메뉴 건너뛰기




Volumn 13, Issue 6, 2002, Pages 1200-1210

Synthesis and biological evaluation of EC20: A new folate-derived, 99mTc-based radiopharmaceutical

Author keywords

[No Author keywords available]

Indexed keywords

MAMMALS; ORGANIC ACIDS; TUMORS;

EID: 0036862058     PISSN: 10431802     EISSN: None     Source Type: Journal    
DOI: 10.1021/bc0200430     Document Type: Article
Times cited : (215)

References (73)
  • 1
    • 0030019317 scopus 로고    scopus 로고
    • 67Ga-deferoxamine-folate, a potential radiopharmaceutical for tumor imaging
    • 67Ga-deferoxamine-folate, a potential radiopharmaceutical for tumor imaging. Bioconjugate Chem. 7, 56-62.
    • (1996) Bioconjugate Chem. , vol.7 , pp. 56-62
    • Wang, S.1
  • 2
    • 0030163022 scopus 로고    scopus 로고
    • Tumor-selective radiopharmaceutical targeting via receptor-mediated endocytosis of Gallium-67-deferoxamine-folate
    • Mathias, C. J., et al. (1996) Tumor-selective radiopharmaceutical targeting via receptor-mediated endocytosis of Gallium-67-deferoxamine-folate. J. Nuc. Med., 37 (6), 1003-1008.
    • (1996) J. Nuc. Med. , vol.37 , Issue.6 , pp. 1003-1008
    • Mathias, C.J.1
  • 3
    • 0031658693 scopus 로고    scopus 로고
    • Indium-111-DTPA-folate as a potential folate-receptor-targeted radiopharmaceutical
    • Mathias, C. J., et al. (1998) Indium-111-DTPA-folate as a potential folate-receptor-targeted radiopharmaceutical. J. Nucl. Med., 39, 1579-1585.
    • (1998) J. Nucl. Med. , vol.39 , pp. 1579-1585
    • Mathias, C.J.1
  • 4
    • 0032216520 scopus 로고    scopus 로고
    • 99mTc-Ethylenedicysteine-folate: A new tumor imaging agent. Synthesis, labeling and evaluation in animals
    • 99mTc-Ethylenedicysteine-folate: A new tumor imaging agent. Synthesis, labeling and evaluation in animals. Cancer Biother. Radiopharm. 13 (6), 427-435.
    • (1998) Cancer Biother. Radiopharm. , vol.13 , Issue.6 , pp. 427-435
    • Ilgan, S.1
  • 5
    • 0032588840 scopus 로고    scopus 로고
    • 99mTc-HYNIC-folate: A novel receptor-based targeted radiopharmaceutical for tumor imaging
    • 99mTc-HYNIC-folate: A novel receptor-based targeted radiopharmaceutical for tumor imaging. J. Nucl. Med. 40 (9), 1563-1569.
    • (1999) J. Nucl. Med. , vol.40 , Issue.9 , pp. 1563-1569
    • Guo, W.1    Hinkle, G.H.2    Lee, R.J.3
  • 6
    • 0001353259 scopus 로고    scopus 로고
    • 99mTc-OXA-Folate show uptake of both isomers in folate-receptor (+) KB cell lines
    • 99mTc-OXA-Folate show uptake of both isomers in folate-receptor (+) KB cell lines. Soc. Nucl. Med. Proc. 47th Annual Meeting 41 (5), 119P.
    • (2000) Soc. Nucl. Med. Proc. 47th Annual Meeting , vol.41 , Issue.5
    • Linder, K.E.1
  • 7
    • 0029328546 scopus 로고
    • Somatostatin receptor imaging of neuroendocrine tumors with indium-111 pentetreotide (Octreoscan)
    • Olsen, J. O., et al. (1995) Somatostatin receptor imaging of neuroendocrine tumors with indium-111 pentetreotide (Octreoscan). Semin. Nucl. Med. 25 (3), 251-61.
    • (1995) Semin. Nucl. Med. , vol.25 , Issue.3 , pp. 251-261
    • Olsen, J.O.1
  • 8
    • 0028047017 scopus 로고
    • Vasoactive intestinal peptide-receptor imaging for the localization of intestinal adenocarcinomas and endocrine tumors
    • Virgolini, I, et al. (1994) Vasoactive intestinal peptide-receptor imaging for the localization of intestinal adenocarcinomas and endocrine tumors. N. Engl. J. Med. 331 (17), 1116-1121.
