Geometry-affinity relationships of the selective serotonin receptor ligand 9-(aminomethyl)-9,10-dihydroanthracene

Journal of Medicinal Chemistry

Volumn 45, Issue 8, 2002, Pages 1656-1664

  Runyon, Scott P ^a   Peddi, Srinivas ^a   Savage, Jason E ^b   Roth, Bryan L ^b   Glennon, Richard A ^a   Westkaemper, Richard B ^a  

^a VIRGINIA COMMONWEALTH UNIVERSITY   (United States)

^b CASE WESTERN RESERVE UNIVERSITY SCHOOL OF MEDICINE   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

9 (AMINOMETHYL) 9,10 DIHYDROANTHRACENE; ANTHRACENE DERIVATIVE; PHENETHYLAMINE; SEROTONIN; SEROTONIN 2 ANTAGONIST; SEROTONIN 2A RECEPTOR; SEROTONIN ANTAGONIST; TRICYCLIC AROMATIC COMPOUND; UNCLASSIFIED DRUG;

ANIMAL CELL; ARTICLE; BINDING AFFINITY; DRUG CONFORMATION; DRUG RECEPTOR BINDING; DRUG SYNTHESIS; GEOMETRY; HYDROGEN BOND; LIGAND BINDING; MOLECULAR MODEL; NONHUMAN; STRUCTURE ACTIVITY RELATION;

3T3 CELLS; ANIMALS; ANTHRACENES; MICE; MODELS, MOLECULAR; MOLECULAR CONFORMATION; RADIOLIGAND ASSAY; RECEPTOR, SEROTONIN, 5-HT2A; RECEPTORS, SEROTONIN; STRUCTURE-ACTIVITY RELATIONSHIP; TRANSFECTION;

EID: 0037061595     PISSN: 00222623     EISSN: None     Source Type: Journal    
DOI: 10.1021/jm010354g     Document Type: Article

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