Synthesis and in vitro pharmacology of substituted quinoline-2,4-dicarboxylic acids as inhibitors of vesicular glutamate transport

Journal of Medicinal Chemistry

Volumn 45, Issue 11, 2002, Pages 2260-2276

  Carrigan, Christina N ^a   Bartlett, Richard D ^a   Esslinger, C Sean ^a   Cybulski, Kimberly A ^a   Tongcharoensirikul, Pakamas ^a   Bridges, Richard J ^a   Thompson, Charles M ^a  

^a UNIVERSITY OF MONTANA   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

ANILINE DERIVATIVE; CARBOXYLIC ACID DERIVATIVE; DICARBOXYLIC ACID DERIVATIVE; DIMETHYL 6 BROMOQUINOLINEDICARBOXYLATE; DIMETHYL KETOGLUTACONATE; GLUTAMATE TRANSPORTER; KETONE DERIVATIVE; PROTON TRANSPORTING ADENOSINE TRIPHOSPHATASE; QUINOLINE 2,4 DICARBOXYLIC ACID DERIVATIVE; QUINOLINE DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; DRUG PROTEIN BINDING; DRUG SYNTHESIS; HYDROLYSIS; IN VITRO STUDY; POLYMERIZATION; STRUCTURE ACTIVITY RELATION; SYNAPSE VESICLE;

ANIMALS; CARRIER PROTEINS; GLUTAMIC ACID; KINETICS; MALE; QUINOLINES; RATS; RATS, SPRAGUE-DAWLEY; STRUCTURE-ACTIVITY RELATIONSHIP; SYNAPTIC VESICLES; TELENCEPHALON;

EID: 0037161590     PISSN: 00222623     EISSN: None     Source Type: Journal    
DOI: 10.1021/jm010261z     Document Type: Article

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