메뉴 건너뛰기




Volumn 307, Issue 2, 2003, Pages 315-321

Suspensions of pro-drug insulin greatly prolong normoglycemic patterns in diabetic rats

Author keywords

Diabetes; FMS3 insulin; Glucose lowering profiles; Long acting insulin; Normoglycemia; Prodrug insulin

Indexed keywords

(2 SULFO 9 FLUORENYLMETHOXYCARBONYL) 3 INSULIN; ANTIDIABETIC AGENT; INSULIN DERIVATIVE; ISOPHANE INSULIN; PRODRUG; PROTAMINE; UNCLASSIFIED DRUG; ZINC ION;

EID: 0038690338     PISSN: 0006291X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0006-291X(03)01200-2     Document Type: Article
Times cited : (6)

References (31)
  • 1
    • 0003058777 scopus 로고    scopus 로고
    • Insulin therapy
    • K.G.M.M. Albert, P. Zimmet, & R.A. Defronzo. Chichester, UK: Wiley
    • Home P.D. Insulin therapy. Albert K.G.M.M., Zimmet P., Defronzo R.A. The International Textbook of Diabetes. second ed. 1996;899-928 Wiley, Chichester, UK.
    • (1996) The International Textbook of Diabetes second ed. , pp. 899-928
    • Home, P.D.1
  • 2
    • 0000588546 scopus 로고
    • Crystaline and amorphous insulin-zinc compounds with prolonged action
    • Hallas-Moller K., Peterson K., Schlichtrull J. Crystaline and amorphous insulin-zinc compounds with prolonged action. Science. 116:1952;394-399.
    • (1952) Science , vol.116 , pp. 394-399
    • Hallas-Moller, K.1    Peterson, K.2    Schlichtrull, J.3
  • 3
    • 0020131685 scopus 로고
    • Evaluation of adenosine and related nucleosides as physiological regulators in adipose tissue
    • Shechter Y. Evaluation of adenosine and related nucleosides as physiological regulators in adipose tissue. Endocrinology. 110:1982;1579-1583.
    • (1982) Endocrinology , vol.110 , pp. 1579-1583
    • Shechter, Y.1
  • 4
    • 0020410062 scopus 로고
    • Evaluation of factors responsible for the inability of insulin to antagonize lipolysis due to high concentrations of catecholamines
    • Shechter Y., Reitman P., Hizi A. Evaluation of factors responsible for the inability of insulin to antagonize lipolysis due to high concentrations of catecholamines. Biochem. Biophys. Res. Commun. 109:1982;776-785.
    • (1982) Biochem. Biophys. Res. Commun. , vol.109 , pp. 776-785
    • Shechter, Y.1    Reitman, P.2    Hizi, A.3
  • 5
    • 0006178809 scopus 로고
    • The endocrine pancreas and diabetes mellitus
    • R.H. Williams. Philadelphia: W.B. Saunders
    • Porte D. Jr., Halter J.B. The endocrine pancreas and diabetes mellitus. Williams R.H. Textbook of Endocrinology. sixth ed. 1981;716-743 W.B. Saunders, Philadelphia.
    • (1981) Textbook of Endocrinology sixth ed. , pp. 716-743
    • Porte D., Jr.1    Halter, J.B.2
  • 6
    • 0002680280 scopus 로고
    • Insulin, oral hypoglycemic agents and the pharmacology of the endocrine pancreas
    • A.G. Gilman, T.W. Rall, A.S. Nies, & P. Taylor. New York/Oxford: Pergamon Press
    • Kahn C.R., Shehcter Y. Insulin, oral hypoglycemic agents and the pharmacology of the endocrine pancreas. Gilman A.G., Rall T.W., Nies A.S., Taylor P. Goodman and Gilman Handbook of Pharmacology. 1990;1463-1495 Pergamon Press, New York/Oxford.
    • (1990) Goodman and Gilman Handbook of Pharmacology , pp. 1463-1495
    • Kahn, C.R.1    Shehcter, Y.2
  • 7
    • 0021692099 scopus 로고
    • From glycogen to ketones and back
    • Foster D.W. From glycogen to ketones and back. Diabetes. 33:1984;1188-1199.
    • (1984) Diabetes , vol.33 , pp. 1188-1199
    • Foster, D.W.1
  • 8
    • 0002096610 scopus 로고    scopus 로고
    • Insulin, oral hypoglycemic agents and the pharmacology of the endocrine pancreas
    • J.G. Handman, L.E. Limbial, P.B. Molinoff, & R.W. Ruddon. New York: Pergamon Press
    • Davis S.N., Granner D.K. Insulin, oral hypoglycemic agents and the pharmacology of the endocrine pancreas. Handman J.G., Limbial L.E., Molinoff P.B., Ruddon R.W. Goodman and Gilman. The Pharmacological Basis of Therapeutics. ninth ed. 1996;1487-1517 Pergamon Press, New York.
