Drug Depend, 2002, 66 (Suppl. 1) S192].
6. Aldrich, J. V. In Burger's Medicinal Chemistry and Drug Discovery; Wolff, M. E., Ed.; John Wiley & Sons: New York, 1996; Vol. 3, p 321.
7. Patani G.A., LaVoie E.J. Chem. Rev. 96:1996;3147.
8. Wentland M.P., Albertson N.F., Pierson A.K. J. Med. Chem. 23:1980;71.
9. Danso-Danquah R., Bai X., Zhang X., Mascarella S.W., Williams W., Sine B., Bowen W.D., Carroll F.I. J. Med. Chem. 38:1995;2978.
10. Carter, A.; Ensinger, H.; Grauert, M.; Kuhn, F. J.; Merz, H.; Mueller, E.; Stransky, W.; Streller, I. Eur. Pat. Appl. 521422, 1993; Chem. Abstr. 1993, 119, 117602.
11. Vyas D., Joshi Y.C., Joshi B.C. J. Inst. Chem. (India). 54:1982;213.
12. McCurdy C.R., Jones R.M., Portoghese P.S. Org. Lett. 2:2000;819.
13. Allen, R. C.; Wettlaufer, D. G. US Patent 4,929,622, 1990; Chem. Abstr. 1990, 113, 212033.
14. Newman A.H., Bevan K., Bowery N., Tortella F.C. J. Med. Chem. 35:1992;4135.
15. (a) Wentland M.P., Ye Y., Cioffi C.L., Lou R., Zhou Q., Xu G., Duan W., Dehnhardt C.M., Sun X., Cohen D.J., Bidlack J.M. J. Med. Chem. 46:2003;838.
16. (b) Wentland M.P., Xu G., Cioffi C.L., Ye Y., Duan W., Cohen D.J., Colasurdo A.M., Bidlack J.M. Bioorg. Med. Chem. Lett. 10:2000;183.
17. (a) Michne W.F., Albertson N.F. J. Med. Chem. 15:1972;1278 (b) Albertson, N. F. US Patent 4,161,598, 1979; Chem. Abstr. 1979, 91, 175227.
18. (a) Michne W.F., Albertson N.F. J. Med. Chem. 15:1972;1278 (b) Albertson, N. F. US Patent 4,161,598, 1979; Chem. Abstr. 1979, 91, 175227.
19. Chakrabarty M., Khasnobis S., Harigaya Y., Konda Y. Syn. Commun. 30:2000;187.
20. Huang X.H., Buchwald S.L. Org. Lett. 3:2001;3417.
21. Archer S., Seyed-Mozaffari A., Jiang Q., Bidlack J.M. J. Med. Chem. 37:1994;1578.
22. Hansch, C.; Leo, A.; Hoekman, D. In Exploring QSAR: Hydrophobic, Electronic, and Steric Constants; American Chemical Society: Washington, 1995; p 217.