Synthesis and antifungal activity of new imidazole derivatives of 1,4- benzothiazine

Medicinal Chemistry Research

Volumn 9, Issue 5, 1999, Pages 291-305

  Schiaffella, Fausto ^a   Guarraci, Alessia ^a   Fringuelli, Renata ^a   Pitzurra, Lucia ^a   Bistoni, Francesco ^a   Vecchiarelli, Anna ^a  

^a UNIVERSITY OF PERUGIA   (Italy)

Author keywords

[No Author keywords available]

Indexed keywords

BENZOTHIAZINE DERIVATIVE; FLUCONAZOLE; IMIDAZOLE DERIVATIVE; PYRROLE DERIVATIVE;

ANIMAL EXPERIMENT; ANIMAL MODEL; ANTIFUNGAL ACTIVITY; ARTICLE; CANDIDA ALBICANS; CANDIDIASIS; CONTROLLED STUDY; DRUG STRUCTURE; DRUG SYNTHESIS; IMMUNOPOTENTIATION; MOUSE; NONHUMAN; STRUCTURE ACTIVITY RELATION; SURVIVAL;

EID: 0032732619     PISSN: 10542523     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article

References (23)

1. st International Conference on Chemistry of Antibiotics and Related Microbial Products, Bologna, Italy, September, 1998. PC15
2. Schroter, G. P. J.; Hoelscher, M.; Putman, C. W.; Porter, K. A.; Starzl, T. E. Ann. Surg. 1977, 186, 115-122.
3. Beck-Sague, C.; Jarvis, W. R. J. Infect. Dis. 1993, 167, 1247-1251.
4. Bodey, G. P. J. Chronic Dis. 1996, 19, 667-687.
5. Georgopapadakou, N. H.; Walsh, T. J. Antimicrob. Agents Chemother. 1996, 40, 279-291.
6. White, T. C.; Marr, K. A.; Bowden, R. A. Clin. Microbiol. Rev. 1998, 11, 382-402.
7. Sheehan, D. J.; Hitchcock, A. C.; Sibley, C. M. Clin. Microbiol. Rev. 1999, 12, 40-79.
8. Kauffman, C. A.; Carver, P. L. Drugs 1997, 53, 539-549.
9. Fromtling, R. A. Clin. Microbiol. Rev. 1998, 1, 187-219.
10. Fringuelli, R.; Schiaffella, F.; Bistoni, F.; Pitzurra, L.; Vecchiarelli, A. Bioorg. Med. Chem. 1998, 6, 103-108.
11. Pitzurra, L.; Fringuelli, R.; Perito, S.; Schiaffella, F.; Barluzzi, R.; Bistoni, F.; Vecchiarelli, A.; Antimicrob. Agents Chemother. in press.
12. National Committee for Clinical Laboratory Standards. Reference method for broth dilution antifungal susceptibility testing for yeasts; approved standard. NCCLS Document M27-A, 1997.
13. Anaissie, E. J.; Karyotakis, N. C.; Hachem, R.; Dignani, M. C.; Rex, J. H.; Paetznick, V. L. J. Infect. Dis. 1994, 170, 384-389.
14. Rex, J. H.; Galgiani, J. N.; Bartlett, M. S.; Espinel-Ingroff, A.; Ghannoum, M. A.; Lancaster, M.; Odds, F. C.; Rinaldi, M. G.; Barry, A. L.; Subcommittee on Antifungal Susceptibility Testing of the National Committee for Clinical Laboratory Standards Clin. Infect. Dis., 1997, 24, 235-247.
15. Rex, J. H.; Nelson, P. W.; Paetznick V. L.; Lozano-Chin, M.; Espaniel-Ingroff, A.; Anaissie, E. J. Antimicrob. Agents Chemother. 1998, 42, 129-134.
16. Vecchiarelli, A.; Mazzolla, R.; Farinelli, S.; Cassone, A.; Bistoni, F. J. Gen. Microbiol. 1983, 134, 2583-2592.
17. SRC-LOGKOW for Microsoft Windows. Copyright [c] W. Meylan, 1993-1999.
18. Ricci, A.; Cagnoli, N. Ann. Chim. 1955, 45, 172-179.
19. Cecchetti, V.; Fringuelli, R.; Schiaffella, F.; Fravolini, A.; Bruni, G.; Fiaschi, A.I.; Segre, G. Eur. J. Med. Chem. 1989, 24, 479-484.
20. Shridhar, D. R.; Reddy Sastri, C. V.; Bansal, O. P.; Singh, P. P.; Tripathi, R. M.; Seshagiri Rao, C.; Junnarkar, A.Y. Indian J. Med. 1983, 22B, 1236-1242.
21. van Uden, N.; Buckley, H. In The Yeasts: A Taxonomic Study. Candida Berkhout; Lodder J. Editor; North Holland: Amsterdam, 1970, 914.
22. Vecchiarelli, A.; Cenci, E.; Marconi, P.; Rossi, R.; Riccardi, C.; Bistoni, F. J. Med. Microbiol. 1989, 30, 183-192.
23. Norman, G.R.; Streiner, D.L. In PDQ Statistics; Decker B. C. Inc., Toronto, Ontario, Canada, 1986, 79-92.