-
1
-
-
0012621789
-
-
Sainsbury, M., Ed.; Elsevier: Amsterdam
-
For recent reviews on pyrazines see: (a) McCullough, K. L. In Heterocyclic Compounds. Rodd's Chemistry of Carbon Compounds, 2nd ed., 2nd supplement; Sainsbury, M., Ed.; Elsevier: Amsterdam, 2000; Vol. 4, Parts I-J, pp 99-171.
-
(2000)
Heterocyclic Compounds. Rodd's Chemistry of Carbon Compounds, 2nd Ed., 2nd Supplement
, vol.4
, Issue.PARTS I-J
, pp. 99-171
-
-
McCullough, K.L.1
-
2
-
-
0033854165
-
-
(b) Urban, S.; Hickford, S. J. H.; Blunt, J. W.; Munro, M. H. G. Curr. Org. Chem. 2000, 4, 765.
-
(2000)
Curr. Org. Chem.
, vol.4
, pp. 765
-
-
Urban, S.1
Hickford, S.J.H.2
Blunt, J.W.3
Munro, M.H.G.4
-
4
-
-
33750059386
-
-
Katritzky, A. R., Rees, C. W., Boulton, A. J., Eds.; Elsevier: Oxford
-
Sato, N. In Comprehensive Heterocyclic Chemistry II; Katritzky, A. R., Rees, C. W., Boulton, A. J., Eds.; Elsevier: Oxford, 1996; Vol. 6, pp 233-278.
-
(1996)
Comprehensive Heterocyclic Chemistry II
, vol.6
, pp. 233-278
-
-
Sato, N.1
-
5
-
-
0042997346
-
-
For recent contributions see: (a) Gohlke, H.; Gundisch, D.; Schwarz, S.; Seitz, G.; Tilotta, M. C.; Wegge, T. J. Med. Chem. 2002, 45, 1065.
-
(2002)
J. Med. Chem.
, vol.45
, pp. 1065
-
-
Gohlke, H.1
Gundisch, D.2
Schwarz, S.3
Seitz, G.4
Tilotta, M.C.5
Wegge, T.6
-
6
-
-
0001117244
-
-
(b) Ragnarsson, U.; Grehn, L.; Maia, H. L.; Monteiro, L. S. Org. Lett. 2001, 3, 2021.
-
(2001)
Org. Lett.
, vol.3
, pp. 2021
-
-
Ragnarsson, U.1
Grehn, L.2
Maia, H.L.3
Monteiro, L.S.4
-
7
-
-
0035854311
-
-
Liu, W.; Wise, D. S.; Townsend, L. B. J. Org. Chem. 2001, 66, 4783.
-
(2001)
J. Org. Chem.
, vol.66
, pp. 4783
-
-
Liu, W.1
Wise, D.S.2
Townsend, L.B.3
-
8
-
-
0035025587
-
-
Cavalier, J. F.; Burton, M.; Dussart, F.; Marchand, F.; Rees, J. F.; Marchant-Brynaert, J. Bioorg. Med. Chem. 2001, 9, 1037.
-
(2001)
J. Bioorg. Med. Chem.
, vol.9
, pp. 1037
-
-
Cavalier, J.F.1
Burton, M.2
Dussart, F.3
Marchand, F.4
Rees, J.F.5
-
9
-
-
0035375884
-
-
(e) Shibata, K.; Fukuwatari, T.; Sugimoto, E. Biochemistry 2001, 65, 1339.
-
(2001)
Biochemistry
, vol.65
, pp. 1339
-
-
Shibata, K.1
Fukuwatari, T.2
Sugimoto, E.3
-
10
-
-
0033644299
-
-
(a) LaCour, T. G.; Guo, C.; Boyd, M. R.; Fuchs, P. L. Org. Lett. 2000, 2, 33.
-
(2000)
Org. Lett.
, vol.2
, pp. 33
-
-
LaCour, T.G.1
Guo, C.2
Boyd, M.R.3
Fuchs, P.L.4
-
11
-
-
0033844267
-
-
(b) Basler, S.; Brunck, A.; Jautelat, R.; Winterfeldt, E. Helv. Chim. Acta 2000, 83, 1854.