    • (1994) N. Engl. J. Med. , vol.331 , Issue.17 , pp. 1116-1121
    • Virgolini, I.1
  • 9
    • 0032717783 scopus 로고    scopus 로고
    • 131I-labeled chimeric monoclonal antibody MOv18 in ovarian cancer patients: A pilot study
    • 131I-labeled chimeric monoclonal antibody MOv18 in ovarian cancer patients: A pilot study. Tumor Targeting 4, 179-188.
    • (1999) Tumor Targeting , vol.4 , pp. 179-188
    • Van Zanten-Przybysz, I.1
  • 10
    • 0033032914 scopus 로고    scopus 로고
    • Tumor imaging via indium 111-labeled DTPA-adeno-sylcobalamin
    • Collins, D. A., Hogenkamp, H. P., and Gebhard, M. W. (1999) Tumor imaging via indium 111-labeled DTPA-adeno-sylcobalamin. Mayo Clin. Proc. 74 (7), 687-91.
    • (1999) Mayo Clin. Proc. , vol.74 , Issue.7 , pp. 687-691
    • Collins, D.A.1    Hogenkamp, H.P.2    Gebhard, M.W.3
  • 11
    • 0028010079 scopus 로고
    • Immunoscintigraphy with three step monoclonal pretargeting technique in diagnosis of uveal melanoma: Preliminary results
    • Modorati, G., et al. (1994) Immunoscintigraphy with three step monoclonal pretargeting technique in diagnosis of uveal melanoma: Preliminary results. Br. J. Ophthalmol. 78 (1), 19-23.
    • (1994) Br. J. Ophthalmol. , vol.78 , Issue.1 , pp. 19-23
    • Modorati, G.1
  • 12
    • 45349111034 scopus 로고
    • A simple qualitative determination of human antibodies to murine immunoglobulins (HAMA) in serum samples
    • Seccamani, E., et al. (1989) A simple qualitative determination of human antibodies to murine immunoglobulins (HAMA) in serum samples. Int. J. Radiat. Appl. Instrum. B, 16 (2), 167-170.
    • (1989) Int. J. Radiat. Appl. Instrum. B , vol.16 , Issue.2 , pp. 167-170
    • Seccamani, E.1
  • 13
    • 0025362523 scopus 로고
    • In vivo tumor targeting of a recombinant single-chain antigen-binding protein
    • Colcher, D., et al. (1990) In vivo tumor targeting of a recombinant single-chain antigen-binding protein. J. Natl. Cancer Inst. 82 (14), 1191-1197.
    • (1990) J. Natl. Cancer Inst. , vol.82 , Issue.14 , pp. 1191-1197
    • Colcher, D.1
  • 14
    • 0035135353 scopus 로고    scopus 로고
    • Folate-mediated targeting: From diagnostics to drug and gene delivery
    • Leamon, C. P., Low, P. S. (2001) Folate-mediated targeting: From diagnostics to drug and gene delivery. Drug Discov. Today, 6 (1), 44-51.
    • (2001) Drug Discov. Today , vol.6 , Issue.1 , pp. 44-51
    • Leamon, C.P.1    Low, P.S.2
  • 15
    • 0033976955 scopus 로고    scopus 로고
    • Development of a tumortargeting MR contrast agent using the high-affinity folate receptor
    • Konda, S. D., et al. (2000) Development of a tumortargeting MR contrast agent using the high-affinity folate receptor. Invest. Radiol. 35 (1), 50-57.
    • (2000) Invest. Radiol. , vol.35 , Issue.1 , pp. 50-57
    • Konda, S.D.1
  • 16
    • 0031564203 scopus 로고    scopus 로고
    • Folate-maytansinoids: Targetselective drugs of low molecular weight
    • Ladino, C. A., et al. (1997) Folate-maytansinoids: Targetselective drugs of low molecular weight. Int. J. Cancer 73, 859-864.
