Azalide 3,6-ketals: Antibacterial activity and structure-activity relationships of aryl and hetero aryl substituted analogues

Bioorganic and Medicinal Chemistry Letters

Volumn 13, Issue 7, 2003, Pages 1373-1375

  Sakya, Subas M ^a   Bertinato, Peter ^a   Pratt, Bryan ^a   Suarez Contreras, Melani ^a   Lundy, Kristin M ^a   Minich, Martha L ^a   Cheng, Hengmiao ^a   Ziegler, Carl B ^a   Kamicker, Barbara J ^a   Hayashi, Shigeru F ^a   Santoro, Sheryl L ^a   George, David M ^a   Bertsche, Camilla D ^a  

^a PFIZER INC   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

2 FLUORO 4 BENZYLOXYCARBONYLPHENYL; 2 NITROPHENYL; 2,4 METHOXY 6 PYRIMIDINE; 3 NITRO 2 PYRIDYL; 4 CHLORO 6 PHENYL 2,1,3,5 TRIAZINE; 4 NITROPHENYL; 5 CYANO 2 PYRIDYL; 5 NITRO 2 PYRIDYL; ACETAL DERIVATIVE; ANTIINFECTIVE AGENT; PIPERIDINE DERIVATIVE; UNCLASSIFIED DRUG;

ANIMAL EXPERIMENT; ANIMAL MODEL; ANTIBACTERIAL ACTIVITY; ARTICLE; CONTROLLED STUDY; DRUG POTENCY; DRUG SYNTHESIS; MOUSE; NONHUMAN; PASTEURELLA MULTOCIDA; STAPHYLOCOCCUS AUREUS; STRUCTURE ACTIVITY RELATION;

ANIMALS; ANTI-BACTERIAL AGENTS; CATTLE; CATTLE DISEASES; FEMALE; GONADOTROPIN-RELEASING HORMONE; HETEROCYCLIC COMPOUNDS; MASTITIS, BOVINE; MICE; MICROBIAL SENSITIVITY TESTS; PASTEURELLA MULTOCIDA; PASTEURELLOSIS, PNEUMONIC; STAPHYLOCOCCUS AUREUS; STRUCTURE-ACTIVITY RELATIONSHIP;

PASTEURELLA; PASTEURELLA MULTOCIDA; STAPHYLOCOCCUS; STAPHYLOCOCCUS AUREUS;

EID: 0037424707     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-894X(03)00100-8     Document Type: Article

References (9)

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