Histaprodifen, methylhistaprodifen, and dimethylhistaprodifen are potent H1-receptor agonists in the pithed and in the anaesthetized rat

Naunyn-Schmiedeberg's Archives of Pharmacology

Volumn 359, Issue 1, 1999, Pages 11-16

  Malinowska, B ^a   Piszcz, J ^a   Schlicker, E ^b   Kramer, K ^c   Elz, S ^c   Schunack, W ^c  

^a MEDICAL UNIVERSITY OF BIALYSTOK   (Poland)

^b UNIVERSITY OF BONN   (Germany)

^c FREIE UNIVERSITÄT BERLIN   (Germany)

Author keywords

2 (2 Thiazolyl)ethanamine; Anaesthetized rats; Dimethylhistaprodifen; Dimetindene; H1 receptor agonists; Histaprodifen; Methylhistaprodifen; Pithed rats

Indexed keywords

2 (2 THIAZOLYL)ETHYLAMINE; DIMETHYLHISTAPRODIFEN; DIMETINDENE; HISTAMINE AGONIST; HISTAMINE H1 RECEPTOR; HISTAPRODIFEN; METHYLHISTAPRODIFEN; N(G) NITROARGININE METHYL ESTER; PRAZOSIN; PROPRANOLOL; RANITIDINE; RAUWOLSCINE; THIOPERAMIDE; UNCLASSIFIED DRUG;

ANIMAL EXPERIMENT; ARTICLE; CONTROLLED STUDY; DEPRESSOR RESPONSE; DIASTOLIC BLOOD PRESSURE; DOSE RESPONSE; DRUG EFFECT; DRUG MECHANISM; DRUG RECEPTOR BINDING; INTRAPERITONEAL DRUG ADMINISTRATION; INTRAVENOUS DRUG ADMINISTRATION; MALE; NONHUMAN; RAT; RECEPTOR AFFINITY; RECEPTOR BLOCKING; RECEPTOR OCCUPANCY; RECEPTOR SENSITIVITY; SPINAL ANIMAL;

EID: 0032996710     PISSN: 00281298     EISSN: None     Source Type: Journal    
DOI: 10.1007/PL00005316     Document Type: Article

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