    • (1997) Int. J. Cancer , vol.73 , pp. 859-864
    • Ladino, C.A.1
  • 17
    • 0028220371 scopus 로고
    • Inhibition of leukaemia cell proliferation by folic acid-polylysine-mediated introduction of c-myb antisense oligodeoxynucleotides into HL-60 cells
    • Citro, G., et al. (1994) Inhibition of leukaemia cell proliferation by folic acid-polylysine-mediated introduction of c-myb antisense oligodeoxynucleotides into HL-60 cells. Br. J. Cancer 69, 463-467.
    • (1994) Br. J. Cancer , vol.69 , pp. 463-467
    • Citro, G.1
  • 18
    • 0031048069 scopus 로고    scopus 로고
    • Targeted delivery of antisense oligodeoxynucleotides by LPDII
    • Li, S., Huang, L. (1997) Targeted delivery of antisense oligodeoxynucleotides by LPDII. J. Liposome Res. 7 (1), 63-75.
    • (1997) J. Liposome Res. , vol.7 , Issue.1 , pp. 63-75
    • Li, S.1    Huang, L.2
  • 19
    • 0031806033 scopus 로고    scopus 로고
    • Targeted delivery of antisense oligodeoxynucleotides formulated in a novel lipidic vector
    • Li, S., Huang, L. (1998) Targeted delivery of antisense oligodeoxynucleotides formulated in a novel lipidic vector. J. Liposome Res. 8 (2), 239-250.
    • (1998) J. Liposome Res. , vol.8 , Issue.2 , pp. 239-250
    • Li, S.1    Huang, L.2
  • 20
    • 0031683544 scopus 로고    scopus 로고
    • Folate-mediated targeting of antisense oligonucleotides to ovarian cancer cells
    • Li, S., Deshmukh, H. M., and Huang, L. (1998) Folate-mediated targeting of antisense oligonucleotides to ovarian cancer cells. Pharm. Res. 15 (10), 1540-1545.
    • (1998) Pharm. Res. , vol.15 , Issue.10 , pp. 1540-1545
    • Li, S.1    Deshmukh, H.M.2    Huang, L.3
  • 21
    • 0028939524 scopus 로고
    • Multi-unit ribozyme-mediated cleavage of bcr-abl mRNA in myeloid leukemias
    • Leopold, L. H., et al. (1995) Multi-unit ribozyme-mediated cleavage of bcr-abl mRNA in myeloid leukemias. Blood 85 (8), 2162-2170.
    • (1995) Blood , vol.85 , Issue.8 , pp. 2162-2170
    • Leopold, L.H.1
  • 22
    • 0025951931 scopus 로고
    • Delivery of macromolecules into living cells: A method that exploits folate receptor endocytosis
    • Leamon, C. P., Low, P. S. (1991) Delivery of macromolecules into living cells: A method that exploits folate receptor endocytosis. Proc. Natl. Acad. Sci. U.S.A. 88, 5572-5576.
    • (1991) Proc. Natl. Acad. Sci. U.S.A. , vol.88 , pp. 5572-5576
    • Leamon, C.P.1    Low, P.S.2
  • 23
    • 0034128393 scopus 로고    scopus 로고
    • Folic acid targeting of protein conjugates into ascites tumor cells from ovarian cancer patients
    • Ward, C. M., Acheson, N., and Seymour, L. M. (2000) Folic acid targeting of protein conjugates into ascites tumor cells from ovarian cancer patients. J. Drug Targeting 8 (2), 119-123.
    • (2000) J. Drug Targeting , vol.8 , Issue.2 , pp. 119-123
    • Ward, C.M.1    Acheson, N.2    Seymour, L.M.3
  • 24
    • 0032873312 scopus 로고    scopus 로고
    • Folate-targeted enzyme prodrug cancer therapy utilizing penicillin-V amidase and a doxorubicin prodrug
    • Lu, J. Y., et al. (1999) Folate-targeted enzyme prodrug cancer therapy utilizing penicillin-V amidase and a doxorubicin prodrug. J. Drug Targeting 7 (1), 43-53.
    • (1999) J. Drug Targeting , vol.7 , Issue.1 , pp. 43-53
    • Lu, J.Y.1
  • 25
    • 0026496180 scopus 로고
    • Cytotoxicity of momordin-folate conjugates in cultured human cells
    • Leamon, C. P.; Low, P. S. (1992) Cytotoxicity of momordin-folate conjugates in cultured human cells. J. Biol. Chem. 267, 24966-24971.
