Increasing the inhibitory potency of L-arabino-imidazolo-[1,2]-piperidinose towards β-D-glucosidase and β-D-galactosidase

Tetrahedron Letters

Volumn 44, Issue 18, 2003, Pages 3667-3670

  Dubost, Estelle ^a   Tschamber, Théophile ^a   Streith, Jacques ^a  

^a UNIVERSITÉ DE HAUTE ALSACE   (France)

Author keywords

Azasugars; Glycosidase inhibitors; Imidazolo piperidinoses

Indexed keywords

ARABINOIMIDAZOLO[1,2]PIPERIDINOSE; BETA GALACTOSIDASE; BETA GLUCOSIDASE; PIPERIDINE DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; DRUG SYNTHESIS; ENZYME INHIBITION;

EID: 0037471472     PISSN: 00404039     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0040-4039(03)00696-8     Document Type: Article

References (10)

1. Lillelund V.H., Jensen H.H., Liang X., Bols M. Chem. Rev. 102:2002;515-553.
2. Gessier F., Tschamber T., Tarnus C., Neuburger M., Huber W., Streith J. Eur. J. Org. Chem. 2001;4111-4125.
3. Aoyagi T., Suda H., Uotani K., Kojima F., Aoyama T., Horiguchi K., Hamada M., Takeuchi T. J. Antibiot. 45:1992;1404-1408.
4. Aoyama T., Naganawa H., Suda H., Uotani K., Aoyagi T., Takeuchi T. J. Antibiot. 45:1992;1557-1558.
5. Panday N., Canac Y., Vasella A. Helv. Chim. Acta. 83:2000;58-79.
6. Sonogashira K., Tohda Y., Hagihara N. Tetrahedron Lett. 16:1975;4467-4470.
7. Rothenberg A.S., Dauplaise D.L., Panzer H.P. Angew. Chem., Int. Ed. 22:1983;560.
8. Schaumann, E. E. Houben-Weyl, Methoden der organischen Chemie, E8c, Georg Thieme Verlag: Stuttgart, New York, 1994; pp. 1-215.
9. Iddon B. Heterocycles. 23:1985;417-443.
10. Panday N., Vasella A. Synthesis. 1999;1459-1468.