Synthesis, characterization, and molecular structure of a gallium(III) complex of an amine-phenol ligand with activity against chloroquine-sensitive Plasmodium falciparum strains

Journal of Inorganic Biochemistry

Volumn 93, Issue 3-4, 2003, Pages 265-270

  Ocheskey, Joseph A ^a   Polyakov, Valery R ^a   Harpstrite, Scott E ^a   Oksman, Anna ^b   Goldberg, Daniel E ^b   Piwnica Worms, David ^a,b   Sharma, Vijay ^a  

^a WASHINGTON UNIVERSITY SCHOOL OF MEDICINE   (United States)

^b WASHINGTON UNIVERSITY SCHOOL OF MEDICINE   (United States)

Author keywords

Chloroquine; Gallium(III); Malaria; Metallo antimalarial; Plasmodium falciparium; Resistance

Indexed keywords

[1,12 BIS(2 HYDROXY 5 METHOXYBENZYL) 1,5,8,12 TETRAAZADODECANE]GALLIUM; ANTIMALARIAL AGENT; BENZYL DERIVATIVE; CHLOROQUINE; GALLIUM; PHENOL DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; COMPLEX FORMATION; CONTROLLED STUDY; DRUG ACTIVITY; DRUG MECHANISM; DRUG SENSITIVITY; DRUG STRUCTURE; DRUG SYNTHESIS; NONHUMAN; PLASMODIUM FALCIPARUM;

AMINES; ANIMALS; ANTIMALARIALS; CHLOROQUINE; CRYSTALLOGRAPHY, X-RAY; DOSE-RESPONSE RELATIONSHIP, DRUG; DRUG RESISTANCE; GALLIUM; LIGANDS; MOLECULAR STRUCTURE; ORGANOMETALLIC COMPOUNDS; PHENOL; PLASMODIUM FALCIPARUM;

PLASMODIUM FALCIPARUM;

EID: 0037439861     PISSN: 01620134     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0162-0134(02)00592-5     Document Type: Article

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