    • (1992) J. Biol. Chem. , vol.267 , pp. 24966-24971
    • Leamon, C.P.1    Low, P.S.2
  • 26
    • 0027423248 scopus 로고
    • Cytotoxicity of folate-pseudomonas exotoxin conjugates toward tumor cells
    • Leamon, C. P., Pastan, I., and Low, P. S. (1993) Cytotoxicity of folate-pseudomonas exotoxin conjugates toward tumor cells. J. Biol. Chem. 268, 24847-24854.
    • (1993) J. Biol. Chem. , vol.268 , pp. 24847-24854
    • Leamon, C.P.1    Pastan, I.2    Low, P.S.3
  • 27
    • 0028301330 scopus 로고
    • Selective targeting of malignant cells with cytotoxin-folate conjugates
    • Leamon, C. P., Low, P. S. (1994) Selective targeting of malignant cells with cytotoxin-folate conjugates. J. Drug Targeting 2, 101-112.
    • (1994) J. Drug Targeting , vol.2 , pp. 101-112
    • Leamon, C.P.1    Low, P.S.2
  • 28
    • 0029073423 scopus 로고
    • Conjugates of folate and anti-T-cell-receptor antibodies specifically target folate-receptor-positive tumor cells for lysis
    • Kranz, D. M., et al. (1995) Conjugates of folate and anti-T-cell-receptor antibodies specifically target folate-receptor-positive tumor cells for lysis. Proc. Natl. Acad. Sci. U.S.A. 92, 9057-9061.
    • (1995) Proc. Natl. Acad. Sci. U.S.A. , vol.92 , pp. 9057-9061
    • Kranz, D.M.1
  • 29
    • 0031149555 scopus 로고    scopus 로고
    • Single-chain Fv/folate conjugates mediate efficient lysis of folate-receptor-positive tumor cells
    • Cho, B. K., et al. (1997) Single-chain Fv/folate conjugates mediate efficient lysis of folate-receptor-positive tumor cells. Bioconjugate Chem. 8, 338-346.
    • (1997) Bioconjugate Chem. , vol.8 , pp. 338-346
    • Cho, B.K.1
  • 30
    • 0032580490 scopus 로고    scopus 로고
    • Targeting tumor cells with bispecific antibodies and T cells
    • Kranz, D. M., et al. (1998) Targeting tumor cells with bispecific antibodies and T cells. J. Controlled Release 53, 77-84.
    • (1998) J. Controlled Release , vol.53 , pp. 77-84
    • Kranz, D.M.1
  • 31
    • 0032845322 scopus 로고    scopus 로고
    • Bispecific agents target endogenous murine T cells against human tumor xenografts
    • Rund, L. A., et al. (1999) Bispecific agents target endogenous murine T cells against human tumor xenografts. Int. J. Cancer 83, 141-149.
    • (1999) Int. J. Cancer , vol.83 , pp. 141-149
    • Rund, L.A.1
  • 32
    • 0028001056 scopus 로고
    • Delivery of liposomes into cultured KB cells via folate receptor- mediated endocytosis
    • Lee, R. J., Low, P. S. (1994) Delivery of liposomes into cultured KB cells via folate receptor- mediated endocytosis. J. Biol. Chem. 269, 3198-3204.
    • (1994) J. Biol. Chem. , vol.269 , pp. 3198-3204
    • Lee, R.J.1    Low, P.S.2
  • 33
    • 0028794831 scopus 로고
    • Folate-mediated tumor cell targeting of liposome-entrapped doxorubicin in vitro
    • Lee, R. J., Low, P. S. (1995) Folate-mediated tumor cell targeting of liposome-entrapped doxorubicin in vitro. Biochim. Biophys. Acta 1233, 134-144.
    • (1995) Biochim. Biophys. Acta , vol.1233 , pp. 134-144
    • Lee, R.J.1    Low, P.S.2
  • 34
    • 0029975059 scopus 로고    scopus 로고
    • Peptide-mediated release of folate-targeted liposome contents from endosomal compartments
    • Vogel, K., et al. (1996) Peptide-mediated release of folate-targeted liposome contents from endosomal compartments. J. Am. Chem. Soc. 118 (7), 1581-1586.
