A convenient synthesis of 5-(O, O-dialkylphosphoryl)-4-aryl-3,4-dihydropyrimidin-2 (1H)-ones

Heteroatom Chemistry

Volumn 14, Issue 1, 2003, Pages 13-17

  Gong, Denghuang ^a   Zhang, Ling ^a   Yuan, Chengye ^a  

^a SHANGHAI INSTITUTE OF ORGANIC CHEMISTRY   (China)

Author keywords

[No Author keywords available]

Indexed keywords

ALDEHYDES; ALKALI METAL ALLOYS; CATALYSTS; COLUMN CHROMATOGRAPHY; CONDENSATION; INFRARED SPECTROSCOPY; MELTING; QUENCHING; SILICA GEL; SYNTHESIS (CHEMICAL); UREA;

CHEMICAL SHIFTS;

AROMATIC COMPOUNDS;

EID: 0037273986     PISSN: 10427163     EISSN: None     Source Type: Journal    
DOI: 10.1002/hc.10058     Document Type: Article

References (21)

1. Biginelli, P. Gazz Chim Ital 1893, 23, 360.
2. (a) Dondoni, A.; Massi, A. Tetrahedron Lett 2001, 42, 7975;
3. (b) Lu, J.; Bai, Y.; Wang, Z.; Yang, B.; Ma, H. Tetrahedron Lett 2000, 41, 9075;
4. (c) Ma, Y.; Qian, C.; Wang, L.; Yang, M. J Org Chem 2000, 65, 3864;
5. (d) Kappe, C. O. Eur J Med Chem 2000, 35, 1043;
6. (e) Kappe, C. O. Acc Chem Res 2000, 33, 879;
7. (f) Brindaban, C. R.; Alakananda, H.; Umasish, J. J Org Chem 2000, 65, 6270;
8. (g) Hu, E. H.; Sidler, D. R.; Dolling, U. H. J Org Chem 1998, 63, 3454;
9. (h) Kappe, C. O. Tetrahedron 1993, 49, 6937.
10. (a) Atwal, K. S.; Rovnyak, G. C.; Kimball, S. D.; Floyd, D. M.; Moreland, S.; Swanson, B. N.; Gougoutas, J. Z.; Schwartz, J.; Smillie, K. M.; Malley, M. F. J Med Chem 1990, 33, 2629;
11. (b) Atwai, K. S.; Swanson, B. N.; Unger, S. E.; Floyd, D. M.; Moreland, S.; Hedberg, A.; O'Reilly, B. C. J Med Chem 1991, 34, 806.
12. (a) Snider, B. B.; Shi, Z. J Org Chem 1993, 58, 3828;
13. (b) Overman, L. E.; Rabinowitz, M. H.; Renhowe, P. A. J Am Chem Soc 1995, 117, 2657.
14. (a) Snider, B. B.; Busuyek, M. V. J Nat Prod 1999, 62, 1707;
15. (b) Patil, A. D.; Kumar, N. V.; Kokke, W. C.; Bean, M. F.; Freyer, A. J.; Debrosse, C.; Mai, S.; Truneh, A.; Faulkner, D. J.; Carte, B.; Breen, A. L.; Hertzberg, R. P.; Johnson, R. K.; Westley, J. W.; Ports, B. C. M. J Org Chem 1995, 60, 1182;
16. (c) Snider, B.; Chen, J.; Patil, A. D.; Freyer, A. Tetrahedron Lett 1996, 37, 6977;
17. (d) Rama Rao, A. V.; Gurjar, M. K.; Vasudevan, J. J Chem Soc, Chem Commun 1995, 1369.
18. (a) Hutchinson, D. W. Antiviral Res 1985, 5, 193;
19. (b) Sunberg, R. J.; Ebetion, F. H.; Mosher, C. T.; Roof, C. F. CHEMTECH 1991, 21, 304.
20. Kitamura, M.; Tokunaga, M.; Noyari, R.; J Am Chem Soc 1995, 117, 2931.
21. Folkers, K.; Harwood, H.; Johnson, T. B. J Am Chem Soc 1932, 54, 3751.