N-[18F]fluoroethyl-4-piperidyl acetate ([18F]FEtP4A): A PET tracer for imaging brain acetylcholinesterase in vivo

Bioorganic and Medicinal Chemistry

Volumn 11, Issue 12, 2003, Pages 2519-2527

  Zhang, Ming Rong ^a,b   Furutsuka, Kenji ^a,b   Maeda, Jun ^a,b   Kikuchi, Tatsuya ^a,c   Kida, Takayo ^a,b   Okauchi, Takashi ^a,b   Irie, Toshiaki ^a   Suzuki, Kazutoshi ^a  

^a NATIONAL INSTITUTE OF RADIOLOGICAL SCIENCES   (Japan)

^b 141 0032   (Japan)

^c CHIBA UNIVERSITY   (Japan)

Author keywords

[No Author keywords available]

Indexed keywords

ACETYLCHOLINESTERASE; N FLUOROETHYL 4 PIPERIDYLACETATE F 18; TRACER; UNCLASSIFIED DRUG; ACETIC ACID DERIVATIVE; CARBON; DIAGNOSTIC AGENT; FLUORINE; N FLUOROETHYL 4 PIPERIDYL ACETATE; N METHYL 4 PIPERIDYL ACETATE; N-FLUOROETHYL-4-PIPERIDYL ACETATE; N-METHYL-4-PIPERIDYL ACETATE; PIPERIDINE DERIVATIVE; RADIOPHARMACEUTICAL AGENT;

ANIMAL TISSUE; ARTICLE; AUTORADIOGRAPHY; BLOOD BRAIN BARRIER; BRAIN; CEREBELLUM; CHEMICAL REACTION; CONTROLLED STUDY; CORPUS STRIATUM; DRUG DISTRIBUTION; DRUG HYDROLYSIS; FRONTAL CORTEX; HIGH PERFORMANCE LIQUID CHROMATOGRAPHY; HYDROPHILICITY; IMAGE DISPLAY; MALE; METABOLITE; MONKEY; NONHUMAN; PLASMA; POSITRON EMISSION TOMOGRAPHY; RADIOACTIVITY; RAT; REACTION TIME; ANIMAL; COMPARATIVE STUDY; COMPUTER ASSISTED EMISSION TOMOGRAPHY; ENZYMOLOGY; HYDROLYSIS; MACACA; METABOLISM; SCINTISCANNING; SENSITIVITY AND SPECIFICITY; SYNTHESIS;

PRIMATES;

ACETATES; ACETYLCHOLINESTERASE; ANIMALS; AUTORADIOGRAPHY; BRAIN; CARBON RADIOISOTOPES; FLUORINE RADIOISOTOPES; HYDROLYSIS; MACACA MULATTA; MALE; PIPERIDINES; RADIOPHARMACEUTICALS; RATS; SENSITIVITY AND SPECIFICITY; TOMOGRAPHY, EMISSION-COMPUTED;

EID: 0037659282     PISSN: 09680896     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0968-0896(03)00177-9     Document Type: Article

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