    • (1996) J. Am. Chem. Soc. , vol.118 , Issue.7 , pp. 1581-1586
    • Vogel, K.1
  • 35
    • 0032508960 scopus 로고    scopus 로고
    • Diplasmenylcholine-folate liposomes: An efficient vehicle for intracellular drug delivery
    • Rui, Y., et al. (1998) Diplasmenylcholine-folate liposomes: An efficient vehicle for intracellular drug delivery. J. Am. Chem. Soc. 120 (44), 11213-11218.
    • (1998) J. Am. Chem. Soc. , vol.120 , Issue.44 , pp. 11213-11218
    • Rui, Y.1
  • 36
    • 0033106119 scopus 로고    scopus 로고
    • Targeting folate receptor with folate linked to extremities of poly (ethylene glycol)-grafted liposomes: In vitro studies
    • Gabizon, A., et al. (1999) Targeting folate receptor with folate linked to extremities of poly (ethylene glycol)-grafted liposomes: In vitro studies. Bioconjugate Chem. 10 (2), 289-98.
    • (1999) Bioconjugate Chem. , vol.10 , Issue.2 , pp. 289-298
    • Gabizon, A.1
  • 37
    • 0028430957 scopus 로고
    • Folate receptor mediated DNA delivery into tumor cells: Potosomal disruption results in enhanced gene expression
    • Gottschalk, S., et al. (1994) Folate receptor mediated DNA delivery into tumor cells: Potosomal disruption results in enhanced gene expression. Gene Ther. 1, 185-191.
    • (1994) Gene Ther. , vol.1 , pp. 185-191
    • Gottschalk, S.1
  • 38
    • 0029360588 scopus 로고
    • Transfection of folate-polylysine DNA complexes: Evidence for lysosomal delivery
    • Mislick, K. A., et al. (1995) Transfection of folate-polylysine DNA complexes: Evidence for lysosomal delivery. Bioconjugate Chem. 6, 512-515.
    • (1995) Bioconjugate Chem. , vol.6 , pp. 512-515
    • Mislick, K.A.1
  • 39
    • 0029907239 scopus 로고    scopus 로고
    • Targeted gene delivery by tropism-modified adenoviral vectors
    • Douglas, J. T., et al. (1996) Targeted gene delivery by tropism-modified adenoviral vectors. Nat. Biotech. 14, 1574-1578.
    • (1996) Nat. Biotech. , vol.14 , pp. 1574-1578
    • Douglas, J.T.1
  • 40
    • 0033230555 scopus 로고    scopus 로고
    • Folate copolymer-mediated transfection of cultured cells
    • Leamon, C. P., Weigl, D., and Hendren, R. W. (1999) Folate copolymer-mediated transfection of cultured cells. Bioconjugate Chem. 10, 947-957.
    • (1999) Bioconjugate Chem. , vol.10 , pp. 947-957
    • Leamon, C.P.1    Weigl, D.2    Hendren, R.W.3
  • 41
    • 3342894973 scopus 로고    scopus 로고
    • Receptor-targeted gene delivery via folate-conjugated polyethylenimine
    • Guo, W., Lee, R. J. (1999) Receptor-targeted gene delivery via folate-conjugated polyethylenimine. PharmSci 1 (4), 19.
    • (1999) PharmSci , vol.1 , Issue.4 , pp. 19
    • Guo, W.1    Lee, R.J.2
  • 42
    • 0032726144 scopus 로고    scopus 로고
    • Optimization of folate-conjugated liposomal vectors for folate receptor-mediated gene therapy
    • Reddy, J. A., et al. (1999) Optimization of folate-conjugated liposomal vectors for folate receptor-mediated gene therapy. J. Pharm. Sci. 88 (11), 1112-1118.
    • (1999) J. Pharm. Sci. , vol.88 , Issue.11 , pp. 1112-1118
    • Reddy, J.A.1
  • 43
    • 0033971786 scopus 로고    scopus 로고
    • Enhanced folate receptor mediated gene therapy using a novel pH-senistive lipid formulation
    • Reddy, J. A., Low, P. S. (2000) Enhanced folate receptor mediated gene therapy using a novel pH-senistive lipid formulation. J. Controlled Release 64, 27-37.
