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Bioorganic and Medicinal Chemistry Letters

Volumn 12, Issue 10, 2002, Pages 1331-1334

Structure-based optimisation of 2-aminobenzylstatine derivatives: Potent and selective inhibitors of the chymotrypsin-like activity of the human 20S proteasome

(7) Furet, Pascal a Imbach, Patricia a Fuerst, Peter a Lang, Marc a Noorani, Maria a Zimmermann, Johann a García Echeverría, Carlos a

a NOVARTIS PHARMA AG (Switzerland)

Author keywords

[No Author keywords available]

Indexed keywords

CHYMOTRYPSIN; PROTEASOME; PROTEASOME INHIBITOR; STATINE DERIVATIVE;

ARTICLE; DRUG EFFECT; DRUG IDENTIFICATION; DRUG POTENCY; DRUG SELECTIVITY; DRUG STRUCTURE; DRUG SYNTHESIS; ENZYME ACTIVITY; ENZYME INHIBITION; HUMAN; STRUCTURE ACTIVITY RELATION;

BENZYL COMPOUNDS; CHYMOTRYPSIN; CYSTEINE ENDOPEPTIDASES; DRUG DESIGN; HUMANS; KINETICS; MODELS, MOLECULAR; MOLECULAR CONFORMATION; MULTIENZYME COMPLEXES; PROTEASE INHIBITORS; PROTEASOME ENDOPEPTIDASE COMPLEX; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 0037140857 PISSN: 0960894X EISSN: None Source Type: Journal
DOI: 10.1016/S0960-894X(02)00178-6 Document Type: Article

Times cited : (27)

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* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.