Analogue based design of MMP-13 (Collagenase-3) inhibitors

Bioorganic and Medicinal Chemistry Letters

Volumn 12, Issue 19, 2002, Pages 2689-2693

  Sarma, J A R P ^a   Rambabu, G ^b   Srikanth, K ^a   Raveendra, D ^c   Vithal, M ^b  

^a GVK BIOSCIENCES PVT LTD   (India)

^b OSMANIA UNIVERSITY   (India)

^c INDIAN INSTITUTE OF CHEMICAL TECHNOLOGY   (India)

Author keywords

[No Author keywords available]

Indexed keywords

COLLAGENASE 3; COLLAGENASE INHIBITOR;

ALGORITHM; ARTICLE; CALCULATION; DRUG DESIGN; ENZYME INHIBITION; IC 50; PREDICTION; QUANTITATIVE STRUCTURE ACTIVITY RELATION; STRUCTURE ANALYSIS; VALIDATION PROCESS;

ALGORITHMS; COLLAGENASES; MATRIX METALLOPROTEINASE 13; MODELS, MOLECULAR; PROTEASE INHIBITORS; PROTEIN CONFORMATION; QUANTITATIVE STRUCTURE-ACTIVITY RELATIONSHIP; RECEPTORS, DRUG; REGRESSION ANALYSIS;

EID: 0037037350     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-894X(02)00559-0     Document Type: Article

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