    • (2000) J. Controlled Release , vol.64 , pp. 27-37
    • Reddy, J.A.1    Low, P.S.2
  • 44
    • 0000630588 scopus 로고
    • Imaging of folate receptors with I-125 labeled folate using small animal imaging system built with plastic scintillating optical fibers
    • abstract
    • Antich, P., et al. (1994) Imaging of folate receptors with I-125 labeled folate using small animal imaging system built with plastic scintillating optical fibers. J. Nucl. Med. 35, 222 (abstract).
    • (1994) J. Nucl. Med. , vol.35 , pp. 222
    • Antich, P.1
  • 45
    • 0033625094 scopus 로고    scopus 로고
    • Synthesis of [(99m)Tc]DTPA-folate and its evaluation as a folate-receptor-targeted radiopharmaceutical
    • Mathias, C. J., et al. (2000) Synthesis of [(99m)Tc]DTPA-folate and its evaluation as a folate-receptor-targeted radiopharmaceutical. Bioconjugate Chem. 11 (2), 253-7.
    • (2000) Bioconjugate Chem. , vol.11 , Issue.2 , pp. 253-257
    • Mathias, C.J.1
  • 47
    • 0029118446 scopus 로고
    • Carrier- and receptor-mediated transport of folate antagonists targeting folate-dependent enzymes: Correlates of molecular structure and biological activity
    • Westerhof, G. R., et al. (1995) Carrier- and receptor-mediated transport of folate antagonists targeting folate-dependent enzymes: Correlates of molecular structure and biological activity. Mol. Pharm. 48, 459-471.
    • (1995) Mol. Pharm. , vol.48 , pp. 459-471
    • Westerhof, G.R.1
  • 48
    • 0027280460 scopus 로고
    • Membrane folate-binding proteins are responsible for folate- protein conjugate endocytosis into cultured cells
    • Leamon, C. P., Low, P. S. (1993) Membrane folate-binding proteins are responsible for folate- protein conjugate endocytosis into cultured cells. Biochem. J. 291, 855-860.
    • (1993) Biochem. J. , vol.291 , pp. 855-860
    • Leamon, C.P.1    Low, P.S.2
  • 50
    • 0030111293 scopus 로고    scopus 로고
    • Labeling cyclic glycoprotein IIb/IIIa receptor antagonists with 99mTc by the preformed chelate approach: Effects of chelators on properties of [99mTc]-chelator-peptide conjugates
    • Liu, S., et al. (1996) Labeling cyclic glycoprotein IIb/IIIa receptor antagonists with 99mTc by the preformed chelate approach: Effects of chelators on properties of [99mTc]-chelator-peptide conjugates. Bioconjugate Chem. 7 (2), 196-202.
    • (1996) Bioconjugate Chem. , vol.7 , Issue.2 , pp. 196-202
    • Liu, S.1
  • 51
    • 0029685434 scopus 로고    scopus 로고
    • Labeling a hydrazino nicotinamide-modified cyclic IIb/IIIa receptor antagonist with 99mTc using aminocarboxylates as coligands
    • Liu, S., et al. (1996) Labeling a hydrazino nicotinamide-modified cyclic IIb/IIIa receptor antagonist with 99mTc using aminocarboxylates as coligands. Bioconjugate Chem. 7 (1), 63-71.
    • (1996) Bioconjugate Chem. , vol.7 , Issue.1 , pp. 63-71
    • Liu, S.1
  • 52
    • 0024028846 scopus 로고
    • Approaches to radiolabeling of antibodies for diagnosis and therapy of cancer
    • Fritzberg, A. R., et al. (1988) Approaches to radiolabeling of antibodies for diagnosis and therapy of cancer. Pharm. Res. 5 (6), 325-334.
    • (1988) Pharm. Res. , vol.5 , Issue.6 , pp. 325-334
    • Fritzberg, A.R.1
  • 53
    • 45949128492 scopus 로고
    • The use of diaminodithiol for labeling small molecules with technetium-99m
    • Liang, F. H., Virzi, F., and Hnatowich, D. J. (1987) The use of diaminodithiol for labeling small molecules with technetium-99m. Int. J. Radiat. Appl. Instrum. B 14 (1), 63-67.
