Biarylpropylsulfonamides as novel, potent potentiators of 2-amino-3-(5-methyl-3-hydroxyisoxazol-4-yl)-propanoic acid (AMPA) receptors [1]

Journal of Medicinal Chemistry

Volumn 43, Issue 23, 2000, Pages 4354-4358

  Ornstein, P L ^a   Zimmerman, D M ^a   Arnold, M B ^a   Bleisch, T J ^a   Cantrell, B ^a   Simon, R ^a   Zarrinmayeh, H ^a   Baker, S R ^a   Gates, M ^a   Tizzano, J P ^a   Bleakman, D ^a   Mandelzys, A ^a   Jarvie, K R ^a   Ho, K ^a   Deverill, M ^a   Kamboj, R K ^a  

^a ELI LILLY AND COMPANY   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

2 PYRROLIDONE DERIVATIVE; 6 QUINOXALINECARBOXYLIC ACID PIPERIDIDE; 7 CHLORO 3,4 DIHYDRO 3 METHYL 2H 1,2,4 BENZOTHIADIAZINE 1,1 DIOXIDE; AMPA RECEPTOR; AMPA RECEPTOR AGONIST; ANIRACETAM; BENZAMIDE; CYCLOTHIAZIDE; PIRACETAM; PROPYLSULFONAMIDE DERIVATIVE; UNCLASSIFIED DRUG;

CALCIUM CELL LEVEL; CONCENTRATION RESPONSE; CONTROLLED STUDY; DRUG ACTIVITY; DRUG MECHANISM; DRUG POTENCY; DRUG STRUCTURE; DRUG SYNTHESIS; HUMAN; HUMAN CELL; IN VITRO STUDY; LETTER; STRUCTURE ACTIVITY RELATION;

CELL LINE; HUMANS; RECEPTORS, AMPA; STRUCTURE-ACTIVITY RELATIONSHIP; SULFONAMIDES;

EID: 0034676313     PISSN: 00222623     EISSN: None     Source Type: Journal    
DOI: 10.1021/jm0002836     Document Type: Letter

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