Autoinhibitory function of the sympathetic prejunctional neuropeptide Y Y2 receptor evidenced by BIIE0246

European Journal of Pharmacology

Volumn 439, Issue 1-3, 2002, Pages 113-119

  Malmström, Rickard E ^a   Lundberg, Jon O N ^a   Weitzberg, Eddie ^b  

^a KAROLINSKA INSTITUTE   (Sweden)

^b KAROLINSKA UNIVERSITY HOSPITAL   (Sweden)

Author keywords

BIIE0246; Neuropeptide Y Y2 receptor; Prejunctional; Sympathetic transmission

Indexed keywords

N [2 [1,2 DIHYDRO 3,5(4H) DIOXO 1,2 DIPHENYL 1,2,4 TRIAZOL 4 YL]ETHYL] N2 [[1 [2 [4 [5,11 DIHYDRO 6(6H) OXODIBENZ[B,E]AZEPIN 11 YL] 1 PIPERAZINYL] 2 OXOETHYL]CYCLOPENTYL]ACETYL]ARGININAMIDE; N2 [[1 [2 [4 (5,11 DIHYDRO 6(6H) OXODIBENZ[B,E]AZEPIN 11 YL) 1 PIPERAZINYL] 2 OXOETHYL]CYCLOPENTYL]ACETYL] N [2 (1,2 DIHYDRO 3,5(4H) DIOXO 1,2 DIPHENYL 3H 1,2,4 TRIAZOL 4 YL)ETHYL]ARGINAMIDE; NEUROPEPTIDE Y; NEUROPEPTIDE Y RECEPTOR ANTAGONIST; NEUROPEPTIDE Y2 RECEPTOR; RESERPINE; UNCLASSIFIED DRUG;

ADRENERGIC TRANSMISSION; ANIMAL EXPERIMENT; ANIMAL TISSUE; ARTICLE; BLOOD VESSEL TONE; CONTROLLED STUDY; ELECTROSTIMULATION; EVOKED RESPONSE; FEMALE; IMMUNOREACTIVITY; KIDNEY; MALE; NERVE CONDUCTION; NERVE TRANSECTION; NEUROTRANSMISSION; NONHUMAN; PRIORITY JOURNAL; SPLEEN; SWINE; SYMPATHETIC NERVE; VASOCONSTRICTION; VASODILATATION;

ANIMALS; ARGININE; BENZAZEPINES; BLOOD FLOW VELOCITY; BLOOD PRESSURE; ELECTRIC STIMULATION; FEMALE; HEART RATE; KIDNEY; MALE; NEUROPEPTIDE Y; RECEPTORS, NEUROPEPTIDE Y; RENAL CIRCULATION; RESERPINE; SPLEEN; SWINE; SYMPATHETIC NERVOUS SYSTEM;

EID: 0037192539     PISSN: 00142999     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0014-2999(02)01371-7     Document Type: Article

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