A general approach toward the synthesis of 8-acylamidopyrazolo[1,5-a]-1,3,5-triazines

Tetrahedron Letters

Volumn 44, Issue 4, 2003, Pages 703-705

  Raboisson, Pierre ^a,c   Schultz, Dominique ^a   Lugnier, Claire ^b   Mathieu, Romain ^a   Bourguignon, Jean Jacques ^a  

^a Laboratoire de Pharmacochimie   (France)

^b UNIVERSITÉ DE STRASBOURG   (France)

^c JOHNSON AND JOHNSON   (United States)

Author keywords

Activating group; Adenine; Bioisoster; Pyrazolo 1,5 a 1,3,5 triazine

Indexed keywords

8 ACYLAMIDOPYRAZOLO[1,5 A] 1,3,5 TRIAZINE; 8 AMINO 4 [N (4 AMINOPHENYL) N (METHYL)AMINO]PYRAZOLO[1,5 A] 1,3,5 TRIAZINE; AMINE; TRIAZINE DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; CHEMICAL STRUCTURE; SYNTHESIS;

EID: 0037454985     PISSN: 00404039     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0040-4039(02)02661-8     Document Type: Article

References (10)

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8. 4: C, 47.42; H, 3.37; N, 29.78. Found: C, 47.56; H, 3.54; N, 29.79.
9. 7: C, 57.98; H, 5.61; N, 36.41. Found: C, 57.88; H, 5.58; N, 36.63.
10. 6O: C, 49.08; H, 5.49; N, 38.16. Found: C, 49.27; H, 5.19; N, 38.02.