1,4-Benzothiazine and 1,4-Benzoxazine imidazole derivatives with antifungal activity: A docking study

Bioorganic and Medicinal Chemistry

Volumn 10, Issue 11, 2002, Pages 3415-3423

  Macchiarulo, Antonio ^a   Costantino, Gabriele ^a   Fringuelli, Daniele ^a   Vecchiarelli, Anna ^a   Schiaffella, Fausto ^a   Fringuelli, Renata ^a  

^a UNIVERSITY OF PERUGIA   (Italy)

Author keywords

[No Author keywords available]

Indexed keywords

BENZOTHIAZINE DERIVATIVE; BENZOXAZINE DERIVATIVE; CYTOCHROME P450; FLUCONAZOLE; FUNGAL ENZYME; IMIDAZOLE DERIVATIVE;

ANTIFUNGAL ACTIVITY; ARTICLE; CANDIDA ALBICANS; CRYSTAL STRUCTURE; DRUG PROTEIN BINDING; MOLECULAR MODEL; MYCOBACTERIUM TUBERCULOSIS; SEQUENCE HOMOLOGY;

AMINO ACID SEQUENCE; ANTIFUNGAL AGENTS; BACTERIAL PROTEINS; CANDIDA ALBICANS; CYTOCHROME P-450 ENZYME SYSTEM; ENZYME INHIBITORS; FUNGAL PROTEINS; FUNGI; IMIDAZOLES; ISOMERISM; MODELS, BIOLOGICAL; MODELS, MOLECULAR; MOLECULAR CONFORMATION; MOLECULAR SEQUENCE DATA; MYCOBACTERIUM; SEQUENCE HOMOLOGY; THIAZINES;

CANDIDA; CANDIDA ALBICANS; MURINAE; MYCOBACTERIUM; MYCOBACTERIUM TUBERCULOSIS;

EID: 0036836970     PISSN: 09680896     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0968-0896(02)00263-8     Document Type: Article

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