-
(2000)
Helv. Chim. Acta
, vol.83
, pp. 1854
-
-
Basler, S.1
Brunck, A.2
Jautelat, R.3
Winterfeldt, E.4
-
12
-
-
0033530099
-
-
LaCour, T. G.; Guo, C.; Ma, S.; Jeong, J. U.; Boyd, M. R.; Matsunaga, S.; Fusetani, N.; Fuchs, P. L. Bioorg. Med. Chem. Lett. 1999, 9, 2587.
-
(1999)
Bioorg. Med. Chem. Lett.
, vol.9
, pp. 2587
-
-
LaCour, T.G.1
Guo, C.2
Ma, S.3
Jeong, J.U.4
Boyd, M.R.5
Matsunaga, S.6
Fusetani, N.7
Fuchs, P.L.8
-
13
-
-
0029822350
-
-
Guo, C.; Bhandaru, S.; Fuchs, P. L.; Boyd, M. R. J. Am. Chem. Soc. 1996, 118, 10672.
-
(1996)
J. Am. Chem. Soc.
, vol.118
, pp. 10672
-
-
Guo, C.1
Bhandaru, S.2
Fuchs, P.L.3
Boyd, M.R.4
-
14
-
-
0036164484
-
-
(a) Suzuki, Y.; Suzuki, A.; Tamaru, A.; Katsukawa, C.; Oda, H. J. Clin. Microbiol. 2002, 40, 501.
-
(2002)
J. Clin. Microbiol.
, vol.40
, pp. 501
-
-
Suzuki, Y.1
Suzuki, A.2
Tamaru, A.3
Katsukawa, C.4
Oda, H.5
-
15
-
-
0036804084
-
-
(b) Zhang, Y.; Permar, S.; Sun, Z. J. Clin. Microbiol. 2002, 40, 42.
-
(2002)
J. Clin. Microbiol.
, vol.40
, pp. 42
-
-
Zhang, Y.1
Permar, S.2
Sun, Z.3
-
17
-
-
0033834868
-
-
Zimhony, O.; Cox, J. S.; Welch, J. T.; Vilcheze, C.; Jacobs, W. R. Nat. Med. (NY) 2000, 6, 1043.
-
(2000)
Nat. Med. (NY)
, vol.6
, pp. 1043
-
-
Zimhony, O.1
Cox, J.S.2
Welch, J.T.3
Vilcheze, C.4
Jacobs, W.R.5
-
18
-
-
0031941640
-
-
(a) Cynamon, M. H.; Speirs, R. J.; Welch, J. T. Antimicrob. Agents Chemother. 1998, 42, 462.
-
(1998)
Antimicrob. Agents Chemother.
, vol.42
, pp. 462
-
-
Cynamon, M.H.1
Speirs, R.J.2
Welch, J.T.3
-
19
-
-
0029780824
-
-
(b) Bergmann, K. E.; Cynamon, M. H.; Welch, J. T. J. Med. Chem. 1996, 39, 3394.
-
(1996)
J. Med. Chem.
, vol.39
, pp. 3394
-
-
Bergmann, K.E.1
Cynamon, M.H.2
Welch, J.T.3
-
20
-
-
0029069432
-
-
Speirs, R. J.; Welch, J. T.; Cynamon, M. H. Antimicrob. Agents Chemother. 1995, 39, 1269.
-
(1995)
Antimicrob. Agents Chemother.
, vol.39
, pp. 1269
-
-
Speirs, R.J.1
Welch, J.T.2
Cynamon, M.H.3
-
24
-
-
0036340599
-
-
For recent reviews on azirines, see: (a) Palacios, F.; Ochoa de Retana, A. M.; Martinez de Marigorta, E.; de los Santos, J. M. Org. Prep. Proced. Int. 2002, 34, 219-269.
-
(2002)
Org. Prep. Proced. Int.
, vol.34
, pp. 219-269
-
-
Palacios, F.1
Ochoa De Retana, A.M.2
Martinez De Marigorta, E.3
De Los Santos, J.M.4
-
26
-
-
0034950899
-
-
Palacios, F.; Ochoa de Retana, A. M.; Martinez de Marigorta, E.; de los Santos, J. M. Eur. J. Org. Chem. 2001, 2401-2414.
