Molecular characterization of specific H1-receptor agonists histaprodifen and its Nα-substituted analogues on bovine aortic H1-receptors

Naunyn-Schmiedeberg's Archives of Pharmacology

Volumn 367, Issue 5, 2003, Pages 538-546

  Čarman Kržan, Marija ^a   Bavec, Aljoša ^a   Zorko, Matjaž ^a   Schunack, Walter ^b  

^a UNIVERSITY OF LJUBLJANA   (Slovenia)

^b FREIE UNIVERSITÄT BERLIN   (Germany)

Author keywords

Cardiovascular system; G proteins; H1 receptor agonists; Histaprodifens

Indexed keywords

DIMETHYLHISTAPRODIFEN; GUANINE NUCLEOTIDE BINDING PROTEIN; GUANOSINE 5' O (3 THIOTRIPHOSPHATE); GUANOSINE TRIPHOSPHATASE; GUANOSINE TRIPHOSPHATE; HISTAMINE; HISTAMINE H1 RECEPTOR; HISTAMINE H1 RECEPTOR AGONIST; HISTAMINE H1 RECEPTOR ANTAGONIST; HISTAPRODIFEN; MEPYRAMINE; METHYLHISTAPRODIFEN; SUPRAHISTAPRODIFEN; TRIPROLIDINE; TRITIUM; UNCLASSIFIED DRUG;

ANIMAL TISSUE; ARTICLE; BINDING COMPETITION; CATTLE; CONTROLLED STUDY; DISSOCIATION CONSTANT; DRUG BINDING SITE; DRUG POTENCY; DRUG RECEPTOR BINDING; DRUG STRUCTURE; MALE; NONHUMAN; RECEPTOR AFFINITY; THORACIC AORTA; VASCULAR SMOOTH MUSCLE;

ANIMALS; AORTA, THORACIC; BINDING SITES; CATTLE; GTP-BINDING PROTEINS; GTPASE-ACTIVATING PROTEINS; HISTAMINE; HISTAMINE AGONISTS; MALE; PROTEIN BINDING; PYRILAMINE; RECEPTORS, HISTAMINE H1; STRUCTURE-ACTIVITY RELATIONSHIP; TRITIUM;

EID: 0038119922     PISSN: 00281298     EISSN: None     Source Type: Journal    
DOI: 10.1007/s00210-003-0702-y     Document Type: Article

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