Halogenated diazirines as photolabel mimics of the inhaled haloalkane anesthetics

Journal of Medicinal Chemistry

Volumn 45, Issue 9, 2002, Pages 1879-1886

  Eckenhoff, Roderic G ^a   Knoll, Frank J ^b   Greenblatt, Eric P ^a   Dailey, William P ^b  

^a UNIVERSITY OF PENNSYLVANIA   (United States)

^b UNIVERSITY OF PENNSYLVANIA   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

1 AZIDO 2 BROMO 2 CHLORO 1,1 DIFLUOROETHANE; 3 (2 BROMO 2 CHLORO 1,1 DIFLUOROETHYL) 3H DIAZIRINE; 3 BROMO 3 (2 CHLORO 1,1,2 TRIFLUOROETHYL) 3H DIAZIRINE; 3 FLUORO 3 (2 CHLORO 1,1,2 TRIFLUOROETHYL) 3H DIAZIRINE; 4 AMINOBUTYRIC ACID A RECEPTOR; COMPLEMENTARY DNA; HALOTHANE; INHALATION ANESTHETIC AGENT; UNCLASSIFIED DRUG;

ANESTHESIA MECHANISM; ANIMAL CELL; ANIMAL EXPERIMENT; ARTICLE; CONCENTRATION RESPONSE; DRUG BINDING SITE; DRUG POTENCY; DRUG SYNTHESIS; HALOGENATION; INHALATION ANESTHESIA; NONHUMAN; OOCYTE; PHOTOAFFINITY LABELING; TADPOLE; XENOPUS;

ANESTHETICS, INHALATION; ANIMALS; CATTLE; CHLORIDE CHANNELS; DIAZOMETHANE; HALOTHANE; HUMANS; HYDROGEN; LARVA; MOLECULAR MIMICRY; MOLECULAR STRUCTURE; OOCYTES; PATCH-CLAMP TECHNIQUES; PHOTOAFFINITY LABELS; PHOTOCHEMISTRY; PROTEIN FOLDING; RECEPTORS, GABA-A; SERUM ALBUMIN; SPECTROMETRY, FLUORESCENCE; TRITIUM; XENOPUS;

EID: 0037171769     PISSN: 00222623     EISSN: None     Source Type: Journal    
DOI: 10.1021/jm0104926     Document Type: Article

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