    • (1987) Int. J. Radiat. Appl. Instrum. B , vol.14 , Issue.1 , pp. 63-67
    • Liang, F.H.1    Virzi, F.2    Hnatowich, D.J.3
  • 55
    • 0028399009 scopus 로고
    • Bifunctional chelator for facile preparation of neutral technetium complexes
    • Baidoo, K. E., Lever, S. Z., and Scheffel, U., (1994) Bifunctional chelator for facile preparation of neutral technetium complexes. Bioconjugate Chem. 5 (2), 114-118.
    • (1994) Bioconjugate Chem. , vol.5 , Issue.2 , pp. 114-118
    • Baidoo, K.E.1    Lever, S.Z.2    Scheffel, U.3
  • 56
    • 0029921430 scopus 로고    scopus 로고
    • Bifunctional NHS-BAT ester for antibody conjugation and stable technetium-99m labeling: Conjugation chemistry, immunoreactivity and kit formulation
    • Eisenhut, M., et al. (1996) Bifunctional NHS-BAT ester for antibody conjugation and stable technetium-99m labeling: Conjugation chemistry, immunoreactivity and kit formulation. J. Nucl. Med. 37 (2), 362-70.
    • (1996) J. Nucl. Med. , vol.37 , Issue.2 , pp. 362-370
    • Eisenhut, M.1
  • 57
    • 0001743347 scopus 로고    scopus 로고
    • Rhenium (V) and Technetium (V) Oxo complexes of an N (2)N'S peptidic chelator: Evidence of interconversion between the syn and anti conformations
    • Wong, E., et al. (1997) Rhenium (V) and Technetium (V) Oxo complexes of an N (2)N'S peptidic chelator: Evidence of interconversion between the syn and anti conformations. Inorg. Chem. 36 (25), 5799-5808.
    • (1997) Inorg. Chem. , vol.36 , Issue.25 , pp. 5799-5808
    • Wong, E.1
  • 58
    • 0000078975 scopus 로고
    • Synthesis and characterization of neutral MVO (M = technetium, rhenium) aminethiol complexes containing a pendant phenylpiperidine group
    • Francesconi, L. C., et al. (1993) Synthesis and characterization of neutral MVO (M = technetium, rhenium) aminethiol complexes containing a pendant phenylpiperidine group. Inorg. Chem. 32 (14), 3114-3124.
    • (1993) Inorg. Chem. , vol.32 , Issue.14 , pp. 3114-3124
    • Francesconi, L.C.1
  • 59
    • 25344433818 scopus 로고
    • Linking deprotonation and denticity of chelate ligands. Rhenium (V) Oxo analogues of 99mTechnetium radiopharmaceuticals containing N2S2 chelate ligands
    • Marzilli, L. G., et al. (1994) Linking deprotonation and denticity of chelate ligands. Rhenium (V) Oxo analogues of 99mTechnetium radiopharmaceuticals containing N2S2 chelate ligands. Inorg. Chem. 33 (22), 4850-4860.
    • (1994) Inorg. Chem. , vol.33 , Issue.22 , pp. 4850-4860
    • Marzilli, L.G.1
  • 60
    • 0033378420 scopus 로고    scopus 로고
    • Folate-mediated drug delivery: Effect of alternative conjugation chemistry
    • Leamon, C. P., DePrince, R. B., and Hendren, R. W. (1999) Folate-mediated drug delivery: Effect of alternative conjugation chemistry. J. Drug Targeting 7 (3), 157-169.
    • (1999) J. Drug Targeting , vol.7 , Issue.3 , pp. 157-169
    • Leamon, C.P.1    DePrince, R.B.2    Hendren, R.W.3
  • 61
    • 0026652116 scopus 로고
    • The biological chemistry of folate receptors
    • Antony, A. C. (1992) The biological chemistry of folate receptors. Blood 79 (11), 2807-2820.
    • (1992) Blood , vol.79 , Issue.11 , pp. 2807-2820
    • Antony, A.C.1
  • 62
    • 0027130695 scopus 로고
    • The in vivo metabolic stability of dipeptide analogues of the quinazoline antifolate, ICI 198583, in mice
    • Jodrell, D. I., et al. (1993) The in vivo metabolic stability of dipeptide analogues of the quinazoline antifolate, ICI 198583, in mice. Biochem. Pharm. 46 (12), 2229-2234.
