Synthesis and activity of novel benzoxazole derivatives of mannopeptimycin glycopeptide antibiotics

Bioorganic and Medicinal Chemistry Letters

Volumn 13, Issue 15, 2003, Pages 2607-2610

  Sum, Phaik Eng ^a   How, David ^a   Torres, Nancy ^a   Newman, Howard ^a   Petersen, Peter J ^a   Mansour, Tarek S ^a  

^a WYETH RESEARCH   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

ALDEHYDE; AMINOPHENOL; ANTIBIOTIC AGENT; ANTIINFECTIVE AGENT; BENZOXAZOLE DERIVATIVE; DYES, REAGENTS, INDICATORS, MARKERS AND BUFFERS; GLYCOPEPTIDE; MANNOPEPTIMYCIN GLYCOPEPTIDE; POLYPEPTIDE ANTIBIOTIC AGENT;

ANTIMICROBIAL ACTIVITY; ARTICLE; DRUG EFFECT; DRUG SYNTHESIS; ELECTROSPRAY MASS SPECTROMETRY; ENTEROCOCCUS; GRAM NEGATIVE BACTERIUM; GRAM POSITIVE BACTERIUM; HIGH PERFORMANCE LIQUID CHROMATOGRAPHY; IN VITRO STUDY; MICROBIOLOGICAL EXAMINATION; MINIMUM INHIBITORY CONCENTRATION; NONHUMAN; PHYSICAL CHEMISTRY; STAPHYLOCOCCUS AUREUS; STREPTOCOCCUS; STRUCTURE ACTIVITY RELATION; SYNTHESIS;

EID: 0038495948     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-894X(03)00512-2     Document Type: Article

References (10)

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4. (b) He H., Williamson R.T., Shen B., Graziani E.I., Yang H.Y., Sakya S.M., Petersen P.J., Carter G.T. J. Am. Chem. Soc. 124:2002;9729.
5. Petersen, P. J.; Weiss, W. J.; Lenoy, E. B.; He, H.; Testa, R. T.; Bradford, P. A. 41st Interscience Conference on Antimicrobial Agents and Chemotherapy, Chicago, IL, Dec 16-19, 2001; abstract F-1148.
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8. 2+.
9. 2+.
10. 2+.