    • (1996) Goodman and Gilman. The Pharmacological Basis of Therapeutics ninth ed. , pp. 1487-1517
    • Davis, S.N.1    Granner, D.K.2
  • 9
    • 0025913586 scopus 로고
    • Subcutaneous absorption of insulin in insulin-dependent diabetic patients
    • Hildebrant P. Subcutaneous absorption of insulin in insulin-dependent diabetic patients. Dan. Med. Bull. 38:1991;337-346.
    • (1991) Dan. Med. Bull. , vol.38 , pp. 337-346
    • Hildebrant, P.1
  • 10
    • 0030981739 scopus 로고    scopus 로고
    • Pharmacokinetic considerations of new insulin formulations and routes of administration
    • Hoffman A., Ziv E. Pharmacokinetic considerations of new insulin formulations and routes of administration. Clin. Pharmacokinet. 33:1997;285-301.
    • (1997) Clin. Pharmacokinet. , vol.33 , pp. 285-301
    • Hoffman, A.1    Ziv, E.2
  • 11
    • 0032819174 scopus 로고    scopus 로고
    • Insulin analogues and their potential in the management of diabetes mellitus
    • Bolli G.B., DiMarchi R.D., Park G.D., Pramming S., Koivisto V.A. Insulin analogues and their potential in the management of diabetes mellitus. Diabetologia. 42:1999;1151-1167.
    • (1999) Diabetologia , vol.42 , pp. 1151-1167
    • Bolli, G.B.1    DiMarchi, R.D.2    Park, G.D.3    Pramming, S.4    Koivisto, V.A.5
  • 12
    • 0028092036 scopus 로고
    • Improving insulin therapy: Achievements and challenges
    • Galloway J.A., Chance R.E. Improving insulin therapy: achievements and challenges. Horm. Metab. Res. 26:1994;591-608.
    • (1994) Horm. Metab. Res. , vol.26 , pp. 591-608
    • Galloway, J.A.1    Chance, R.E.2
  • 13
    • 0038258356 scopus 로고
    • Insulin treatment and diabetes; Half a century of therapeutic misadventure?
    • W.M.G. Tanbridge. Bath, UK: Pitman
    • Albert K.G.M.M. Insulin treatment and diabetes; half a century of therapeutic misadventure? Tanbridge W.M.G. Advanced Medicine. 1981;1-13 Pitman, Bath, UK.
    • (1981) Advanced Medicine , pp. 1-13
    • Albert, K.G.M.M.1
  • 15
    • 0024413243 scopus 로고
    • Effect of raising injection site temperature on isophane insulin crystal dissociation
    • Thow J.C., Johnston A.B. Effect of raising injection site temperature on isophane insulin crystal dissociation. Diabetes Care. 12:1989;432-434.
    • (1989) Diabetes Care , vol.12 , pp. 432-434
    • Thow, J.C.1    Johnston, A.B.2
  • 16
    • 0019943337 scopus 로고
    • Absorption of isophane (NPH) insulin and its clinical implications
    • Lauritzen T., Pramming S., Gale E., Deckert T., Binder C. Absorption of isophane (NPH) insulin and its clinical implications. Br. Med. J. 285:1982;159-162.
    • (1982) Br. Med. J. , vol.285 , pp. 159-162
    • Lauritzen, T.1    Pramming, S.2    Gale, E.3    Deckert, T.4    Binder, C.5
  • 17
    • 0030754515 scopus 로고    scopus 로고
    • Intensified insulin therapy and the risk of severe hypolycaemia
    • Bolt S., Bolt U., Berger M., Mulhauser I. Intensified insulin therapy and the risk of severe hypolycaemia. Diabetologia. 40:1997;926-932.
    • (1997) Diabetologia , vol.40 , pp. 926-932
    • Bolt, S.1    Bolt, U.2    Berger, M.3    Mulhauser, I.4
  • 18
    • 0031794057 scopus 로고    scopus 로고
    • Risk factors of severe hypoglycaemia in adult patients with Type I diabetes - a prospective population based study
    • Muhlhauser I., Overmann H., Bender R., Bolt V., Berger M. Risk factors of severe hypoglycaemia in adult patients with Type I diabetes - a prospective population based study. Diabetologia. 41:1998;1274-1282.
    • (1998) Diabetologia , vol.41 , pp. 1274-1282
    • Muhlhauser, I.1    Overmann, H.2    Bender, R.3    Bolt, V.4    Berger, M.5
  • 19
    • 0032991564 scopus 로고    scopus 로고
    • New concept for long-acting insulin. Spontaneous conversion of inactive modified insulin to the active hormone in circulation; 9-fluorenylmethoxycarbonyl derivative of insulin
    • Gershonov E., Shechter Y., Fridkin M. New concept for long-acting insulin. Spontaneous conversion of inactive modified insulin to the active hormone in circulation; 9-fluorenylmethoxycarbonyl derivative of insulin. Diabetes. 48:1999;1437-1442.