    • (1993) Biochem. Pharm. , vol.46 , Issue.12 , pp. 2229-2234
    • Jodrell, D.I.1
  • 63
    • 0031871186 scopus 로고    scopus 로고
    • 111In]In-DTPA-Folate, a folate-receptor-targeted radiopharmaceutical
    • 111In]In-DTPA-Folate, a folate-receptor-targeted radiopharmaceutical. Nuc. Med. Biol. 25, 585-587.
    • (1998) Nuc. Med. Biol. , vol.25 , pp. 585-587
    • Mathias, C.J.1    Green, M.A.2
  • 64
    • 0026329982 scopus 로고
    • Cloning of a tumor-associated antigen: MOv18 and MOv19 antibodies recognize a folate-binding protein
    • Coney, L. R., et al. (1991) Cloning of a tumor-associated antigen: MOv18 and MOv19 antibodies recognize a folate-binding protein. Cancer Res. 51, 6125-6132.
    • (1991) Cancer Res. , vol.51 , pp. 6125-6132
    • Coney, L.R.1
  • 65
    • 0026752798 scopus 로고
    • Distribution of the folate receptor GP38 in normal and malignant cell lines and tissues
    • Weitman, S. D., et al. (1992) Distribution of the folate receptor GP38 in normal and malignant cell lines and tissues. Cancer Res. 52, 3396-3401.
    • (1992) Cancer Res. , vol.52 , pp. 3396-3401
    • Weitman, S.D.1
  • 66
    • 0028301752 scopus 로고
    • Differential regulation of folate receptor isoforms in normal and malignant tissues in vivo and in established cell lines
    • Ross, J. F., Chaudhuri, P. K., and Ratnam, M. (1994) Differential regulation of folate receptor isoforms in normal and malignant tissues in vivo and in established cell lines. Cancer 73, 2432-2443.
    • (1994) Cancer , vol.73 , pp. 2432-2443
    • Ross, J.F.1    Chaudhuri, P.K.2    Ratnam, M.3
  • 67
    • 0026476410 scopus 로고
    • Cellular localization of the folate receptor: Potential role in drug toxicity and folate homeostasis
    • Weitman, S. D., et al. (1992) Cellular localization of the folate receptor: Potential role in drug toxicity and folate homeostasis. Cancer Research 52, 6708-6711.
    • (1992) Cancer Research , vol.52 , pp. 6708-6711
    • Weitman, S.D.1
  • 68
    • 0028148692 scopus 로고
    • The folate receptor in central nervous system malignancies of childhood
    • Weitman, S. D., Frazier, K. M., and Kamen, B. A. (1994) The folate receptor in central nervous system malignancies of childhood. J. Neurol. Oncol. 21, 107.
    • (1994) J. Neurol. Oncol. , vol.21 , pp. 107
    • Weitman, S.D.1    Frazier, K.M.2    Kamen, B.A.3
  • 69
    • 0025055061 scopus 로고
    • Patterns of antigen distribution in human carcinomas
    • Mattes, M. J., et al. (1990) Patterns of antigen distribution in human carcinomas. Cancer Res. Suppl. 50, 880S.
    • (1990) Cancer Res. Suppl. , vol.50
    • Mattes, M.J.1
  • 70
    • 0027406702 scopus 로고
    • Trophoblast and ovarian cancer antigen LK26
    • Garin-Chesa, P., et al. (1993) Trophoblast and ovarian cancer antigen LK26. Am. J. Pathol. 142 (2), 557-567.
    • (1993) Am. J. Pathol. , vol.142 , Issue.2 , pp. 557-567
    • Garin-Chesa, P.1
  • 71
    • 0030910859 scopus 로고    scopus 로고
    • Overexpression of folate binding protein in ovarian cancers
    • Toffoli, G., et al. (1997) Overexpression of folate binding protein in ovarian cancers. Int. J. Cancer 74, 193-198.
    • (1997) Int. J. Cancer , vol.74 , pp. 193-198
    • Toffoli, G.1
  • 72
    • 0026049546 scopus 로고
    • High-affinity folate binding in human choroid plexus
    • Holm, J., et al. (1991) High-affinity folate binding in human choroid plexus. Biochem. J. 280, 267-271.
    • (1991) Biochem. J. , vol.280 , pp. 267-271
    • Holm, J.1


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.