-
(2001)
Eur. J. Org. Chem.
, pp. 2401-2414
-
-
Palacios, F.1
Ochoa De Retana, A.M.2
Martinez De Marigorta, E.3
De Los Santos, J.M.4
-
27
-
-
0034685718
-
-
Palacios, F.; Ochoa de Retana, A. M.; Gil, J. I.; Ezpeleta, J. M. J. Org. Chem. 2000, 65, 3213-3217.
-
(2000)
J. Org. Chem.
, vol.65
, pp. 3213-3217
-
-
Palacios, F.1
Ochoa De Retana, A.M.2
Gil, J.I.3
Ezpeleta, J.M.4
-
28
-
-
0034622355
-
-
Palacios, F.; Ochoa de Retana, A. M.; Gil, J. I. Tetrahedron Lett. 2000, 41, 5363-5366.
-
(2000)
Tetrahedron Lett.
, vol.41
, pp. 5363-5366
-
-
Palacios, F.1
Ochoa De Retana, A.M.2
Gil, J.I.3
-
29
-
-
0033534492
-
The asymmetric synthesis of diethyl 2-phenyl-2H-azirine-3-phosphonate (62%) and the isomeric 3-phenyl-2H-azirine-2-phosphonate (15%) from chiral aziridines has been reported
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The asymmetric synthesis of diethyl 2-phenyl-2H-azirine-3-phosphonate (62%) and the isomeric 3-phenyl-2H-azirine-2-phosphonate (15%) from chiral aziridines has been reported. Davis, F. A.; McCoull, W. Tetrahedron Lett. 1999, 40, 249-252.
-
(1999)
Tetrahedron Lett.
, vol.40
, pp. 249-252
-
-
Davis, F.A.1
McCoull, W.2
-
30
-
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0037149045
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The asymmetric synthesis of dimethyl 2-aryl-2H-azirine-3-phosphonates with a small proportion of the isomeric 3-aryl-2H-azirine-2-phosphonate by Swern oxidation of chiral cis-aziridine phosphonates and the use as a dienophile in cycloaddition reactions of 2H-azirine-3-phosphonates have been recently reported
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The asymmetric synthesis of dimethyl 2-aryl-2H-azirine-3-phosphonates with a small proportion of the isomeric 3-aryl-2H-azirine-2-phosphonate by Swern oxidation of chiral cis-aziridine phosphonates and the use as a dienophile in cycloaddition reactions of 2H-azirine-3-phosphonates have been recently reported. Davis, F. A.; Wu, Y.; Yan, H.; Prasad, K. R.; McCoull, W. Org. Lett. 2002, 4, 655-658.
-
(2002)
Org. Lett.
, vol.4
, pp. 655-658
-
-
Davis, F.A.1
Wu, Y.2
Yan, H.3
Prasad, K.R.4
McCoull, W.5
-
31
-
-
0035077764
-
-
(a) Aurichio, S.; Grassi, S.; Malpezzi, L.; Sartori, A. S.; Truscello, A. M. Eur. J. Org. Chem 2001, 1183-1187.
-
(2001)
Eur. J. Org. Chem
, pp. 1183-1187
-
-
Aurichio, S.1
Grassi, S.2
Malpezzi, L.3
Sartori, A.S.4
Truscello, A.M.5
-
35
-
-
0000247447
-
-
(e) Alper, H.; Prickett, J. E.; Wollwitz, S. J. Am. Chem. Soc. 1977, 99, 4330-4333.
-
(1977)
J. Am. Chem. Soc.
, vol.99
, pp. 4330-4333
-
-
Alper, H.1
Prickett, J.E.2
Wollwitz, S.3
-
37
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0041494730
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note
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2 atmosphere. The crude product was purified by chromatography using silica gel (hexane/ethyl acetate).
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40
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0042496543
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note
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2 atmosphere. The crude product was purified by chromatography using silica gel (hexane/ethyl acetate).
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41
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0042496544
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note
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4, and evaporated under vacuum. The crude product was purified by chromatography using silica gel (hexane/ethyl acetate).
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