Design, synthesis, and structure-activity relationships of substituted piperazinone-based transition state factor Xa inhibitors

Bioorganic and Medicinal Chemistry Letters

Volumn 13, Issue 4, 2003, Pages 729-732

  Su, Ting ^a   Yang, Hua ^a   Volkots, Deborah ^a   Woolfrey, John ^a   Dam, Suiko ^a   Wong, Paul ^a   Sinha, Uma ^a   Scarborough, Robert M ^a   Zhu, Bing Yan ^a  

^a MILLENNIUM PHARMACEUTICALS INC   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

BLOOD CLOTTING FACTOR 10A INHIBITOR; PIPERAZINE DERIVATIVE;

ARTICLE; CRYSTAL STRUCTURE; DRUG DESIGN; DRUG SYNTHESIS; IC 50; STRUCTURE ACTIVITY RELATION;

EID: 0037292995     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-894X(02)01038-7     Document Type: Article

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