    • (1999) Diabetes , vol.48 , pp. 1437-1442
    • Gershonov, E.1    Shechter, Y.2    Fridkin, M.3
  • 22
    • 0034762854 scopus 로고    scopus 로고
    • A new concept for prolonging the half-life of peptides, proteins, and low molecular weight drugs in vivo
    • Shechter Y., Goldwaser I., Lavon I.et al. A new concept for prolonging the half-life of peptides, proteins, and low molecular weight drugs in vivo. Drug. Future. 26:2001;669-676.
    • (2001) Drug. Future , vol.26 , pp. 669-676
    • Shechter, Y.1    Goldwaser, I.2    Lavon, I.3
  • 23
    • 0024062933 scopus 로고
    • Insulin-degradation: Mechanism, products, and significance
    • Duckworth W.C. Insulin-degradation: mechanism, products, and significance. Endocr. Rev. 9:1988;319-345.
    • (1988) Endocr. Rev. , vol.9 , pp. 319-345
    • Duckworth, W.C.1
  • 24
    • 0000110345 scopus 로고
    • 9-(2-Sulfo)fluorenylmethoxy carbonyl chloride, a new reagent for the purification of synthetic peptides
    • Merrifield R.B., Bach A.E. 9-(2-Sulfo)fluorenylmethoxy carbonyl chloride, a new reagent for the purification of synthetic peptides. J. Org. Chem. 43:1978;4808-4816.
    • (1978) J. Org. Chem. , vol.43 , pp. 4808-4816
    • Merrifield, R.B.1    Bach, A.E.2
  • 25
    • 0023219921 scopus 로고
    • Oral administration of vanadate normalizes blood glucose levels in streptozotocin-treated rats
    • Meyerovitch J., Farfel Z., Sack Y., Shechter Y. Oral administration of vanadate normalizes blood glucose levels in streptozotocin-treated rats. J. Biol. Chem. 262:1987;6658-6662.
    • (1987) J. Biol. Chem. , vol.262 , pp. 6658-6662
    • Meyerovitch, J.1    Farfel, Z.2    Sack, Y.3    Shechter, Y.4
  • 26
    • 77956751025 scopus 로고
    • Insulin: The structure in the crystal and its reflection in chemistry and biology
    • Blundell T., Dodson G., Hodgkin D., Mercola D. Insulin: the structure in the crystal and its reflection in chemistry and biology. Adv. Protein Chem. 26:1972;279-402.
    • (1972) Adv. Protein Chem. , vol.26 , pp. 279-402
    • Blundell, T.1    Dodson, G.2    Hodgkin, D.3    Mercola, D.4
  • 28
    • 0037920808 scopus 로고
    • The effect of various substances on the action of insulin
    • Fisher A.M., Scott D.A. The effect of various substances on the action of insulin. J. Pharmacol. 58:1936;93-104.
    • (1936) J. Pharmacol. , vol.58 , pp. 93-104
    • Fisher, A.M.1    Scott, D.A.2
  • 29
    • 0018379923 scopus 로고
    • Effect of streptozotocin-diabetes on insulin binding, glucose transport, and intracellular glucose metabolism in isolated rat adipocytes
    • Kobayashi M., Olefsky J.M. Effect of streptozotocin-diabetes on insulin binding, glucose transport, and intracellular glucose metabolism in isolated rat adipocytes. Diabetes. 28:1979;95-97.
    • (1979) Diabetes , vol.28 , pp. 95-97
    • Kobayashi, M.1    Olefsky, J.M.2
  • 30
    • 0033543662 scopus 로고    scopus 로고
    • L-Glutamic acid ( γ) -monohydroxamate; A potentiator of vanadium-evoked glucose metabolism in vitro and in vivo
    • Goldwaser I., Li J., Gershonov E., Armoni M., Karnieli E., Fridkin M., Shechter Y. L-Glutamic acid (. γ) -monohydroxamate; a potentiator of vanadium-evoked glucose metabolism in vitro and in vivo J. Biol. Chem. 274:1999;26617-26624.
    • (1999) J. Biol. Chem. , vol.274 , pp. 26617-26624
    • Goldwaser, I.1    Li, J.2    Gershonov, E.3    Armoni, M.4    Karnieli, E.5    Fridkin, M.6    Shechter, Y.7
  • 31
    • 0025060803 scopus 로고
    • Perspective in diabetes; Insulin-mimetic effects of vanadate: Possible implications for future treatment of diabetes
    • Shechter Y. Perspective in diabetes; insulin-mimetic effects of vanadate: possible implications for future treatment of diabetes. Diabetes. 39:1990;1-5.
    • (1990) Diabetes , vol.39 , pp. 1-5
    • Shechter, Y.1


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.