Dry-media one-pot syntheses of fluorinated-2,3-dihydro-1,5-benzothiazepines under microwave activation

Green Chemistry

Volumn 4, Issue 6, 2002, Pages 599-602

  Dandia, Anshu ^a   Sati, Meha ^a   Loupy, André ^b  

^a UNIVERSITY OF RAJASTHAN   (India)

^b UNIVERSITÉ PARIS SUD   (France)

Author keywords

[No Author keywords available]

Indexed keywords

EID: 0036928550     PISSN: 14639262     EISSN: None     Source Type: Journal    
DOI: 10.1039/b207004a     Document Type: Article

References (53)

1. K. Weiss, P. Fitscha, A. Gazso, D. Gludovacz and H. Sinzinger, Prog. Clin. Biol. Res., 1989,301, 353; Chem. Abstr., 1989,111, 70642v.
2. K. Weiss, P. Fitscha, A. Gazso, D. Gludovacz and H. Sinzinger, Prog. Clin. Biol. Res., 1989, 301, 353; Chem. Abstr., 1989, 111, 70642v.
3. M. Takeda, A. Oishi, H. Nakajima and T. Nagao, (Tanabe Seiyaku Co. Ltd.) Jpn.Kokai Tokyo Koho JP. 61, 1986,103, 828 [86, 103 828] (Cl A61 K31/55), 1986, Appl. 84/225, 030, 1984; Chem. Abstr., 1986, 105, 183965x.
4. M. Takeda, A. Oishi, H. Nakajima and T. Nagao, (Tanabe Seiyaku Co. Ltd.) Jpn.Kokai Tokyo Koho JP. 61, 1986,103, 828 [86, 103 828] (Cl A61 K31/55), 1986, Appl. 84/225, 030, 1984; Chem. Abstr., 1986, 105, 183965x.
5. R. Filler, Chem. Tech., 1974, 4, 752.
6. (a) A. Odawara and T. Ikeo, Jpn. Kokai. Tokkyo. Koho JP. 06, 1994, 183, 978 [94, 183, 978] (Cl. A 61. K 31/55), Appl. 92/341, 753; Chem. Abstr., 1992, 122, 96150c;
7. (a) A. Odawara and T. Ikeo, Jpn. Kokai. Tokkyo. Koho JP. 06, 1994, 183, 978 [94, 183, 978] (Cl. A 61. K 31/55), Appl. 92/341, 753; Chem. Abstr., 1992, 122, 96150c;
8. (b) A. Lochead, J. C. Muller, C. Denys and H. Dumas, Eur. Pat. Appl. EP 1989,338, 892 (C 1 CO7 D 281/10), FR Appl., 88/5, 131, 1988; Chem. Abstr., 1990, 112, 158278m.
9. (b) A. Lochead, J. C. Muller, C. Denys and H. Dumas, Eur. Pat. Appl. EP 1989,338, 892 (C 1 CO7 D 281/10), FR Appl., 88/5, 131, 1988; Chem. Abstr., 1990, 112, 158278m.
10. K. S. Atwal, S. Z. Ahmed, D. M. Floyd, S. Moreland and A. Hedberg, Biorg. Med. Chem. Lett., 1993, 3, 2797.
11. D. M. Floyd, S. D. Kimball, J. Krapcho, J. Das, C. F. Turk, R. V. Mosquin, M. W. Lago, K. J. Duff, V. G. Lee and R. E. White, J. Med. Chem., 1992, 35(4), 756.
12. Y. Inada, M. Tanabe, K. Itoh, H. Sugihara and K. Nishikawa, Jpn., J. Pharmacol., 1988, 48(3), 323; Chem. Abstr., 1989, 110, 539x.
13. Y. Inada, M. Tanabe, K. Itoh, H. Sugihara and K. Nishikawa, Jpn., J. Pharmacol., 1988, 48(3), 323; Chem. Abstr., 1989, 110, 539x.
14. N. K. Ahmed, Can. Pat. Appl., CA2, 030, 159 [C1. A61 K31/55], 1991;US Appl., 441, 083, 1989; Chem. Abstr., 1991, 115, 198515f.
15. N. K. Ahmed, Can. Pat. Appl., CA2, 030, 159 [C1. A61 K31/55], 1991;US Appl., 441, 083, 1989; Chem. Abstr., 1991, 115, 198515f.
16. M. Upreti, S. Pant, A. Dandia and U. C. Pant, Phosphorus, Sulfur Silicon, 1996, 113, 165.
17. W. D. Stephens and L. Field, J. Org. Chem., 1959, 24, 1576.
18. A. Levai and R. Bognar, Acta. Chim. Acad. Sci. Hung., 1976, 88, 293.
19. H. Duddeck, M. Kaiser and A. Levai, Liebigs Ann. Chem., 1985, 869.
20. A. Levai and R. Bognar, Acta. Chim. Acad. Sci. Hung., 1977, 92, 415.
21. W. Reid and W. Marx, Chem. Ber., 1957, 90, 2683.
