Kinetic analysis of the agonistic and blocking properties of pentobarbital on recombinant rat α1β2γ2S GABAA receptor channels

European Journal of Pharmacology

Volumn 435, Issue 1, 2002, Pages 1-8

  Krampfl, Klaus ^a   Wolfes, Heiner ^a   Dengler, Reinhard ^a   Bufler, Johannes ^a  

^a HANNOVER MEDICAL SCHOOL   (Germany)

Author keywords

Computer simulation; Fast application; GABAA receptor; Pentobarbital

Indexed keywords

4 AMINOBUTYRIC ACID; 4 AMINOBUTYRIC ACID A RECEPTOR; PENTOBARBITAL; RECEPTOR SUBTYPE; RECOMBINANT RECEPTOR;

ARTICLE; CELL LINE; CONTROLLED STUDY; DOSE RESPONSE; DRUG ACTIVITY; DRUG MECHANISM; DRUG RECEPTOR BINDING; ELECTROPHYSIOLOGY; GABAERGIC SYSTEM; HUMAN; HUMAN CELL; ION CURRENT; KINETICS; PRIORITY JOURNAL; PROTEIN EXPRESSION; QUANTITATIVE ANALYSIS; REBOUND; RECEPTOR BLOCKING; REGULATORY MECHANISM;

ANIMALS; CELLS, CULTURED; GABA MODULATORS; HUMANS; KINETICS; PATCH-CLAMP TECHNIQUES; PENTOBARBITAL; RATS; RECEPTORS, GABA-A;

EID: 0037126975     PISSN: 00142999     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0014-2999(01)01558-8     Document Type: Article

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