From the DNA gyrase inhibitor cyclothialidine to a new class of antibacterial agents

Chimia

Volumn 57, Issue 4, 2003, Pages 184-186

  Goetschi, Erwin ^a   Angehrn, Peter ^b   Gmuender, Hans ^b   Hebeisen, Paul ^b   Kostrewa, Dirk ^b   Link, Helmut ^b   Luebbers, Thomas ^b   Masciadri, Raffaello ^b   Reindl, Peter ^b   Ricklin, Fabienne ^b   Theil, Frank Peter ^b  

^a F HOFFMANN LA ROCHE LTD   (Switzerland)

^b NONE

Author keywords

Antibacterials; Cyclothialidine; DNA gyrase inhibitor; Natural products

Indexed keywords

ANTIINFECTIVE AGENT; CIPROFLOXACIN; CYCLOTHIALIDINE; DNA TOPOISOMERASE (ATP HYDROLYSING); GYRASE INHIBITOR; NOVOBIOCIN; RO 091437; UNCLASSIFIED DRUG; VANCOMYCIN;

BACTERIAL GROWTH; BACTERIAL STRAIN; CHEMICAL MODIFICATION; CONFERENCE PAPER; DRUG EFFICACY; DRUG IDENTIFICATION; DRUG MECHANISM; DRUG POTENCY; DRUG SCREENING; DRUG STRUCTURE; ENZYME ISOLATION; GRAM NEGATIVE BACTERIUM; GRAM POSITIVE BACTERIUM; GROWTH INHIBITION; NONHUMAN; STRUCTURE ACTIVITY RELATION;

EID: 0038582387     PISSN: 00094293     EISSN: None     Source Type: Journal    
DOI: 10.2533/000942903777679505     Document Type: Conference Paper

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