22. C. H. Hankovszky and K. Hideg, Acta. Chim. Acad. Sci. Hung., 1971, 68, 403.
23. H. Inoue, M. Konda, T. Hoshiyama, H. Otsaka, K. Takashi, M. Gaino, T. Date, K. Aoe, M. Takeda, S. Murata, H. Narita and T. Nagao, J. Med. Chem., 1991, 34, 675.
24. H. Kugita, H. Inoue, M. Ikezaki and S. Takeo, Chem. Pharm. Bull., 1970, 18, 2028.
25. (a) M. Jeselnik, R. S. Varma, S. Polanc and M. Kocevar, Green Chem., 2002, 4, 35;
26. (b) P. Lidström, J. Tierney, B. Wathey and J. Westman, Tetrahedron, 2001, 57, 9225;
27. (c) A. Loupy and L. Perreux, Tetrahedron, 2001, 57, 9199;
28. (d) A. De. LA. Hoz, A. D-Ortis, A. Moreno and F. Langa, Microrev., Eur. J. Org. Chem., 2000, 3659;
29. (e) N. Elander, J. R. Jones, S.-Y. Lu and S. Stone-Elender, Chem. Soc. Rev., 2000, 29, 239;
30. (f) S. Deshayes, M. Liagre, A. Loupy, J. Luche and A. Petit, Tetrahedron, 1999, 55, 10851;
31. (g) R. S. Varma, Green Chem., 1999, 1, 43;
32. (h) A. Loupy, A. Petit, J. Hamelin, F. Texier-Boullet, P. Jacquault and D. Mathe, Synthesis, 1998, 1213.
33. (a) A. Dandia, R. Singh, H. Sachdeva and K. Arya, J. Fluorine Chem., 2001, 111, 61;
34. (b) A. Dandia, H. Sachdeva and R. Singh, J. Chem. Res. (S), 2000, 272;
35. (c) A. Dandia, M. Upreti, B. Rani, U. C. Pant and I. J. Gupta, J. Fluorine Chem., 1998, 91, 171;
36. (d) A. Dandia, M. Saha and H. Taneja, J. Fluorine Chem., 1998, 90, 17;
37. (e) A. Dandia, M. Saha and B. Rani, J. Chem. Res. (S), 1998, 360;
38. (f) U. C. Pant, M. Upreti, S. Pant, A. Dandia, G. K. Patnaik and A. K. Goel, Phosphorus, Sulfur Silicon, 1997, 126, 193;
39. (g) A. Dandia, B. Rani, M. Saha and I. J. Gupta, Phosphorus, Sulfur Silicon, 1997, 130, 217.
40. (a) H. Marquez, A. Plutin, Y. Rodriguez, E. Perez and A. Loupy, Synth. Commun., 2000, 30, 1067;
41. (b) M. Suarez, A. Loupy, E. Salfran, L. Moran and E. Rolando, Heterocycles, 1999, 51, 21;
42. (c) R. Perez, E. Perez, M. Suarez, L. Gonzalez, A. Loupy, M. L. Jimeno and C. Ochoa, Org. Prep. Proced. Int., 1997, 29, 671;
43. (d) M. Suarez, A. Loupy, E. Perez, L. Moran, G. Gerona, A. Morales and M. Autie, Heterocycl. Commun., 1996, 2, 275.
44. B. Perio, M. J. Dozias, P. Jacqualt and J. Hamelin, Tetrahedron Lett., 1997, 38, 7867; K. Toshima, Y. Ushiki, G. Matsuo and S. Matsumara, Tetrahedron Lett., 1997, 38, 7375.
45. B. Perio, M. J. Dozias, P. Jacqualt and J. Hamelin, Tetrahedron Lett., 1997, 38, 7867; K. Toshima, Y. Ushiki, G. Matsuo and S. Matsumara, Tetrahedron Lett., 1997, 38, 7375.
46. (a) B. Syassi, K. Bougrin and M. Soufiaoui, Tetrahedron Lett., 1997, 38, 8855;
47. (b) E. R. Perez, A. L. Marrero, R. Perez and M. A. Autie, Tetrahedron Lett., 1995, 36, 1779;
48. (c) R. S. Varma, M. Varma and A. K. Chatterjee, J. Chem. Soc., Perkin Trans 1, 1993, 999;
49. (d) A. Ben Alloum, B. Labiad and D. Villemin, J. Chem. Soc., Chem. Commun., 1989, 607.
50. (a) R. A. Abramovitch, Org. Prep. Proced. Int., 1991, 23, 685;
51. (b) R. N. Gedye, F. E. Smith and K. C. Westaway, Can. J. Chem., 1988, 66, 17.
52. A. Loupy, L. Perreux, M. Liagre, K. Burle and M. Moneuse, Pure Appl. Chem., 2001, 73, 161.
53. U. C. Pant, B. S. Gaur and M. Chugh, Indian J. Chem., Sect. B, 1987, 26, 947.